DD287502A5 - Verfahren zur herstellung von n-piperidylbenzamiden - Google Patents

Verfahren zur herstellung von n-piperidylbenzamiden Download PDF

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Publication number
DD287502A5
DD287502A5 DD86293410A DD29341086A DD287502A5 DD 287502 A5 DD287502 A5 DD 287502A5 DD 86293410 A DD86293410 A DD 86293410A DD 29341086 A DD29341086 A DD 29341086A DD 287502 A5 DD287502 A5 DD 287502A5
Authority
DD
German Democratic Republic
Prior art keywords
group
compound
formula
amino
methyl
Prior art date
Application number
DD86293410A
Other languages
German (de)
English (en)
Inventor
Armando V Noverola
Jose M P Soto
Fernando P Noguera
Jacinto M Mauri
Robert W G Spickett
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ��������@�K@�Kk�� filed Critical ��������@�K@�Kk��
Publication of DD287502A5 publication Critical patent/DD287502A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
    • C07D211/66—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4 having a hetero atom as the second substituent in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/10—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DD86293410A 1985-08-06 1986-08-04 Verfahren zur herstellung von n-piperidylbenzamiden DD287502A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858519707A GB8519707D0 (en) 1985-08-06 1985-08-06 Chemical compounds

Publications (1)

Publication Number Publication Date
DD287502A5 true DD287502A5 (de) 1991-02-28

Family

ID=10583372

Family Applications (1)

Application Number Title Priority Date Filing Date
DD86293410A DD287502A5 (de) 1985-08-06 1986-08-04 Verfahren zur herstellung von n-piperidylbenzamiden

Country Status (28)

Country Link
US (1) US4772618A (fr)
EP (1) EP0213775B1 (fr)
JP (1) JPH0662614B2 (fr)
KR (1) KR920001763B1 (fr)
CN (1) CN1022830C (fr)
AR (2) AR243521A1 (fr)
AT (1) ATE49206T1 (fr)
AU (1) AU596110B2 (fr)
CA (1) CA1300154C (fr)
DD (1) DD287502A5 (fr)
DE (1) DE3667975D1 (fr)
DK (1) DK370586A (fr)
EG (1) EG18154A (fr)
ES (2) ES2000706A6 (fr)
FI (1) FI89168C (fr)
GB (1) GB8519707D0 (fr)
GR (1) GR862060B (fr)
HU (1) HU201060B (fr)
IE (1) IE58751B1 (fr)
IL (1) IL79469A0 (fr)
MX (1) MX3375A (fr)
MY (1) MY101352A (fr)
NO (1) NO168706C (fr)
NZ (1) NZ217078A (fr)
PH (1) PH25019A (fr)
PL (1) PL150228B1 (fr)
PT (2) PT83146B (fr)
ZA (1) ZA865537B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2640139A1 (fr) * 1988-12-14 1990-06-15 Delagrange Laboratoires Application de benzamides substitues comme gastromoteurs
US5374637A (en) * 1989-03-22 1994-12-20 Janssen Pharmaceutica N.V. N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives
GB9005014D0 (en) * 1990-03-06 1990-05-02 Janssen Pharmaceutica Nv N.(4.piperidinyl)(dihydrobenzofuran or dihydro.2h.benzopyran)carboxamide derivatives
JP2999669B2 (ja) * 1993-08-24 2000-01-17 株式会社三和化学研究所 ベンゾ［ｂ］フランカルボキサミド誘導体、その製法及び用途
JPH0820586A (ja) * 1994-07-05 1996-01-23 Sanwa Kagaku Kenkyusho Co Ltd １−アザビシクロ［３．３．０］オクタン誘導体、その塩及び製法並びに用途
JPH0873463A (ja) 1994-07-05 1996-03-19 Sanwa Kagaku Kenkyusho Co Ltd ベンゾピランカルボキサミド誘導体、その塩及び製法並びに用途
CN1052228C (zh) * 1996-01-17 2000-05-10 中国科学院大连化学物理研究所 N-甲酰基哌啶及其同系物的制备方法
CN1091104C (zh) * 1998-04-02 2002-09-18 中国科学院大连化学物理研究所 一种n－甲酰基哌啶的制备方法
CN1649766A (zh) 2002-06-11 2005-08-03 安芸电器株式会社 自行车的前照灯以及前照灯电路
WO2005068461A1 (fr) * 2004-01-07 2005-07-28 Aryx Therapeutics Composes stereo-isomeres et methodes de traitement de troubles gastro-intestinaux et du systeme nerveux central
GB0525661D0 (en) * 2005-12-16 2006-01-25 Glaxo Group Ltd Novel compounds
JP5845263B2 (ja) * 2010-09-01 2016-01-20 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプＪａｎｓｓｅｎ Ｐｈａｒｍａｃｅｕｔｉｃａ Ｎａａｍｌｏｚｅ Ｖｅｎｎｏｏｔｓｃｈａｐ ５−ｈｔ２ｂ受容体アンタゴニスト
CN110950843B (zh) * 2019-11-28 2022-12-27 广东东阳光药业有限公司 取代的苯酰胺衍生物及其用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1019781A (fr) 1963-03-05
US3342826A (en) 1964-01-13 1967-09-19 Ile De France Heterocyclic aminoalkyl benzamides
GB1507462A (en) * 1974-03-21 1978-04-12 Gallardo Antonio Sa N-heterocyclic substituted benzamides methods for their preparation and compositions containing them
GB1574418A (en) * 1976-11-16 1980-09-03 Anphar Sa Piperidine derivatives
CA1183847A (fr) * 1981-10-01 1985-03-12 Georges Van Daele N-(3-hydroxy-4-piperidinyl)benzamide; derives

