DE69712745T2 - Pyrrolopyrimidinen und verfahren zu deren herstellung - Google Patents

Pyrrolopyrimidinen und verfahren zu deren herstellung

Info

Publication number
DE69712745T2
DE69712745T2 DE69712745T DE69712745T DE69712745T2 DE 69712745 T2 DE69712745 T2 DE 69712745T2 DE 69712745 T DE69712745 T DE 69712745T DE 69712745 T DE69712745 T DE 69712745T DE 69712745 T2 DE69712745 T2 DE 69712745T2
Authority
DE
Germany
Prior art keywords
formula
substituted
dilower
alkyl
lower alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69712745T
Other languages
German (de)
English (en)
Other versions
DE69712745D1 (de
Inventor
Guido Bold
Joerg Frei
Peter Traxler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis Pharma GmbH Austria
Novartis AG
Original Assignee
Novartis Erfindungen Verwaltungs GmbH
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Erfindungen Verwaltungs GmbH, Novartis AG filed Critical Novartis Erfindungen Verwaltungs GmbH
Publication of DE69712745D1 publication Critical patent/DE69712745D1/de
Application granted granted Critical
Publication of DE69712745T2 publication Critical patent/DE69712745T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DE69712745T 1996-01-23 1997-01-13 Pyrrolopyrimidinen und verfahren zu deren herstellung Expired - Lifetime DE69712745T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH17596 1996-01-23
PCT/EP1997/000127 WO1997027199A1 (en) 1996-01-23 1997-01-13 Pyrrolopyrimidines and processes for their preparation

Publications (2)

Publication Number Publication Date
DE69712745D1 DE69712745D1 (de) 2002-06-27
DE69712745T2 true DE69712745T2 (de) 2002-10-31

Family

ID=4180979

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69712745T Expired - Lifetime DE69712745T2 (de) 1996-01-23 1997-01-13 Pyrrolopyrimidinen und verfahren zu deren herstellung

Country Status (9)

Country Link
US (1) US6140317A (enExample)
EP (1) EP0888349B1 (enExample)
JP (1) JP4275733B2 (enExample)
AT (1) ATE217873T1 (enExample)
AU (1) AU1441497A (enExample)
DE (1) DE69712745T2 (enExample)
ES (1) ES2177925T3 (enExample)
PT (1) PT888349E (enExample)
WO (1) WO1997027199A1 (enExample)

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DE69712745D1 (de) 2002-06-27
US6140317A (en) 2000-10-31
ATE217873T1 (de) 2002-06-15
EP0888349A1 (en) 1999-01-07
AU1441497A (en) 1997-08-20
ES2177925T3 (es) 2002-12-16
JP2000503005A (ja) 2000-03-14
WO1997027199A1 (en) 1997-07-31
JP4275733B2 (ja) 2009-06-10
EP0888349B1 (en) 2002-05-22

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