AU2003295396B2 - Heteroaryl-pyramidine derivatives as JAK inhibitors - Google Patents
Heteroaryl-pyramidine derivatives as JAK inhibitors Download PDFInfo
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- AU2003295396B2 AU2003295396B2 AU2003295396A AU2003295396A AU2003295396B2 AU 2003295396 B2 AU2003295396 B2 AU 2003295396B2 AU 2003295396 A AU2003295396 A AU 2003295396A AU 2003295396 A AU2003295396 A AU 2003295396A AU 2003295396 B2 AU2003295396 B2 AU 2003295396B2
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- iva
- ivb
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- hydrogen
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Landscapes
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| US42357902P | 2002-11-04 | 2002-11-04 | |
| US60/423,579 | 2002-11-04 | ||
| PCT/US2003/035163 WO2004041814A1 (en) | 2002-11-04 | 2003-11-04 | Heteroaryl-pyramidine derivatives as jak inhibitors |
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| TWI329105B (en) * | 2002-02-01 | 2010-08-21 | Rigel Pharmaceuticals Inc | 2,4-pyrimidinediamine compounds and their uses |
| CN103169708B (zh) | 2002-07-29 | 2018-02-02 | 里格尔药品股份有限公司 | 用2,4‑嘧啶二胺化合物治疗或者预防自体免疫性疾病的方法 |
| JP4886511B2 (ja) * | 2003-07-30 | 2012-02-29 | ライジェル ファーマシューティカルズ， インコーポレイテッド | ２，４−ピリミジンジアミン化合物による自己免疫疾患の治療または予防方法 |
| RU2007107177A (ru) * | 2004-07-28 | 2008-09-10 | Айрм Ллк (Bm) | Соединения и композиции, как модуляторы ядерных рецепторов стероидных гормонов |
| WO2006047492A2 (en) | 2004-10-22 | 2006-05-04 | Amgen Inc. | Substituted nitrogen-containing heterocycles as vanilloid receptor ligands and their uses as medicament |
| ATE540035T1 (de) | 2004-11-24 | 2012-01-15 | Rigel Pharmaceuticals Inc | Spiro-2,4-pyrimidindiamin-verbindungen und ihre verwendungen |
| KR101484499B1 (ko) | 2005-02-14 | 2015-01-20 | 존슨 앤드 존슨 비젼 케어, 인코포레이티드 | 안과용 렌즈의 제조방법, 안과용 장치 및 콘택트 렌즈 |
| EP1883302A4 (en) * | 2005-05-03 | 2009-05-20 | Rigel Pharmaceuticals Inc | JAK KINASE HEMMER AND ITS USE |
| US20070203161A1 (en) | 2006-02-24 | 2007-08-30 | Rigel Pharmaceuticals, Inc. | Compositions and methods for inhibition of the jak pathway |
| JP5225079B2 (ja) | 2005-06-08 | 2013-07-03 | ライジェル ファーマシューティカルズ， インコーポレイテッド | Ｊａｋ経路の阻害のための組成物および方法 |
| PL1951684T3 (pl) | 2005-11-01 | 2017-03-31 | Targegen, Inc. | Biarylowe meta-pirymidynowe inhibitory kinaz |
| US8604042B2 (en) | 2005-11-01 | 2013-12-10 | Targegen, Inc. | Bi-aryl meta-pyrimidine inhibitors of kinases |
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| AU2006316322B2 (en) * | 2005-11-22 | 2011-08-25 | Merck Canada Inc. | Tricyclic compounds useful as inhibitors of kinases |
| EP2474545B1 (en) | 2005-12-13 | 2016-11-09 | Incyte Holdings Corporation | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors |
| EA200870217A1 (ru) * | 2006-01-30 | 2009-02-27 | Экселиксис, Инк. | 4-арил-2-аминопиримидины или 4-арил-2-аминоалкилпиримидины в качестве модуляторов jak-2 и содержащие их фармацевтические композиции |
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| GB9523675D0 (en) | 1995-11-20 | 1996-01-24 | Celltech Therapeutics Ltd | Chemical compounds |
| CN1438890A (zh) * | 2000-02-25 | 2003-08-27 | 弗·哈夫曼-拉罗切有限公司 | 腺苷受体调制剂 |
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- 2003-11-04 US US10/700,936 patent/US7259161B2/en not_active Expired - Fee Related
- 2003-11-04 DE DE60316013T patent/DE60316013T2/de not_active Expired - Lifetime
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- 2003-11-04 JP JP2004550483A patent/JP4688498B2/ja not_active Expired - Fee Related
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| US7259161B2 (en) | 2007-08-21 |
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| EP1562938B1 (en) | 2007-08-29 |
| AU2003295396A1 (en) | 2004-06-07 |
| DE60316013T2 (de) | 2008-05-29 |
| EP1562938A1 (en) | 2005-08-17 |
| US20040097504A1 (en) | 2004-05-20 |
| DE60316013D1 (de) | 2007-10-11 |
| ATE371656T1 (de) | 2007-09-15 |
| JP2011016839A (ja) | 2011-01-27 |
| WO2004041814A1 (en) | 2004-05-21 |
| JP2006514006A (ja) | 2006-04-27 |
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