FR2880891B1 - Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation - Google Patents

Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation

Info

Publication number
FR2880891B1
FR2880891B1 FR0500555A FR0500555A FR2880891B1 FR 2880891 B1 FR2880891 B1 FR 2880891B1 FR 0500555 A FR0500555 A FR 0500555A FR 0500555 A FR0500555 A FR 0500555A FR 2880891 B1 FR2880891 B1 FR 2880891B1
Authority
FR
France
Prior art keywords
manufacture
compositions containing
containing same
substituted pyrazolo
pyridines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0500555A
Other languages
English (en)
Other versions
FR2880891A1 (fr
Inventor
Baptiste Ronan
Michel Tabart
Frank Halley
Eric Bacque
Catherine Souaille
Antonio Ugolini
Fabrice Viviani
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Priority to FR0500555A priority Critical patent/FR2880891B1/fr
Priority to PE2006000065A priority patent/PE20061119A1/es
Priority to DO2006000015A priority patent/DOP2006000015A/es
Priority to ARP060100172A priority patent/AR052357A1/es
Priority to BRPI0606504-0A priority patent/BRPI0606504A2/pt
Priority to MX2007008790A priority patent/MX2007008790A/es
Priority to PT06709121T priority patent/PT1845978E/pt
Priority to RU2007131274/04A priority patent/RU2375360C2/ru
Priority to CA002595041A priority patent/CA2595041A1/fr
Priority to EP06709121A priority patent/EP1845978B1/fr
Priority to AU2006207442A priority patent/AU2006207442A1/en
Priority to JP2007551703A priority patent/JP2008527025A/ja
Priority to PL06709121T priority patent/PL1845978T3/pl
Priority to SI200630831T priority patent/SI1845978T1/sl
Priority to CNA2006800089292A priority patent/CN101146534A/zh
Priority to ES06709121T priority patent/ES2351160T3/es
Priority to DK06709121.5T priority patent/DK1845978T3/da
Priority to TW095101823A priority patent/TW200639173A/zh
Priority to AT06709121T priority patent/ATE477799T1/de
Priority to DE602006016233T priority patent/DE602006016233D1/de
Priority to PCT/FR2006/000114 priority patent/WO2006077319A1/fr
Priority to KR1020077018866A priority patent/KR20070098923A/ko
Priority to UY29341A priority patent/UY29341A1/es
Priority to SV2006002384A priority patent/SV2006002384A/es
Priority to PA20068660301A priority patent/PA8660301A1/es
Publication of FR2880891A1 publication Critical patent/FR2880891A1/fr
Application granted granted Critical
Publication of FR2880891B1 publication Critical patent/FR2880891B1/fr
Priority to IL184524A priority patent/IL184524A0/en
Priority to US11/778,870 priority patent/US8008322B2/en
Priority to HR20100624T priority patent/HRP20100624T8/xx
Priority to CY20101101043T priority patent/CY1110926T1/el
Priority to US13/084,077 priority patent/US20110190337A1/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
FR0500555A 2005-01-19 2005-01-19 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation Expired - Fee Related FR2880891B1 (fr)

Priority Applications (30)

Application Number Priority Date Filing Date Title
FR0500555A FR2880891B1 (fr) 2005-01-19 2005-01-19 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
PE2006000065A PE20061119A1 (es) 2005-01-19 2006-01-16 PIRAZOLO PIRIDINAS SUSTITUIDAS COMO INHIBIDORES DE CINASAS FAK, KDR Y Tie
ARP060100172A AR052357A1 (es) 2005-01-19 2006-01-17 Pirazolo piridinas sustituidas moduladoras de la actividad de quinasas
DO2006000015A DOP2006000015A (es) 2005-01-19 2006-01-17 Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación
DE602006016233T DE602006016233D1 (de) 2005-01-19 2006-01-18 Substituierte pyrazolopyridine, diese enthaltende sowie deren verwendung
PT06709121T PT1845978E (pt) 2005-01-19 2006-01-18 Pirazolo piridinas substituídas, composições que as contêm, processo de preparação e utilização
RU2007131274/04A RU2375360C2 (ru) 2005-01-19 2006-01-18 Замещенные пиразолопиридины, композиции, содержащие их, способ получения и применение
CA002595041A CA2595041A1 (fr) 2005-01-19 2006-01-18 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
EP06709121A EP1845978B1 (fr) 2005-01-19 2006-01-18 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
AU2006207442A AU2006207442A1 (en) 2005-01-19 2006-01-18 Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use
JP2007551703A JP2008527025A (ja) 2005-01-19 2006-01-18 置換されたピラゾロピリジン類、これらを含有する組成物、これらの製造方法及びこれらの使用
PL06709121T PL1845978T3 (pl) 2005-01-19 2006-01-18 Podstawione pirazolopirydyny, kompozycje je zawierające, sposób ich wytwarzania i ich zastosowanie
SI200630831T SI1845978T1 (sl) 2005-01-19 2006-01-18 Substituirani pirazolo piridini, sestavki ki jih vsebujejo, postopki za pripravo in uporabo
CNA2006800089292A CN101146534A (zh) 2005-01-19 2006-01-18 取代吡唑并吡啶,含有它们的组合物,制备方法与用途
ES06709121T ES2351160T3 (es) 2005-01-19 2006-01-18 Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación y utilización.
DK06709121.5T DK1845978T3 (da) 2005-01-19 2006-01-18 Substituerede pyrazolopyridiner, sammensætninger, som indeholder disse, fremgangsmåde til fremstilling heraf, og anvendelse heraf
BRPI0606504-0A BRPI0606504A2 (pt) 2005-01-19 2006-01-18 pirazolo piridinas substituìdas, composições que as contêm, processo de fabricação e utilização
AT06709121T ATE477799T1 (de) 2005-01-19 2006-01-18 Substituierte pyrazolopyridine, diese enthaltende zusammensetzungen, verfahren zur herstellung davon sowie deren verwendung
MX2007008790A MX2007008790A (es) 2005-01-19 2006-01-18 Pirazolo piridinas sustituidas, composiciones que las contienen, metodo de produccion de las mismas, y su uso.
PCT/FR2006/000114 WO2006077319A1 (fr) 2005-01-19 2006-01-18 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation
KR1020077018866A KR20070098923A (ko) 2005-01-19 2006-01-18 치환된 피라졸로피리딘, 그를 함유하는 조성물, 그의 제조방법 및 그의 용도
TW095101823A TW200639173A (en) 2005-01-19 2006-01-18 Substituted pyrazolopyridines, compositions containing same, manufacturing process therefor and use thereof
SV2006002384A SV2006002384A (es) 2005-01-19 2006-01-19 Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion
PA20068660301A PA8660301A1 (es) 2005-01-19 2006-01-19 Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion
UY29341A UY29341A1 (es) 2005-01-19 2006-01-19 Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación
IL184524A IL184524A0 (en) 2005-01-19 2007-07-10 Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use
US11/778,870 US8008322B2 (en) 2005-01-19 2007-07-17 Substituted pyrazolopyridines, compositions containing them, method for the production thereof, and their use
HR20100624T HRP20100624T8 (en) 2005-01-19 2010-11-18 Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use
CY20101101043T CY1110926T1 (el) 2005-01-19 2010-11-18 Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση
US13/084,077 US20110190337A1 (en) 2005-01-19 2011-04-11 Substituted pyrazolopyridines, compositions containing them, method for the production thereof, and their use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0500555A FR2880891B1 (fr) 2005-01-19 2005-01-19 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation

