ATE221544T1 - Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin- carbonsäure - Google Patents

Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin- carbonsäure

Info

Publication number
ATE221544T1
ATE221544T1 AT96904996T AT96904996T ATE221544T1 AT E221544 T1 ATE221544 T1 AT E221544T1 AT 96904996 T AT96904996 T AT 96904996T AT 96904996 T AT96904996 T AT 96904996T AT E221544 T1 ATE221544 T1 AT E221544T1
Authority
AT
Austria
Prior art keywords
carboxylic acid
pct
azabizylo
naphtyridine
peptide
Prior art date
Application number
AT96904996T
Other languages
English (en)
Inventor
Tamim F Braish
Michael J Castaldi
Harry A Watson Jr
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE221544T1 publication Critical patent/ATE221544T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT96904996T 1995-06-15 1996-03-27 Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin- carbonsäure ATE221544T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49082795A 1995-06-15 1995-06-15
PCT/IB1996/000257 WO1997000268A1 (en) 1995-06-15 1996-03-27 Process for preparing derivatives of azabicyclo naphthyridine carboxylic acid comprising a dipeptide

Publications (1)

Publication Number Publication Date
ATE221544T1 true ATE221544T1 (de) 2002-08-15

Family

ID=23949631

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96904996T ATE221544T1 (de) 1995-06-15 1996-03-27 Verfahren zur herstellung von derivaten der ein peptid enthaltenden azabizylo-naphtyridin- carbonsäure

Country Status (10)

Country Link
US (1) US5939550A (de)
EP (1) EP0833837B1 (de)
JP (1) JP3029293B2 (de)
AT (1) ATE221544T1 (de)
CA (1) CA2224616C (de)
DE (1) DE69622715T2 (de)
DK (1) DK0833837T3 (de)
ES (1) ES2178701T3 (de)
PT (1) PT833837E (de)
WO (1) WO1997000268A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000106A (es) 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
US7019142B2 (en) * 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
GB0310593D0 (en) * 2003-05-08 2003-06-11 Leuven K U Res & Dev Peptidic prodrugs
WO2007102061A2 (en) * 2006-03-07 2007-09-13 Wockhardt Ltd Prodrugs of benzoquinolizine-2-carboxylic acid
GB202104712D0 (en) 2021-04-01 2021-05-19 Riedewald Frank Process and system for the recycling of composite materials, mixed and pure waste plastics.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids
WO1991002526A1 (en) * 1989-08-16 1991-03-07 Pfizer Inc. Azabicyclo quinolone carboxylic acids

Also Published As

Publication number Publication date
DE69622715D1 (de) 2002-09-05
EP0833837B1 (de) 2002-07-31
US5939550A (en) 1999-08-17
CA2224616A1 (en) 1997-01-03
DK0833837T3 (da) 2002-09-02
JPH10511983A (ja) 1998-11-17
CA2224616C (en) 2000-05-02
WO1997000268A1 (en) 1997-01-03
ES2178701T3 (es) 2003-01-01
EP0833837A1 (de) 1998-04-08
JP3029293B2 (ja) 2000-04-04
PT833837E (pt) 2002-11-29
DE69622715T2 (de) 2002-11-14

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