DK0833837T3 - Fremgangsmåde til fremstilling af derivater af azabicyclonaphthydridincarboxylsyre omfattende et dipeptid - Google Patents

Fremgangsmåde til fremstilling af derivater af azabicyclonaphthydridincarboxylsyre omfattende et dipeptid

Info

Publication number
DK0833837T3
DK0833837T3 DK96904996T DK96904996T DK0833837T3 DK 0833837 T3 DK0833837 T3 DK 0833837T3 DK 96904996 T DK96904996 T DK 96904996T DK 96904996 T DK96904996 T DK 96904996T DK 0833837 T3 DK0833837 T3 DK 0833837T3
Authority
DK
Denmark
Prior art keywords
pct
carboxylic acid
dipeptide
azabicyclonaphthydridine
derivatives
Prior art date
Application number
DK96904996T
Other languages
English (en)
Inventor
Harry A Watson Jr
Tamim F Braish
Michael J Castaldi
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0833837T3 publication Critical patent/DK0833837T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK96904996T 1995-06-15 1996-03-27 Fremgangsmåde til fremstilling af derivater af azabicyclonaphthydridincarboxylsyre omfattende et dipeptid DK0833837T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49082795A 1995-06-15 1995-06-15
PCT/IB1996/000257 WO1997000268A1 (en) 1995-06-15 1996-03-27 Process for preparing derivatives of azabicyclo naphthyridine carboxylic acid comprising a dipeptide

Publications (1)

Publication Number Publication Date
DK0833837T3 true DK0833837T3 (da) 2002-09-02

Family

ID=23949631

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96904996T DK0833837T3 (da) 1995-06-15 1996-03-27 Fremgangsmåde til fremstilling af derivater af azabicyclonaphthydridincarboxylsyre omfattende et dipeptid

Country Status (10)

Country Link
US (1) US5939550A (da)
EP (1) EP0833837B1 (da)
JP (1) JP3029293B2 (da)
AT (1) ATE221544T1 (da)
CA (1) CA2224616C (da)
DE (1) DE69622715T2 (da)
DK (1) DK0833837T3 (da)
ES (1) ES2178701T3 (da)
PT (1) PT833837E (da)
WO (1) WO1997000268A1 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (es) * 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
GB0310593D0 (en) * 2003-05-08 2003-06-11 Leuven K U Res & Dev Peptidic prodrugs
ES2393802T3 (es) * 2006-03-07 2012-12-28 Wockhardt Limited Profármacos del ácido benzoquinolizin-2-carboxílico
GB202104712D0 (en) 2021-04-01 2021-05-19 Riedewald Frank Process and system for the recycling of composite materials, mixed and pure waste plastics.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
RU2049777C1 (ru) * 1989-08-16 1995-12-10 Пфайзер Инк. Азабицикло-хинолон-карбоновые кислоты или их фармацевтически приемлемые кислотно-аддитивные соли и промежуточные продукты для их получения

Also Published As

Publication number Publication date
DE69622715T2 (de) 2002-11-14
CA2224616C (en) 2000-05-02
ATE221544T1 (de) 2002-08-15
DE69622715D1 (de) 2002-09-05
JP3029293B2 (ja) 2000-04-04
ES2178701T3 (es) 2003-01-01
EP0833837A1 (en) 1998-04-08
JPH10511983A (ja) 1998-11-17
PT833837E (pt) 2002-11-29
WO1997000268A1 (en) 1997-01-03
CA2224616A1 (en) 1997-01-03
EP0833837B1 (en) 2002-07-31
US5939550A (en) 1999-08-17

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