Publications (2)

Publication Number Publication Date
FR2880891A1 FR2880891A1 (fr) 2006-07-21
FR2880891B1 true FR2880891B1 (fr) 2007-02-23

Family

ID=35124733

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0500555A Expired - Fee Related FR2880891B1 (fr) 2005-01-19 2005-01-19 Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation

Country Status (5)

Country Link
CN (1) CN101146534A (fr)
DO (1) DOP2006000015A (fr)
ES (1) ES2351160T3 (fr)
FR (1) FR2880891B1 (fr)
SV (1) SV2006002384A (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2464647B1 (fr) 2009-08-11 2016-09-21 Bristol-Myers Squibb Company Azaindoles en tant qe modulateurs du recepteur btk et leur utilisation
US8673922B2 (en) * 2010-07-15 2014-03-18 Bristol-Myers Squibb Company Azaindazole compounds
GB201015949D0 (en) * 2010-09-22 2010-11-03 Medical Res Council Technology Compounds
EP2638041B1 (fr) * 2010-11-12 2015-07-22 Bristol-Myers Squibb Company Dérivés azaindole substitués
CN103214479A (zh) * 2012-01-18 2013-07-24 武汉东宇生物医药科技有限公司 吡唑类萘脲类酪氨酸激酶抑制剂及其应用
WO2013125543A1 (fr) * 2012-02-20 2013-08-29 武田薬品工業株式会社 Composé hétérocyclique
CN103524421B (zh) * 2013-09-29 2015-04-01 镇江蓝德特药业科技有限公司 新型萘脲类衍生物及其医疗应用
CN104098564A (zh) * 2014-07-30 2014-10-15 天津市斯芬克司药物研发有限公司 一种吡唑并吡啶化合物及其制备方法
CN108117551B (zh) * 2016-11-29 2020-03-27 华东理工大学 取代(1H-吡唑[3,4-b]吡啶)脲类化合物及其抗肿瘤用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL213199B1 (pl) * 2000-08-10 2013-01-31 Pharmacia Italia Spa Zwiazek bicyklo-pirazolowy, sposób wytwarzania go, jego kompozycja farmaceutyczna, oraz kombinatoryczna biblioteka chemiczna
EP1534389A2 (fr) * 2002-07-23 2005-06-01 SmithKline Beecham Corporation Pyrazolopyrimidines en tant qu'inhibiteurs de kinases
JP2006501217A (ja) * 2002-08-12 2006-01-12 スージェン・インコーポレーテッド 新規キナーゼ阻害剤としての3−ピロリル−ピリドピラゾールおよび3−ピロリル−インダゾール
UA81453C2 (en) * 2003-02-27 2008-01-10 Pyrazolopyridine derivates
WO2005000813A1 (fr) * 2003-05-30 2005-01-06 Imclone Systems Incorporated Derives d'heteroarylamino-phenylcetone et leur utilisation en tant qu'inhibiteurs de kinases

Also Published As

Publication number Publication date
DOP2006000015A (es) 2006-07-31
ES2351160T3 (es) 2011-02-01
SV2006002384A (es) 2006-08-25
FR2880891A1 (fr) 2006-07-21
CN101146534A (zh) 2008-03-19

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Year of fee payment: 11

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Effective date: 20160930