DE60316013T2 - Heteroaryl-pyrimidinderivate als jak-inhibitoren - Google Patents
Heteroaryl-pyrimidinderivate als jak-inhibitoren Download PDFInfo
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- DE60316013T2 DE60316013T2 DE60316013T DE60316013T DE60316013T2 DE 60316013 T2 DE60316013 T2 DE 60316013T2 DE 60316013 T DE60316013 T DE 60316013T DE 60316013 T DE60316013 T DE 60316013T DE 60316013 T2 DE60316013 T2 DE 60316013T2
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US42357902P | 2002-11-04 | 2002-11-04 | |
| US423579P | 2002-11-04 | ||
| PCT/US2003/035163 WO2004041814A1 (en) | 2002-11-04 | 2003-11-04 | Heteroaryl-pyramidine derivatives as jak inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60316013D1 DE60316013D1 (de) | 2007-10-11 |
| DE60316013T2 true DE60316013T2 (de) | 2008-05-29 |
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| DE60316013T Expired - Lifetime DE60316013T2 (de) | 2002-11-04 | 2003-11-04 | Heteroaryl-pyrimidinderivate als jak-inhibitoren |
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| US (1) | US7259161B2 (enExample) |
| EP (1) | EP1562938B1 (enExample) |
| JP (2) | JP4688498B2 (enExample) |
| AT (1) | ATE371656T1 (enExample) |
| AU (1) | AU2003295396B2 (enExample) |
| CA (1) | CA2506773A1 (enExample) |
| DE (1) | DE60316013T2 (enExample) |
| ES (1) | ES2289349T3 (enExample) |
| WO (1) | WO2004041814A1 (enExample) |
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| RU2485106C2 (ru) | 2005-06-08 | 2013-06-20 | Райджел Фамэсьютикэлз, Инк. | Соединения, проявляющие активность в отношении jak-киназы (варианты), способ лечения заболеваний, опосредованных jak-киназой, способ ингибирования активности jak-киназы (варианты), фармацевтическая композиция на основе указанных соединений |
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| GB9523675D0 (en) * | 1995-11-20 | 1996-01-24 | Celltech Therapeutics Ltd | Chemical compounds |
| CN1438890A (zh) * | 2000-02-25 | 2003-08-27 | 弗·哈夫曼-拉罗切有限公司 | 腺苷受体调制剂 |
| CN100506801C (zh) * | 2000-09-06 | 2009-07-01 | 诺华疫苗和诊断公司 | 糖元合成酶激酶3的抑制剂 |
| CA2441733A1 (en) * | 2001-03-29 | 2002-10-10 | Vertex Pharmaceuticals Incorporated | Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases |
| JP2005500261A (ja) * | 2001-04-10 | 2005-01-06 | バーテックス ファーマシューティカルズ インコーポレイテッド | Ｓｒｃおよび他のプロテインキナーゼのインヒビターとしてのイソキサゾール誘導体 |
| EP1399440B1 (en) * | 2001-06-15 | 2009-06-03 | Vertex Pharmaceuticals Incorporated | 5-(2-aminopyrimidin-4-yl)benzisoxazoles as protein kinase inhibitors |
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2003
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- 2003-11-04 CA CA002506773A patent/CA2506773A1/en not_active Abandoned
- 2003-11-04 AU AU2003295396A patent/AU2003295396B2/en not_active Ceased
- 2003-11-04 ES ES03786582T patent/ES2289349T3/es not_active Expired - Lifetime
- 2003-11-04 DE DE60316013T patent/DE60316013T2/de not_active Expired - Lifetime
- 2003-11-04 JP JP2004550483A patent/JP4688498B2/ja not_active Expired - Fee Related
- 2003-11-04 EP EP03786582A patent/EP1562938B1/en not_active Expired - Lifetime
- 2003-11-04 AT AT03786582T patent/ATE371656T1/de not_active IP Right Cessation
- 2003-11-04 WO PCT/US2003/035163 patent/WO2004041814A1/en not_active Ceased
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2010
- 2010-09-21 JP JP2010211038A patent/JP2011016839A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP4688498B2 (ja) | 2011-05-25 |
| DE60316013D1 (de) | 2007-10-11 |
| US20040097504A1 (en) | 2004-05-20 |
| AU2003295396A1 (en) | 2004-06-07 |
| WO2004041814A1 (en) | 2004-05-21 |
| AU2003295396B2 (en) | 2009-02-26 |
| US7259161B2 (en) | 2007-08-21 |
| ATE371656T1 (de) | 2007-09-15 |
| ES2289349T3 (es) | 2008-02-01 |
| JP2006514006A (ja) | 2006-04-27 |
| EP1562938A1 (en) | 2005-08-17 |
| JP2011016839A (ja) | 2011-01-27 |
| EP1562938B1 (en) | 2007-08-29 |
| CA2506773A1 (en) | 2004-05-21 |
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