FR2880891B1 - Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation - Google Patents
Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisationInfo
- Publication number
- FR2880891B1 FR2880891B1 FR0500555A FR0500555A FR2880891B1 FR 2880891 B1 FR2880891 B1 FR 2880891B1 FR 0500555 A FR0500555 A FR 0500555A FR 0500555 A FR0500555 A FR 0500555A FR 2880891 B1 FR2880891 B1 FR 2880891B1
- Authority
- FR
- France
- Prior art keywords
- manufacture
- compositions containing
- containing same
- substituted pyrazolo
- pyridines
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Priority Applications (30)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0500555A FR2880891B1 (fr) | 2005-01-19 | 2005-01-19 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
PE2006000065A PE20061119A1 (es) | 2005-01-19 | 2006-01-16 | PIRAZOLO PIRIDINAS SUSTITUIDAS COMO INHIBIDORES DE CINASAS FAK, KDR Y Tie |
ARP060100172A AR052357A1 (es) | 2005-01-19 | 2006-01-17 | Pirazolo piridinas sustituidas moduladoras de la actividad de quinasas |
DO2006000015A DOP2006000015A (es) | 2005-01-19 | 2006-01-17 | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación |
DE602006016233T DE602006016233D1 (de) | 2005-01-19 | 2006-01-18 | Substituierte pyrazolopyridine, diese enthaltende sowie deren verwendung |
PT06709121T PT1845978E (pt) | 2005-01-19 | 2006-01-18 | Pirazolo piridinas substituídas, composições que as contêm, processo de preparação e utilização |
RU2007131274/04A RU2375360C2 (ru) | 2005-01-19 | 2006-01-18 | Замещенные пиразолопиридины, композиции, содержащие их, способ получения и применение |
CA002595041A CA2595041A1 (fr) | 2005-01-19 | 2006-01-18 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
EP06709121A EP1845978B1 (fr) | 2005-01-19 | 2006-01-18 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
AU2006207442A AU2006207442A1 (en) | 2005-01-19 | 2006-01-18 | Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use |
JP2007551703A JP2008527025A (ja) | 2005-01-19 | 2006-01-18 | 置換されたピラゾロピリジン類、これらを含有する組成物、これらの製造方法及びこれらの使用 |
PL06709121T PL1845978T3 (pl) | 2005-01-19 | 2006-01-18 | Podstawione pirazolopirydyny, kompozycje je zawierające, sposób ich wytwarzania i ich zastosowanie |
SI200630831T SI1845978T1 (sl) | 2005-01-19 | 2006-01-18 | Substituirani pirazolo piridini, sestavki ki jih vsebujejo, postopki za pripravo in uporabo |
CNA2006800089292A CN101146534A (zh) | 2005-01-19 | 2006-01-18 | 取代吡唑并吡啶,含有它们的组合物,制备方法与用途 |
ES06709121T ES2351160T3 (es) | 2005-01-19 | 2006-01-18 | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación y utilización. |
DK06709121.5T DK1845978T3 (da) | 2005-01-19 | 2006-01-18 | Substituerede pyrazolopyridiner, sammensætninger, som indeholder disse, fremgangsmåde til fremstilling heraf, og anvendelse heraf |
BRPI0606504-0A BRPI0606504A2 (pt) | 2005-01-19 | 2006-01-18 | pirazolo piridinas substituìdas, composições que as contêm, processo de fabricação e utilização |
AT06709121T ATE477799T1 (de) | 2005-01-19 | 2006-01-18 | Substituierte pyrazolopyridine, diese enthaltende zusammensetzungen, verfahren zur herstellung davon sowie deren verwendung |
MX2007008790A MX2007008790A (es) | 2005-01-19 | 2006-01-18 | Pirazolo piridinas sustituidas, composiciones que las contienen, metodo de produccion de las mismas, y su uso. |
PCT/FR2006/000114 WO2006077319A1 (fr) | 2005-01-19 | 2006-01-18 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
KR1020077018866A KR20070098923A (ko) | 2005-01-19 | 2006-01-18 | 치환된 피라졸로피리딘, 그를 함유하는 조성물, 그의 제조방법 및 그의 용도 |
TW095101823A TW200639173A (en) | 2005-01-19 | 2006-01-18 | Substituted pyrazolopyridines, compositions containing same, manufacturing process therefor and use thereof |
SV2006002384A SV2006002384A (es) | 2005-01-19 | 2006-01-19 | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion |
PA20068660301A PA8660301A1 (es) | 2005-01-19 | 2006-01-19 | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricacion y utilizacion |
UY29341A UY29341A1 (es) | 2005-01-19 | 2006-01-19 | Pirazolo piridinas sustituidas, composiciones que las contienen, procedimiento de fabricación |
IL184524A IL184524A0 (en) | 2005-01-19 | 2007-07-10 | Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use |
US11/778,870 US8008322B2 (en) | 2005-01-19 | 2007-07-17 | Substituted pyrazolopyridines, compositions containing them, method for the production thereof, and their use |
HR20100624T HRP20100624T8 (en) | 2005-01-19 | 2010-11-18 | Substituted pyrazolo-pyridines, compositions containing them, method for the production thereof, and their use |
CY20101101043T CY1110926T1 (el) | 2005-01-19 | 2010-11-18 | Υποκατεστημενες πυραζολο πυριδινες, συνθεσεις που τις περιεχουν, διαδικασια παρασκευης και χρηση |
US13/084,077 US20110190337A1 (en) | 2005-01-19 | 2011-04-11 | Substituted pyrazolopyridines, compositions containing them, method for the production thereof, and their use |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0500555A FR2880891B1 (fr) | 2005-01-19 | 2005-01-19 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2880891A1 FR2880891A1 (fr) | 2006-07-21 |
FR2880891B1 true FR2880891B1 (fr) | 2007-02-23 |
Family
ID=35124733
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0500555A Expired - Fee Related FR2880891B1 (fr) | 2005-01-19 | 2005-01-19 | Pyrazolo pyridines substituees, compositions les contenant, procede de fabrication et utilisation |
Country Status (5)
Country | Link |
---|---|
CN (1) | CN101146534A (fr) |
DO (1) | DOP2006000015A (fr) |
ES (1) | ES2351160T3 (fr) |
FR (1) | FR2880891B1 (fr) |
SV (1) | SV2006002384A (fr) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2464647B1 (fr) | 2009-08-11 | 2016-09-21 | Bristol-Myers Squibb Company | Azaindoles en tant qe modulateurs du recepteur btk et leur utilisation |
US8673922B2 (en) * | 2010-07-15 | 2014-03-18 | Bristol-Myers Squibb Company | Azaindazole compounds |
GB201015949D0 (en) * | 2010-09-22 | 2010-11-03 | Medical Res Council Technology | Compounds |
EP2638041B1 (fr) * | 2010-11-12 | 2015-07-22 | Bristol-Myers Squibb Company | Dérivés azaindole substitués |
CN103214479A (zh) * | 2012-01-18 | 2013-07-24 | 武汉东宇生物医药科技有限公司 | 吡唑类萘脲类酪氨酸激酶抑制剂及其应用 |
WO2013125543A1 (fr) * | 2012-02-20 | 2013-08-29 | 武田薬品工業株式会社 | Composé hétérocyclique |
CN103524421B (zh) * | 2013-09-29 | 2015-04-01 | 镇江蓝德特药业科技有限公司 | 新型萘脲类衍生物及其医疗应用 |
CN104098564A (zh) * | 2014-07-30 | 2014-10-15 | 天津市斯芬克司药物研发有限公司 | 一种吡唑并吡啶化合物及其制备方法 |
CN108117551B (zh) * | 2016-11-29 | 2020-03-27 | 华东理工大学 | 取代(1H-吡唑[3,4-b]吡啶)脲类化合物及其抗肿瘤用途 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PL213199B1 (pl) * | 2000-08-10 | 2013-01-31 | Pharmacia Italia Spa | Zwiazek bicyklo-pirazolowy, sposób wytwarzania go, jego kompozycja farmaceutyczna, oraz kombinatoryczna biblioteka chemiczna |
EP1534389A2 (fr) * | 2002-07-23 | 2005-06-01 | SmithKline Beecham Corporation | Pyrazolopyrimidines en tant qu'inhibiteurs de kinases |
JP2006501217A (ja) * | 2002-08-12 | 2006-01-12 | スージェン・インコーポレーテッド | 新規キナーゼ阻害剤としての3−ピロリル−ピリドピラゾールおよび3−ピロリル−インダゾール |
UA81453C2 (en) * | 2003-02-27 | 2008-01-10 | Pyrazolopyridine derivates | |
WO2005000813A1 (fr) * | 2003-05-30 | 2005-01-06 | Imclone Systems Incorporated | Derives d'heteroarylamino-phenylcetone et leur utilisation en tant qu'inhibiteurs de kinases |
-
2005
- 2005-01-19 FR FR0500555A patent/FR2880891B1/fr not_active Expired - Fee Related
-
2006
- 2006-01-17 DO DO2006000015A patent/DOP2006000015A/es unknown
- 2006-01-18 CN CNA2006800089292A patent/CN101146534A/zh active Pending
- 2006-01-18 ES ES06709121T patent/ES2351160T3/es active Active
- 2006-01-19 SV SV2006002384A patent/SV2006002384A/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DOP2006000015A (es) | 2006-07-31 |
ES2351160T3 (es) | 2011-02-01 |
SV2006002384A (es) | 2006-08-25 |
FR2880891A1 (fr) | 2006-07-21 |
CN101146534A (zh) | 2008-03-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 11 |
|
ST | Notification of lapse |
Effective date: 20160930 |