CY1110926T1 - Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση - Google Patents

Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση

Info

Publication number
CY1110926T1
CY1110926T1 CY20101101043T CY101101043T CY1110926T1 CY 1110926 T1 CY1110926 T1 CY 1110926T1 CY 20101101043 T CY20101101043 T CY 20101101043T CY 101101043 T CY101101043 T CY 101101043T CY 1110926 T1 CY1110926 T1 CY 1110926T1
Authority
CY
Cyprus
Prior art keywords
pyridines
compositions containing
substituted
rocket
preparation procedure
Prior art date
Application number
CY20101101043T
Other languages
Greek (el)
English (en)
Inventor
Baptiste Ronan
Michel Tabart
Frank Halley
Eric Bacque
Catherine Souaille
Antonio Ugolini
Fabrice Viviani
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36593766&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1110926(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from FR0500555A external-priority patent/FR2880891B1/fr
Priority claimed from FR0507505A external-priority patent/FR2888579A1/fr
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of CY1110926T1 publication Critical patent/CY1110926T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CY20101101043T 2005-01-19 2010-11-18 Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση CY1110926T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0500555A FR2880891B1 (fr) 2005-01-19 2005-01-19 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
FR0507505A FR2888579A1 (fr) 2005-07-13 2005-07-13 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
EP06709121A EP1845978B1 (fr) 2005-01-19 2006-01-18 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation

Publications (1)

Publication Number Publication Date
CY1110926T1 true CY1110926T1 (el) 2015-06-10

Family

ID=36593766

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20101101043T CY1110926T1 (el) 2005-01-19 2010-11-18 Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση

Country Status (24)

Country Link
US (2) US8008322B2 (fr)
EP (1) EP1845978B1 (fr)
JP (1) JP2008527025A (fr)
KR (1) KR20070098923A (fr)
AR (1) AR052357A1 (fr)
AT (1) ATE477799T1 (fr)
AU (1) AU2006207442A1 (fr)
BR (1) BRPI0606504A2 (fr)
CA (1) CA2595041A1 (fr)
CY (1) CY1110926T1 (fr)
DE (1) DE602006016233D1 (fr)
DK (1) DK1845978T3 (fr)
HR (1) HRP20100624T8 (fr)
IL (1) IL184524A0 (fr)
MX (1) MX2007008790A (fr)
PA (1) PA8660301A1 (fr)
PE (1) PE20061119A1 (fr)
PL (1) PL1845978T3 (fr)
PT (1) PT1845978E (fr)
RU (1) RU2375360C2 (fr)
SI (1) SI1845978T1 (fr)
TW (1) TW200639173A (fr)
UY (1) UY29341A1 (fr)
WO (1) WO2006077319A1 (fr)

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FR2889526B1 (fr) 2005-08-04 2012-02-17 Aventis Pharma Sa 7-aza-indazoles substitues, compositions les contenant, procede de fabrication et utilisation
TW200815438A (en) * 2006-06-13 2008-04-01 Bayer Schering Pharma Ag Substituted pyrazolopyridines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
EP1870410A1 (fr) * 2006-06-13 2007-12-26 Bayer Schering Pharma Aktiengesellschaft Arylpyrazolopyridines substituées et leurs sels, compositions pharmaceutiques les comprenant, procédé pour leur préparation et leur utilisation
EP2042500A1 (fr) * 2007-09-21 2009-04-01 Bayer Schering Pharma Aktiengesellschaft Composés de N-[4-(1-H-pyrazolo[3,4-c]pyridin-4-yl)phenyl]-N'-[(hetero)aryl]-urée, compositions pharmaceutiques les contenant, procédés de préparation et leur utilisation comme inbibiteurs de la kinase Tie2
EP1932845A1 (fr) * 2006-12-15 2008-06-18 Bayer Schering Pharma Aktiengesellschaft 3-H-pyrazolopyridines leur sels, compositions pharmaceutiques les contenant, procédé pour leur préparation et leur utilisation
UY30796A1 (es) * 2006-12-15 2008-07-31 Bayer Schering Pharma Ag 3-h-pirazolopiridinas y sales de éstas, composiciones farmacéuticas que las comprenden, métodos para prepararlas, y sus usos
US20110160232A1 (en) * 2007-10-04 2011-06-30 Pingda Ren Certain chemical entities and therapeutic uses thereof
MX2010004819A (es) * 2007-11-02 2010-07-05 Vertex Pharma Derivados de [1h-pirazolo[3,4-b]piridin-4-il]-fenilo o piridin-2-ilo como proteina cinasa c-theta.
EP2070929A1 (fr) 2007-12-11 2009-06-17 Bayer Schering Pharma Aktiengesellschaft Composés d'alkynylaryle et sels correspondants, compositions pharmaceutiques contenant ceux-ci, procédés de préparation de ceux-ci et usage de ceux-ci
EP2242755B1 (fr) 2008-01-08 2012-09-12 Array Biopharma, Inc. Pyrrolopyridines en tant qu'inhibiteurs de kinase
WO2009089359A1 (fr) 2008-01-09 2009-07-16 Array Biopharma Inc. Pyrrolopyridines en tant qu'inhibiteurs de kinase
WO2009114874A2 (fr) * 2008-03-14 2009-09-17 Intellikine, Inc. Inhibiteurs de kinases (benzothiazole) et procédés d’utilisation associés
WO2009114870A2 (fr) * 2008-03-14 2009-09-17 Intellikine, Inc. Inhibiteurs de kinases, et procédés d’utilisation associés
EP2313414B1 (fr) 2008-07-08 2015-11-04 Intellikine, LLC Inhibiteurs de kinases et procédés d'utilisation
US8476431B2 (en) * 2008-11-03 2013-07-02 Itellikine LLC Benzoxazole kinase inhibitors and methods of use
EP2408772B1 (fr) * 2009-03-19 2015-07-01 Medical Research Council Technology Composés
WO2011019780A1 (fr) 2009-08-11 2011-02-17 Bristol-Myers Squibb Company Azaindazoles comme modulateurs de la kinase btk et leur utilisation
US8222416B2 (en) * 2009-12-14 2012-07-17 Hoffmann-La Roche Inc. Azaindole glucokinase activators
GB201008134D0 (en) * 2010-05-14 2010-06-30 Medical Res Council Technology Compounds
CN103209960A (zh) 2010-07-26 2013-07-17 百时美施贵宝公司 用作cyp17抑制剂的磺酰胺化合物
GB201015949D0 (en) * 2010-09-22 2010-11-03 Medical Res Council Technology Compounds
EP2638041B1 (fr) 2010-11-12 2015-07-22 Bristol-Myers Squibb Company Dérivés azaindole substitués
TWI592411B (zh) 2011-02-23 2017-07-21 英特爾立秦有限責任公司 激酶抑制劑之組合及其用途
WO2012162627A1 (fr) * 2011-05-26 2012-11-29 The General Hospital Corporation Traitement de maladies angiogéniques ou vasculaires associées
WO2013024002A1 (fr) * 2011-08-12 2013-02-21 F. Hoffmann-La Roche Ag Composés de pyrazolo[3,4-c]pyridine et procédés d'utilisation
US9085578B2 (en) 2012-02-20 2015-07-21 Takeda Pharmaceutical Company Limited Heterocyclic compound
RU2660429C2 (ru) * 2012-09-28 2018-07-06 Мерк Шарп И Доум Корп. Новые соединения, которые являются ингибиторами erk
MX2015008396A (es) 2012-12-28 2016-04-15 Crystalgenomics Inc Derivados de la 2,3-dihidro-isoindol-1-ona, como inhibidores de la btk quinasa y composiciones farmacéuticas que los incluyen.
TWI629275B (zh) * 2013-03-13 2018-07-11 賽諾菲公司 Ｎ－（４－（氮雜吲唑－６－基）－苯基）－磺醯胺及其作為醫藥之用途
CN103524421B (zh) * 2013-09-29 2015-04-01 镇江蓝德特药业科技有限公司 新型萘脲类衍生物及其医疗应用
KR20200140302A (ko) 2018-04-05 2020-12-15 메르크 파텐트 게엠베하 타입 ii irak 억제제로서 헤테로아릴 화합물 및 이의 용도
UY38349A (es) 2018-08-30 2020-03-31 Array Biopharma Inc Compuestos de pirazolo[3,4-b]piridina como inhibidores de cinasas tam y met
AU2022421952A1 (en) * 2021-12-22 2024-07-04 Anaxis Pharma Pty Ltd Arylsulphonamide compounds

