DE60309433T2 - Pharmazeutische zusammensetzungen für proteasehemmer für hepatitis-c-virus - Google Patents
Pharmazeutische zusammensetzungen für proteasehemmer für hepatitis-c-virus Download PDFInfo
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- DE60309433T2 DE60309433T2 DE60309433T DE60309433T DE60309433T2 DE 60309433 T2 DE60309433 T2 DE 60309433T2 DE 60309433 T DE60309433 T DE 60309433T DE 60309433 T DE60309433 T DE 60309433T DE 60309433 T2 DE60309433 T2 DE 60309433T2
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Dermatology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Virology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Communicable Diseases (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35569402P | 2002-02-07 | 2002-02-07 | |
| US355694P | 2002-02-07 | ||
| PCT/US2003/003380 WO2003066103A1 (en) | 2002-02-07 | 2003-02-05 | Pharmaceutical compositions for hepatitis c viral protease inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60309433D1 DE60309433D1 (de) | 2006-12-14 |
| DE60309433T2 true DE60309433T2 (de) | 2007-05-03 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60309433T Expired - Fee Related DE60309433T2 (de) | 2002-02-07 | 2003-02-05 | Pharmazeutische zusammensetzungen für proteasehemmer für hepatitis-c-virus |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US6828301B2 (enExample) |
| EP (1) | EP1474172B1 (enExample) |
| JP (1) | JP2005518423A (enExample) |
| KR (1) | KR20040089605A (enExample) |
| CN (1) | CN1627959A (enExample) |
| AR (1) | AR038823A1 (enExample) |
| AT (1) | ATE344056T1 (enExample) |
| AU (1) | AU2003208989A1 (enExample) |
| BR (1) | BR0307524A (enExample) |
| CA (1) | CA2472249A1 (enExample) |
| CO (1) | CO5611167A2 (enExample) |
| DE (1) | DE60309433T2 (enExample) |
| EA (1) | EA200400991A1 (enExample) |
| EC (1) | ECSP045223A (enExample) |
| ES (1) | ES2276045T3 (enExample) |
| HR (1) | HRP20040720A2 (enExample) |
| IL (1) | IL162673A0 (enExample) |
| MX (1) | MXPA04007699A (enExample) |
| NO (1) | NO20043722L (enExample) |
| PE (1) | PE20030865A1 (enExample) |
| PL (1) | PL371287A1 (enExample) |
| TW (1) | TW200302734A (enExample) |
| UY (1) | UY27650A1 (enExample) |
| WO (1) | WO2003066103A1 (enExample) |
| ZA (1) | ZA200405064B (enExample) |
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| DE60334205D1 (en) | 2002-05-20 | 2010-10-28 | Bristol Myers Squibb Co | Heterocyclische sulfonamid-hepatitis-c-virus-hemmer |
| MY140680A (en) | 2002-05-20 | 2010-01-15 | Bristol Myers Squibb Co | Hepatitis c virus inhibitors |
| DE60324552D1 (en) | 2002-05-20 | 2008-12-18 | Bristol Myers Squibb Co | Substituierte cycloalkyl p1' hepatitis c virus inhibitoren |
| AU2003299519A1 (en) | 2002-05-20 | 2004-05-04 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
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| US20050159345A1 (en) * | 2002-10-29 | 2005-07-21 | Boehringer Ingelheim International Gmbh | Composition for the treatment of infection by Flaviviridae viruses |
| WO2004050068A1 (en) * | 2002-11-29 | 2004-06-17 | Janssen Pharmaceutica N.V. | Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base |
| UY28240A1 (es) * | 2003-03-27 | 2004-11-08 | Boehringer Ingelheim Pharma | Fases cristalinas de un potente inhibidor de la hcv |
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| US7176208B2 (en) * | 2003-04-18 | 2007-02-13 | Enanta Pharmaceuticals, Inc. | Quinoxalinyl macrocyclic hepatitis C serine protease inhibitors |
| ES2361997T3 (es) * | 2003-09-22 | 2011-06-27 | Boehringer Ingelheim International Gmbh | Péptidos macrocíclicos activos contra el virus de la hepatitis c. |
| OA13315A (en) * | 2003-10-14 | 2007-04-13 | Intermune Inc | Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of HCV replication. |
