DD202435A5 - Verbessertes verfahren zur herstellung von penicillansaeureestern - Google Patents

Verbessertes verfahren zur herstellung von penicillansaeureestern Download PDF

Info

Publication number
DD202435A5
DD202435A5 DD82238309A DD23830982A DD202435A5 DD 202435 A5 DD202435 A5 DD 202435A5 DD 82238309 A DD82238309 A DD 82238309A DD 23830982 A DD23830982 A DD 23830982A DD 202435 A5 DD202435 A5 DD 202435A5
Authority
DD
German Democratic Republic
Prior art keywords
penicillanate
dioxide
reaction
ethyl acetate
concentrated
Prior art date
Application number
DD82238309A
Other languages
German (de)
English (en)
Inventor
Vytautas J Jasys
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DD202435A5 publication Critical patent/DD202435A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
DD82238309A 1981-03-23 1982-03-19 Verbessertes verfahren zur herstellung von penicillansaeureestern DD202435A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24648281A 1981-03-23 1981-03-23
US06/341,081 US4381263A (en) 1981-03-23 1982-01-25 Process for the preparation of penicillanic acid esters

Publications (1)

Publication Number Publication Date
DD202435A5 true DD202435A5 (de) 1983-09-14

Family

ID=26938011

Family Applications (2)

Application Number Title Priority Date Filing Date
DD82238309A DD202435A5 (de) 1981-03-23 1982-03-19 Verbessertes verfahren zur herstellung von penicillansaeureestern
DD82251832A DD209835A5 (de) 1981-03-23 1982-03-19 Verbessertes verfahren zur herstellung von penicillansaeureestern

Family Applications After (1)

Application Number Title Priority Date Filing Date
DD82251832A DD209835A5 (de) 1981-03-23 1982-03-19 Verbessertes verfahren zur herstellung von penicillansaeureestern

Country Status (27)

Country Link
US (1) US4381263A (pt)
EP (1) EP0061284B1 (pt)
KR (1) KR860001367B1 (pt)
AU (1) AU535417B2 (pt)
BG (2) BG38938A3 (pt)
CA (1) CA1182107A (pt)
CS (1) CS228920B2 (pt)
DD (2) DD202435A5 (pt)
DE (1) DE3270720D1 (pt)
DK (1) DK161969C (pt)
EG (1) EG15908A (pt)
ES (2) ES510658A0 (pt)
FI (1) FI75165C (pt)
GB (1) GB2095665A (pt)
GR (1) GR75939B (pt)
HU (1) HU189124B (pt)
IE (1) IE52813B1 (pt)
IL (1) IL65309A (pt)
IN (1) IN157712B (pt)
MX (1) MX174205B (pt)
NO (2) NO164598C (pt)
NZ (1) NZ200067A (pt)
PH (2) PH18608A (pt)
PL (1) PL130866B1 (pt)
PT (1) PT74622B (pt)
RO (2) RO87039B1 (pt)
YU (2) YU42762B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4704456A (en) * 1985-11-22 1987-11-03 Pfizer Inc. Process for sultamicillin intermediate
JPH01139584A (ja) * 1987-11-25 1989-06-01 Yoshitomi Pharmaceut Ind Ltd ペニシラン酸化合物の製造法
GB8808701D0 (en) * 1988-04-13 1988-05-18 Erba Carlo Spa Beta-lactam derivatives
DE69103003T2 (de) * 1990-04-13 1994-11-03 Pfizer Inc., Groton, Conn. Verfahren für sultamicillinzwischenprodukt.
ES2161602B1 (es) * 1999-04-08 2003-02-16 Asturpharma S A Sintesis de 6-(d-alfa-(bencilidenaminofenilacetamido))penicilanato de 1,1-dioxopenicilanoiloximetilo y analogos. nuevos intermedios para la sintesis de sultamicilina.
CN100384857C (zh) 2003-11-28 2008-04-30 浙江永宁制药厂 耐β-内酰胺酶的头孢菌素酯化合物及其盐
CN112724162B (zh) * 2020-12-28 2022-06-10 华南农业大学 一种阿莫西林-舒巴坦杂合分子的合成方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5248992B1 (pt) * 1971-07-08 1977-12-14
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE50650B1 (en) * 1979-10-11 1986-06-11 Leo Pharm Prod Ltd Method for producing penicillanic acid derivatives

Also Published As

Publication number Publication date
IN157712B (pt) 1986-05-24
IL65309A0 (en) 1982-05-31
AU535417B2 (en) 1984-03-22
YU42904B (en) 1988-12-31
AU8176582A (en) 1982-09-30
EG15908A (en) 1990-08-30
GR75939B (pt) 1984-08-02
IE820658L (en) 1982-09-23
PL235577A1 (en) 1983-03-14
EP0061284B1 (en) 1986-04-23
ES8305771A1 (es) 1983-04-16
PT74622B (en) 1984-11-26
DK127282A (da) 1982-09-24
MX174205B (es) 1994-04-28
PT74622A (en) 1982-04-01
NO164598B (no) 1990-07-16
BG38938A3 (en) 1986-03-14
YU162984A (en) 1985-03-20
KR830009111A (ko) 1983-12-17
RO83707A (ro) 1984-03-15
RO87039B1 (ro) 1985-05-31
DD209835A5 (de) 1984-05-23
PH18608A (en) 1985-08-21
NO164598C (no) 1990-10-24
RO83707B (ro) 1984-03-30
US4381263A (en) 1983-04-26
FI75165C (fi) 1988-05-09
HU189124B (en) 1986-06-30
FI820993L (fi) 1982-09-24
ES8403133A1 (es) 1984-03-01
RO87039A2 (ro) 1985-05-20
BG38940A3 (en) 1986-03-14
YU42762B (en) 1988-12-31
IE52813B1 (en) 1988-03-16
IL65309A (en) 1985-03-31
DK161969C (da) 1992-02-03
NZ200067A (en) 1985-07-12
DK161969B (da) 1991-09-02
PH18487A (en) 1985-08-02
EP0061284A1 (en) 1982-09-29
NO831057L (no) 1982-09-24
PL130866B1 (en) 1984-09-29
DE3270720D1 (en) 1986-05-28
NO820924L (no) 1982-09-24
FI75165B (fi) 1988-01-29
ES510658A0 (es) 1983-04-16
GB2095665A (en) 1982-10-06
KR860001367B1 (ko) 1986-09-17
ES519053A0 (es) 1984-03-01
YU62182A (en) 1985-03-20
CS228920B2 (en) 1984-05-14
CA1182107A (en) 1985-02-05

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ENJ Ceased due to non-payment of renewal fee