DE2050684A1 - Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo - Google Patents

Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo

Info

Publication number
DE2050684A1
DE2050684A1 DE19702050684 DE2050684A DE2050684A1 DE 2050684 A1 DE2050684 A1 DE 2050684A1 DE 19702050684 DE19702050684 DE 19702050684 DE 2050684 A DE2050684 A DE 2050684A DE 2050684 A1 DE2050684 A1 DE 2050684A1
Authority
DE
Germany
Prior art keywords
piperazines
formula
general formula
halogen
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19702050684
Other languages
German (de)
English (en)
Inventor
Ernst-Otto Dr.; Mentrup Anton Dr.; Schromm Kurt Dr.; 6507 Ingelheim. C07d 51-42 Renth
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
C.H. Boehringer Sohn AG and Co KG
Original Assignee
C.H. Boehringer Sohn AG and Co KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by C.H. Boehringer Sohn AG and Co KG filed Critical C.H. Boehringer Sohn AG and Co KG
Priority to DE19702050684 priority Critical patent/DE2050684A1/de
Priority to HUBO1323A priority patent/HU162740B/hu
Priority to CH1491871A priority patent/CH562236A5/xx
Priority to SE7112983A priority patent/SE395144B/xx
Priority to BG018756A priority patent/BG18869A3/xx
Priority to ES395969A priority patent/ES395969A1/es
Priority to PL1971151024A priority patent/PL77016B1/pl
Priority to FI2885/71A priority patent/FI54922C/fi
Priority to CA125,116A priority patent/CA967159A/en
Priority to AT890171A priority patent/AT313902B/de
Priority to YU2633/71A priority patent/YU34695B/xx
Priority to DK503071A priority patent/DK142580C/da
Publication of DE2050684A1 publication Critical patent/DE2050684A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
    • C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring
    • C07D295/033—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/58—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
DE19702050684 1970-10-15 1970-10-15 Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo Pending DE2050684A1 (en)

Priority Applications (12)

Application Number Priority Date Filing Date Title
DE19702050684 DE2050684A1 (en) 1970-10-15 1970-10-15 Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo
HUBO1323A HU162740B (enExample) 1970-10-15 1971-10-12
CH1491871A CH562236A5 (enExample) 1970-10-15 1971-10-12
SE7112983A SE395144B (sv) 1970-10-15 1971-10-13 Nytt forfarande for framstellning av 1-arylpropyl(2)-piperazinderivat
BG018756A BG18869A3 (bg) 1970-10-15 1971-10-13 Метод за получаване на пиперазинови производни
ES395969A ES395969A1 (es) 1970-10-15 1971-10-14 Procedimiento para la preparacion de derivados de piperazi-na.
PL1971151024A PL77016B1 (enExample) 1970-10-15 1971-10-14
FI2885/71A FI54922C (fi) 1970-10-15 1971-10-14 Nytt foerfarande foer framstaellning av piperazinderivat
CA125,116A CA967159A (en) 1970-10-15 1971-10-14 Process for the production of piperazine derivatives
AT890171A AT313902B (de) 1970-10-15 1971-10-14 Verfahren zur Herstellung von Piperazinderivaten sowie von deren Säureadditionssalzen
YU2633/71A YU34695B (en) 1970-10-15 1971-10-15 Process for preparing piperazine derivatives
DK503071A DK142580C (da) 1970-10-15 1971-10-15 Fremgangsmaade til fremstilling af piperazinderivater

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19702050684 DE2050684A1 (en) 1970-10-15 1970-10-15 Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo

Publications (1)

Publication Number Publication Date
DE2050684A1 true DE2050684A1 (en) 1972-04-20

Family

ID=5785239

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19702050684 Pending DE2050684A1 (en) 1970-10-15 1970-10-15 Neuroleptic 1-aralkyl-4-phenyl-piperazines prodn - by reacting ethylenediamines with oxalic acid derivs,and reducing resulting dioxo

Country Status (12)

Country Link
AT (1) AT313902B (enExample)
BG (1) BG18869A3 (enExample)
CA (1) CA967159A (enExample)
CH (1) CH562236A5 (enExample)
DE (1) DE2050684A1 (enExample)
DK (1) DK142580C (enExample)
ES (1) ES395969A1 (enExample)
FI (1) FI54922C (enExample)
HU (1) HU162740B (enExample)
PL (1) PL77016B1 (enExample)
SE (1) SE395144B (enExample)
YU (1) YU34695B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604838A1 (de) * 1976-02-07 1977-08-11 Knoll Ag Alkylendioxypiperazinderivate

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604838A1 (de) * 1976-02-07 1977-08-11 Knoll Ag Alkylendioxypiperazinderivate

Also Published As

Publication number Publication date
PL77016B1 (enExample) 1975-02-28
FI54922C (fi) 1979-04-10
DK142580B (da) 1980-11-24
FI54922B (fi) 1978-12-29
SE395144B (sv) 1977-08-01
BG18869A3 (bg) 1975-03-20
HU162740B (enExample) 1973-04-28
ES395969A1 (es) 1973-12-16
AT313902B (de) 1974-03-11
YU263371A (en) 1979-07-10
CH562236A5 (enExample) 1975-05-30
CA967159A (en) 1975-05-06
DK142580C (da) 1981-07-13
YU34695B (en) 1979-12-31

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