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| CA2539575C (en) | 2003-11-20 | 2015-01-20 | Boehringer Ingelheim International Gmbh | Method of removing transition metals, especially from metathesis reaction products |
| US7309708B2 (en) | 2003-11-20 | 2007-12-18 | Birstol-Myers Squibb Company | Hepatitis C virus inhibitors |
| WO2005070955A1 (en) * | 2004-01-21 | 2005-08-04 | Boehringer Ingelheim International Gmbh | Macrocyclic peptides active against the hepatitis c virus |
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| EP1765283A4 (en) * | 2004-06-08 | 2012-11-28 | Vertex Pharma | PHARMACEUTICAL COMPOSITIONS |
| HRP20070043A2 (hr) * | 2004-07-16 | 2007-07-31 | Gilead Sciences | Antivirusna sredstva |
| WO2007001406A2 (en) * | 2004-10-05 | 2007-01-04 | Chiron Corporation | Aryl-containing macrocyclic compounds |
| JP2008517896A (ja) * | 2004-10-21 | 2008-05-29 | ファイザー・インク | Ｃ型肝炎ウイルスプロテアーゼの阻害剤並びにそれを用いた組成物及び治療 |
| US20060088591A1 (en) * | 2004-10-22 | 2006-04-27 | Jinghua Yuan | Tablets from a poorly compressible substance |
| BRPI0518239A2 (pt) * | 2004-10-29 | 2008-11-11 | Novartis Ag | composiÇÕes farmacÊuticas espontaneamente dispersÍveis |
| US7323447B2 (en) | 2005-02-08 | 2008-01-29 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US20060240051A1 (en) * | 2005-04-26 | 2006-10-26 | Singleton Andy H | Eutectic blends containing a water soluble vitamin derivative |
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| BRPI0617274A2 (pt) | 2005-10-11 | 2011-07-19 | Intermune Inc | compostos e métodos para a inibição de replicação viral de hepatite c |
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| US7741281B2 (en) | 2005-11-03 | 2010-06-22 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| RU2008152171A (ru) | 2006-07-05 | 2010-08-10 | Интермьюн, Инк. (Us) | Новые ингибиторы вирусной репликации гепатита с |
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| AP3770A (en) | 2010-11-18 | 2016-08-31 | Metalysis Ltd | Electrolysis apparatus |
| JP2014502620A (ja) | 2010-12-30 | 2014-02-03 | エナンタ ファーマシューティカルズ インコーポレイテッド | 大環状ｃ型肝炎セリンプロテアーゼ阻害剤 |
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| US9034832B2 (en) | 2011-12-29 | 2015-05-19 | Abbvie Inc. | Solid compositions |
| US20130302414A1 (en) * | 2012-05-07 | 2013-11-14 | Bristol-Myers Squibb Company | Solubilized capsule formulation of 1,1-dimethylethyl [(1s)-1-carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate |
| WO2014062196A1 (en) * | 2012-10-19 | 2014-04-24 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| US9643999B2 (en) | 2012-11-02 | 2017-05-09 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| EP2914613B1 (en) | 2012-11-02 | 2017-11-22 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| WO2014071007A1 (en) | 2012-11-02 | 2014-05-08 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| WO2014070974A1 (en) | 2012-11-05 | 2014-05-08 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
| EP2964664B1 (en) | 2013-03-07 | 2017-01-11 | Bristol-Myers Squibb Company | Hepatitis c virus inhibitors |
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| EP2899207A1 (en) | 2014-01-28 | 2015-07-29 | Amikana.Biologics | New method for testing HCV protease inhibition |
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Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE445174B (sv) | 1978-03-07 | 1986-06-09 | Sandoz Ag | Farmaceutisk komposition innehallande en cyklosporin och en berarsubstans |
| US5071643A (en) | 1986-10-17 | 1991-12-10 | R. P. Scherer Corporation | Solvent system enhancing the solubility of pharmaceuticals for encapsulation |
| US5342625A (en) | 1988-09-16 | 1994-08-30 | Sandoz Ltd. | Pharmaceutical compositions comprising cyclosporins |
| IL102236A0 (en) | 1991-06-27 | 1993-01-14 | Ltt Inst Co Ltd | Topical preparations containing cyclosporin |
| GB9208712D0 (en) | 1992-04-22 | 1992-06-10 | Sandoz Ltd | Pharmaceutical compositions containing cyclosporin derivates |