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FR2827603B1 (fr) 2001-07-18 2003-10-17 Oreal Composes derives de diaminopyrazole substitues par un radical heteroaromatique et leur utilisation en teinture d'oxydation des fibres keratiniques
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FR2871158A1 (fr) 2004-06-04 2005-12-09 Aventis Pharma Sa Indazoles substitues, compositions les contenant, procede de fabrication et utilisation
JP5112875B2 (ja) * 2004-10-29 2013-01-09 アボット・ラボラトリーズ 新規なキナーゼ阻害薬
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FR2889526B1 (fr) 2005-08-04 2012-02-17 Aventis Pharma Sa 7-aza-indazoles substitues, compositions les contenant, procede de fabrication et utilisation
WO2007056582A1 (fr) 2005-11-09 2007-05-18 Memory Pharmaceuticals Corporation 1-h-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles et chromones, et leur preparation et utilisations
TW200815438A (en) * 2006-06-13 2008-04-01 Bayer Schering Pharma Ag Substituted pyrazolopyridines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
EP1870410A1 (fr) * 2006-06-13 2007-12-26 Bayer Schering Pharma Aktiengesellschaft Arylpyrazolopyridines substituées et leurs sels, compositions pharmaceutiques les comprenant, procédé pour leur préparation et leur utilisation
TW200815437A (en) * 2006-06-13 2008-04-01 Bayer Schering Pharma Ag Substituted aminopyrazolopyridines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same

Also Published As

Publication number Publication date
IL184524A0 (en) 2007-10-31
TW200639173A (en) 2006-11-16
PA8660301A1 (es) 2006-09-08
DE602006016233D1 (de) 2010-09-30
ATE477799T1 (de) 2010-09-15
KR20070098923A (ko) 2007-10-05
RU2007131274A (ru) 2009-02-27
AU2006207442A1 (en) 2006-07-27
EP1845978A1 (fr) 2007-10-24
PE20061119A1 (es) 2006-11-27
PL1845978T3 (pl) 2011-02-28
US20110190337A1 (en) 2011-08-04
SI1845978T1 (sl) 2010-12-31
EP1845978B1 (fr) 2010-08-18
HRP20100624T8 (en) 2011-01-31
WO2006077319A1 (fr) 2006-07-27
US20080039491A1 (en) 2008-02-14
HRP20100624T1 (hr) 2010-12-31
DK1845978T3 (da) 2010-12-13
RU2375360C2 (ru) 2009-12-10
BRPI0606504A2 (pt) 2009-06-30
AR052357A1 (es) 2007-03-14
MX2007008790A (es) 2007-09-11
US8008322B2 (en) 2011-08-30
UY29341A1 (es) 2006-08-31
CA2595041A1 (fr) 2006-07-27
PT1845978E (pt) 2010-11-29
JP2008527025A (ja) 2008-07-24

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