Also Published As

Publication number Publication date
PT83147A (en) 1986-09-01
AR243521A1 (es) 1993-08-31
IL79469A0 (en) 1986-10-31
FI89168C (fi) 1993-08-25
PH25019A (en) 1991-01-28
KR920001763B1 (ko) 1992-03-02
DK370586A (da) 1987-03-27
EP0213775A1 (fr) 1987-03-11
CN86105972A (zh) 1987-04-01
GB8519707D0 (en) 1985-09-11
KR870002071A (ko) 1987-03-28
PL260921A1 (en) 1988-01-07
IE58751B1 (en) 1993-11-03
FI863179A (fi) 1987-02-07
AR242793A1 (es) 1993-05-31
PT83147B (pt) 1988-07-29
HUT44782A (en) 1988-04-28
IE862073L (en) 1987-02-06
NO863139L (no) 1987-02-09
AU596110B2 (en) 1990-04-26
JPH0662614B2 (ja) 1994-08-17
AU6075886A (en) 1987-02-12
CN1022830C (zh) 1993-11-24
FI863179A0 (fi) 1986-08-04
FI89168B (fi) 1993-05-14
EG18154A (en) 1992-11-30
CA1300154C (fr) 1992-05-05
NO168706C (no) 1992-03-25
PT83146A (en) 1986-09-01
NZ217078A (en) 1989-01-27
NO168706B (no) 1991-12-16
PL150228B1 (en) 1990-05-31
MX3375A (es) 1993-12-01
ZA865537B (en) 1987-03-25
NO863139D0 (no) 1986-08-04
ATE49206T1 (de) 1990-01-15
HU201060B (en) 1990-09-28
DK370586D0 (da) 1986-08-04
ES2000706A6 (es) 1988-03-16
ES2000705A6 (es) 1988-03-16
GR862060B (en) 1986-12-24
PT83146B (pt) 1988-07-29
EP0213775B1 (fr) 1990-01-03
DE3667975D1 (en) 1990-02-08
US4772618A (en) 1988-09-20
MY101352A (en) 1991-09-05
JPS62129279A (ja) 1987-06-11

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ENJ Ceased due to non-payment of renewal fee