| US5376688A (en) | 1992-12-18 | 1994-12-27 | R. P. Scherer Corporation | Enhanced solubility pharmaceutical solutions |
| CA2221145A1 (en) | 1995-05-19 | 1996-11-21 | Abbott Laboratories | Self-emulsifying formulations of lipophilic drugs |
| BR9810866B1 (pt) | 1997-07-29 | 2010-07-13 | composição farmacêutica em uma forma de formulação auto-emulsificante para compostos lipofìlicos. | |
| NZ502566A (en) | 1997-07-29 | 2002-03-28 | Upjohn Co | Pharmaceutical composition for acidic lipophilic compounds in a form of a self-emulsifying formulation containing a pyranone and a basic amine |
| US6056977A (en) | 1997-10-15 | 2000-05-02 | Edward Mendell Co., Inc. | Once-a-day controlled release sulfonylurea formulation |
| UA74546C2 (en) | 1999-04-06 | 2006-01-16 | Boehringer Ingelheim Ca Ltd | Macrocyclic peptides having activity relative to hepatitis c virus, a pharmaceutical composition and use of the pharmaceutical composition |
-
2003
- 2003-02-04 US US10/357,919 patent/US6828301B2/en not_active Expired - Lifetime
- 2003-02-05 HR HR20040720A patent/HRP20040720A2/hr not_active Application Discontinuation
- 2003-02-05 EA EA200400991A patent/EA200400991A1/ru unknown
- 2003-02-05 CA CA002472249A patent/CA2472249A1/en not_active Abandoned
- 2003-02-05 BR BR0307524-9A patent/BR0307524A/pt not_active Application Discontinuation
- 2003-02-05 EP EP03707713A patent/EP1474172B1/en not_active Expired - Lifetime
- 2003-02-05 ES ES03707713T patent/ES2276045T3/es not_active Expired - Lifetime
- 2003-02-05 DE DE60309433T patent/DE60309433T2/de not_active Expired - Fee Related
- 2003-02-05 PL PL03371287A patent/PL371287A1/xx not_active Application Discontinuation
- 2003-02-05 UY UY27650A patent/UY27650A1/es not_active Application Discontinuation
- 2003-02-05 AT AT03707713T patent/ATE344056T1/de not_active IP Right Cessation
- 2003-02-05 KR KR10-2004-7012235A patent/KR20040089605A/ko not_active Withdrawn
- 2003-02-05 IL IL16267303A patent/IL162673A0/xx unknown
- 2003-02-05 JP JP2003565526A patent/JP2005518423A/ja active Pending
- 2003-02-05 CN CNA03803395XA patent/CN1627959A/zh active Pending
- 2003-02-05 MX MXPA04007699A patent/MXPA04007699A/es not_active Application Discontinuation
- 2003-02-05 WO PCT/US2003/003380 patent/WO2003066103A1/en not_active Ceased
- 2003-02-05 PE PE2003000135A patent/PE20030865A1/es not_active Application Discontinuation
- 2003-02-05 AU AU2003208989A patent/AU2003208989A1/en not_active Abandoned
- 2003-02-06 TW TW092102382A patent/TW200302734A/zh unknown
- 2003-02-07 AR ARP030100386A patent/AR038823A1/es unknown
-
2004
- 2004-06-25 ZA ZA200405064A patent/ZA200405064B/en unknown
- 2004-08-06 EC EC2004005223A patent/ECSP045223A/es unknown
- 2004-09-06 NO NO20043722A patent/NO20043722L/no not_active Application Discontinuation
- 2004-09-07 CO CO04088288A patent/CO5611167A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EP1474172B1 (en) | 2006-11-02 |
| NO20043722L (no) | 2004-09-06 |
| DE60309433D1 (de) | 2006-12-14 |
| UY27650A1 (es) | 2003-09-30 |
| MXPA04007699A (es) | 2004-11-10 |
| EA200400991A1 (ru) | 2005-02-24 |
| US20030195228A1 (en) | 2003-10-16 |
| JP2005518423A (ja) | 2005-06-23 |
| IL162673A0 (en) | 2005-11-20 |
| CN1627959A (zh) | 2005-06-15 |
| EP1474172A1 (en) | 2004-11-10 |
| ZA200405064B (en) | 2005-05-30 |
| ATE344056T1 (de) | 2006-11-15 |
| AR038823A1 (es) | 2005-01-26 |
| WO2003066103A1 (en) | 2003-08-14 |
| TW200302734A (en) | 2003-08-16 |
| PL371287A1 (en) | 2005-06-13 |
| CA2472249A1 (en) | 2003-08-14 |
| CO5611167A2 (es) | 2006-02-28 |
| KR20040089605A (ko) | 2004-10-21 |
| US6828301B2 (en) | 2004-12-07 |
| HRP20040720A2 (en) | 2005-04-30 |
| ECSP045223A (es) | 2004-09-28 |
| ES2276045T3 (es) | 2007-06-16 |
| PE20030865A1 (es) | 2003-11-26 |
| AU2003208989A1 (en) | 2003-09-02 |
| BR0307524A (pt) | 2004-12-21 |
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