DE69622715T2 - Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin-carbonsäure - Google Patents

Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin-carbonsäure

Info

Publication number
DE69622715T2
DE69622715T2 DE69622715T DE69622715T DE69622715T2 DE 69622715 T2 DE69622715 T2 DE 69622715T2 DE 69622715 T DE69622715 T DE 69622715T DE 69622715 T DE69622715 T DE 69622715T DE 69622715 T2 DE69622715 T2 DE 69622715T2
Authority
DE
Germany
Prior art keywords
pct
azabizylo
naphtyridine
peptide
carbonic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69622715T
Other languages
English (en)
Other versions
DE69622715D1 (de
Inventor
F Braish
J Castaldi
A Watson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of DE69622715D1 publication Critical patent/DE69622715D1/de
Application granted granted Critical
Publication of DE69622715T2 publication Critical patent/DE69622715T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
DE69622715T 1995-06-15 1996-03-27 Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin-carbonsäure Expired - Fee Related DE69622715T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49082795A 1995-06-15 1995-06-15
PCT/IB1996/000257 WO1997000268A1 (en) 1995-06-15 1996-03-27 Process for preparing derivatives of azabicyclo naphthyridine carboxylic acid comprising a dipeptide

Publications (2)

Publication Number Publication Date
DE69622715D1 DE69622715D1 (de) 2002-09-05
DE69622715T2 true DE69622715T2 (de) 2002-11-14

Family

ID=23949631

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69622715T Expired - Fee Related DE69622715T2 (de) 1995-06-15 1996-03-27 Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin-carbonsäure

Country Status (10)

Country Link
US (1) US5939550A (de)
EP (1) EP0833837B1 (de)
JP (1) JP3029293B2 (de)
AT (1) ATE221544T1 (de)
CA (1) CA2224616C (de)
DE (1) DE69622715T2 (de)
DK (1) DK0833837T3 (de)
ES (1) ES2178701T3 (de)
PT (1) PT833837E (de)
WO (1) WO1997000268A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (es) * 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
GB0310593D0 (en) * 2003-05-08 2003-06-11 Leuven K U Res & Dev Peptidic prodrugs
CN101500564B (zh) * 2006-03-07 2012-07-25 沃克哈特有限公司 苯并喹嗪-2-羧酸的前药
GB202104712D0 (en) 2021-04-01 2021-05-19 Riedewald Frank Process and system for the recycling of composite materials, mixed and pure waste plastics.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
WO1991002526A1 (en) * 1989-08-16 1991-03-07 Pfizer Inc. Azabicyclo quinolone carboxylic acids

Also Published As

Publication number Publication date
DE69622715D1 (de) 2002-09-05
CA2224616C (en) 2000-05-02
EP0833837A1 (de) 1998-04-08
WO1997000268A1 (en) 1997-01-03
US5939550A (en) 1999-08-17
JP3029293B2 (ja) 2000-04-04
ES2178701T3 (es) 2003-01-01
ATE221544T1 (de) 2002-08-15
DK0833837T3 (da) 2002-09-02
EP0833837B1 (de) 2002-07-31
PT833837E (pt) 2002-11-29
JPH10511983A (ja) 1998-11-17
CA2224616A1 (en) 1997-01-03

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee