DE60102925T2 - Amino-thiolester-verbindungen, diese enthaltende pharmazeutische und kosmetische zusammensetzungen und ihre anwendungen - Google Patents
Amino-thiolester-verbindungen, diese enthaltende pharmazeutische und kosmetische zusammensetzungen und ihre anwendungen Download PDFInfo
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- DE60102925T2 DE60102925T2 DE60102925T DE60102925T DE60102925T2 DE 60102925 T2 DE60102925 T2 DE 60102925T2 DE 60102925 T DE60102925 T DE 60102925T DE 60102925 T DE60102925 T DE 60102925T DE 60102925 T2 DE60102925 T2 DE 60102925T2
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Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/08—Antiseborrheics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/12—Keratolytics, e.g. wart or anti-corn preparations
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/16—Emollients or protectives, e.g. against radiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
- C07C327/20—Esters of monothiocarboxylic acids
- C07C327/22—Esters of monothiocarboxylic acids having carbon atoms of esterified thiocarboxyl groups bound to hydrogen atoms or to acyclic carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Immunology (AREA)
- Virology (AREA)
- Rheumatology (AREA)
- Molecular Biology (AREA)
- Pulmonology (AREA)
- Ophthalmology & Optometry (AREA)
- Pain & Pain Management (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Toxicology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0007029A FR2809727B1 (fr) | 2000-05-31 | 2000-05-31 | Nouveaux composes aminothiolesters, compositions pharmaceutiques et cosmetiques les contenant et utilisations |
| FR0007029 | 2000-05-31 | ||
| PCT/FR2001/001694 WO2001092220A1 (fr) | 2000-05-31 | 2001-05-31 | Composes aminothiolesters, compositions pharmaceutiques et cosmetiques les contenant et utilisations |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE60102925D1 DE60102925D1 (de) | 2004-05-27 |
| DE60102925T2 true DE60102925T2 (de) | 2005-04-07 |
Family
ID=8850863
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE60102925T Expired - Lifetime DE60102925T2 (de) | 2000-05-31 | 2001-05-31 | Amino-thiolester-verbindungen, diese enthaltende pharmazeutische und kosmetische zusammensetzungen und ihre anwendungen |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8026231B2 (enExample) |
| EP (1) | EP1296946B1 (enExample) |
| JP (1) | JP4855626B2 (enExample) |
| AR (1) | AR028122A1 (enExample) |
| AT (1) | ATE264839T1 (enExample) |
| AU (1) | AU2001274171A1 (enExample) |
| DE (1) | DE60102925T2 (enExample) |
| ES (1) | ES2219530T3 (enExample) |
| FR (1) | FR2809727B1 (enExample) |
| WO (1) | WO2001092220A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2983492B1 (fr) * | 2011-12-06 | 2015-10-30 | Advanced Biodesign | Procede ex vivo de purge tumorale d'un echantillon biologique |
| PL3362094T3 (pl) * | 2015-10-15 | 2021-10-11 | Advanced Biodesign | Kombinacja zawierająca związek tioaminoestrowy lub jego farmaceutycznie dopuszczalną sól oraz związek mogący zwiększyć poziom h2o2 w komórkach nowotworowych osobnika |
| LT3362056T (lt) | 2015-10-15 | 2021-05-10 | Advanced Biodesign | Aminotiolesterio junginiai arba jų farmaciniu požiūriu priimtinos druskos, skirti naudoti vėžio gydyme |
| FR3047734B1 (fr) * | 2016-02-17 | 2019-09-06 | Advanced Biodesign | Procede de preparation de composes aminothiolester et leurs sels |
| US20220265845A1 (en) * | 2019-07-31 | 2022-08-25 | Advanced Biodesign | Aminothiolester compounds and uses thereof |
| EP4035666A1 (en) | 2021-01-29 | 2022-08-03 | Advanced Biodesign | Aminothiolester compound or derivative thereof for use as an immunomodulatory agent |
| FR3119314B1 (fr) | 2021-01-29 | 2025-01-10 | Advanced Biodesign | Nanocapsule lipidique comprenant au moins un composé aminothiolester ou un de ses dérivés pharmaceutiquement acceptable |
| WO2025229179A1 (en) | 2024-05-03 | 2025-11-06 | Advanced Biodesign | Use of aminothiolester compounds in combination with hypomethylating agents (hma) for the prevention and treatment of cancer |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5051528A (en) * | 1990-04-24 | 1991-09-24 | Eastman Kodak Company | Recovery process for ethylene glycol and dimethylterephthalate |
| JPH0797350A (ja) * | 1993-08-02 | 1995-04-11 | Mitsubishi Chem Corp | ベンゾイルアセチレン誘導体 |
| FR2761606B1 (fr) * | 1997-04-08 | 1999-05-14 | Cird Galderma | Utilisation de derives aminothiolesters dans le domaine pharmaceutique |
| KR100488985B1 (ko) | 1997-12-02 | 2005-05-11 | 하인리히 스무다 | 폴리에틸렌테레프탈레이트 폐기물로부터 테레프탈산 및 에틸렌글리콜을 회수하는 방법 |
| FR2777001B1 (fr) * | 1998-04-01 | 2000-06-09 | Cird Galderma | Derives de l'acide 6,8-dimercaptooctanoique substitues en 6-s et/ou en 8-s par le radical (3-methylthiopropanoyl) et compositions pharmaceutiques destinees au traitement des tumeurs cancereuses |
| EP1227075B1 (en) | 1999-10-22 | 2009-07-29 | Teijin Limited | Method for separating and recovering dimethyl terephthalate and ethylene glycol from polyester waste |
| JP3808672B2 (ja) * | 1999-11-26 | 2006-08-16 | 東洋製罐株式会社 | 回収ポリエチレンテレフタレート粉砕品からのテレフタル酸の工業的回収方法 |
-
2000
- 2000-05-31 FR FR0007029A patent/FR2809727B1/fr not_active Expired - Fee Related
-
2001
- 2001-05-30 AR ARP010102577A patent/AR028122A1/es unknown
- 2001-05-31 JP JP2002500835A patent/JP4855626B2/ja not_active Expired - Lifetime
- 2001-05-31 EP EP01940654A patent/EP1296946B1/fr not_active Expired - Lifetime
- 2001-05-31 AU AU2001274171A patent/AU2001274171A1/en not_active Abandoned
- 2001-05-31 WO PCT/FR2001/001694 patent/WO2001092220A1/fr not_active Ceased
- 2001-05-31 ES ES01940654T patent/ES2219530T3/es not_active Expired - Lifetime
- 2001-05-31 AT AT01940654T patent/ATE264839T1/de not_active IP Right Cessation
- 2001-05-31 DE DE60102925T patent/DE60102925T2/de not_active Expired - Lifetime
-
2006
- 2006-03-28 US US11/390,480 patent/US8026231B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| FR2809727A1 (fr) | 2001-12-07 |
| DE60102925D1 (de) | 2004-05-27 |
| WO2001092220A1 (fr) | 2001-12-06 |
| JP4855626B2 (ja) | 2012-01-18 |
| JP2003535076A (ja) | 2003-11-25 |
| EP1296946B1 (fr) | 2004-04-21 |
| AU2001274171A1 (en) | 2001-12-11 |
| AR028122A1 (es) | 2003-04-23 |
| US20070032476A1 (en) | 2007-02-08 |
| ATE264839T1 (de) | 2004-05-15 |
| ES2219530T3 (es) | 2004-12-01 |
| EP1296946A1 (fr) | 2003-04-02 |
| FR2809727B1 (fr) | 2002-07-26 |
| US8026231B2 (en) | 2011-09-27 |
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