CS68791A3 - Novel 1-carboxalkylquinoline-2,3(1h,4h)dione compounds, process for their preparation and use - Google Patents
Novel 1-carboxalkylquinoline-2,3(1h,4h)dione compounds, process for their preparation and use Download PDFInfo
- Publication number
- CS68791A3 CS68791A3 CS91687A CS68791A CS68791A3 CS 68791 A3 CS68791 A3 CS 68791A3 CS 91687 A CS91687 A CS 91687A CS 68791 A CS68791 A CS 68791A CS 68791 A3 CS68791 A3 CS 68791A3
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- compound
- hydrogen
- hydrogen atom
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
- C07D241/52—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
- C07D241/40—Benzopyrazines
- C07D241/44—Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Veterinary Medicine (AREA)
- Anesthesiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK069790A DK69790D0 (da) | 1990-03-16 | 1990-03-16 | Heterocykliske forbindelser, deres fremstilling af anvendelse |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS68791A3 true CS68791A3 (en) | 1992-02-19 |
Family
ID=8096500
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS91687A CS68791A3 (en) | 1990-03-16 | 1991-03-15 | Novel 1-carboxalkylquinoline-2,3(1h,4h)dione compounds, process for their preparation and use |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US5166155A (da) |
| EP (1) | EP0520024B1 (da) |
| JP (1) | JPH05505810A (da) |
| AT (1) | ATE139530T1 (da) |
| AU (1) | AU652560B2 (da) |
| CA (1) | CA2078429A1 (da) |
| CS (1) | CS68791A3 (da) |
| DE (1) | DE69120400T2 (da) |
| DK (2) | DK69790D0 (da) |
| ES (1) | ES2089204T3 (da) |
| FI (1) | FI924118A7 (da) |
| GR (1) | GR3020560T3 (da) |
| HU (1) | HUT62274A (da) |
| IE (1) | IE910685A1 (da) |
| IL (1) | IL97405A (da) |
| NO (1) | NO179949C (da) |
| NZ (1) | NZ237431A (da) |
| PT (1) | PT97047B (da) |
| WO (1) | WO1991013878A1 (da) |
| ZA (1) | ZA911779B (da) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT101004B (pt) * | 1991-10-26 | 1999-10-29 | Schering Ag | Derivados da quinoxalina, processo para a sua preparacao e composicoes farmaceuticas que os contem |
| US6057304A (en) * | 1992-10-26 | 2000-05-02 | Schering Aktiengesellschaft | Quinoxaline-phosphonic acid derivatives |
| PT647137E (pt) * | 1992-06-22 | 2008-11-24 | Univ California | Antagonistas dos receptores da glicina e a sua utilização |
| FR2696466B1 (fr) * | 1992-10-02 | 1994-11-25 | Rhone Poulenc Rorer Sa | Dérivés de 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant. |
| IL109397A0 (en) * | 1993-04-28 | 1994-07-31 | Schering Ag | Quinoxalinedione derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same |
| DE4314592A1 (de) * | 1993-04-28 | 1994-11-03 | Schering Ag | Benzo(f)chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| US5631373A (en) * | 1993-11-05 | 1997-05-20 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon, Eugene Oregon | Alkyl, azido, alkoxy, and fluoro-substituted and fused quinoxalinediones |
| DE4340045A1 (de) * | 1993-11-24 | 1995-06-01 | Basf Ag | Neue Chinoxaline und Arzneimittel daraus |
| IL112235A (en) * | 1994-01-03 | 2000-06-29 | Acea Pharm Inc | 1,4-dihydro-pyrido¬2,3-b¾pyrazine-2,3-dione (5 or 8) oxide derivatives and pharmaceutical compositions containing them |
| DE4428152A1 (de) * | 1994-06-22 | 1996-01-04 | Basf Ag | Neue Amido-chinoxalindione, ihrer Herstellung und Verwendung |
| DE4436852A1 (de) * | 1994-10-14 | 1996-04-18 | Basf Ag | Pyrrolyl-tetrahydrobenzochinoxalindione, ihre Herstellung und Verwendung |
| DE4439492A1 (de) * | 1994-10-25 | 1996-05-02 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| US5559447A (en) * | 1994-11-17 | 1996-09-24 | Cypress Semiconductor | Output buffer with variable output impedance |
| DE19519979A1 (de) * | 1995-05-24 | 1996-11-28 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| DE19521058A1 (de) * | 1995-06-09 | 1996-12-12 | Basf Ag | Verfahren zur Herstellung von Aromaten enthaltenden Polyetherpolyolen |
| DE19545251A1 (de) * | 1995-11-24 | 1997-05-28 | Schering Ag | Neue Chinoxalindionderivate, deren Herstellung und Verwendung in Arzneimitteln |
| GB9604400D0 (en) | 1996-03-01 | 1996-05-01 | Pfizer Ltd | Compounds useful in therapy |
| DE19624808A1 (de) | 1996-06-21 | 1998-01-02 | Basf Ag | Pyrrolylchinoxalindione, ihre Herstellung und Verwendung |
| ATE325128T1 (de) * | 1996-10-24 | 2006-06-15 | Novartis Pharma Gmbh | Substituierte aminoalkanphosphonsäuren |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO179551C (no) * | 1987-11-10 | 1996-10-30 | Novo Nordisk As | Analogifremgangsmåte for fremstilling av terapeutisk virksomme kinoxalinforbindelser |
| DK715888D0 (da) * | 1988-12-22 | 1988-12-22 | Ferrosan As | Quinoxalinforbindelser, deres fremstilling og anvendelse |
| DK716188D0 (da) * | 1988-12-22 | 1988-12-22 | Ferrosan As | Quinoxalinforbindelser, deres fremstilling og anvendelse |
-
1990
- 1990-03-16 DK DK069790A patent/DK69790D0/da not_active Application Discontinuation
-
1991
- 1991-03-01 IE IE068591A patent/IE910685A1/en unknown
- 1991-03-04 IL IL9740591A patent/IL97405A/en not_active IP Right Cessation
- 1991-03-11 ZA ZA911779A patent/ZA911779B/xx unknown
- 1991-03-12 US US07/667,855 patent/US5166155A/en not_active Expired - Fee Related
- 1991-03-14 NZ NZ237431A patent/NZ237431A/xx unknown
- 1991-03-15 AU AU75767/91A patent/AU652560B2/en not_active Ceased
- 1991-03-15 EP EP91906855A patent/EP0520024B1/en not_active Expired - Lifetime
- 1991-03-15 AT AT91906855T patent/ATE139530T1/de not_active IP Right Cessation
- 1991-03-15 FI FI924118A patent/FI924118A7/fi not_active Application Discontinuation
- 1991-03-15 PT PT97047A patent/PT97047B/pt not_active IP Right Cessation
- 1991-03-15 DK DK91906855.1T patent/DK0520024T3/da active
- 1991-03-15 WO PCT/DK1991/000078 patent/WO1991013878A1/en not_active Ceased
- 1991-03-15 DE DE69120400T patent/DE69120400T2/de not_active Expired - Fee Related
- 1991-03-15 CA CA002078429A patent/CA2078429A1/en not_active Abandoned
- 1991-03-15 HU HU922953A patent/HUT62274A/hu unknown
- 1991-03-15 JP JP91506759A patent/JPH05505810A/ja active Pending
- 1991-03-15 CS CS91687A patent/CS68791A3/cs unknown
- 1991-03-15 ES ES91906855T patent/ES2089204T3/es not_active Expired - Lifetime
-
1992
- 1992-09-15 NO NO923586A patent/NO179949C/no unknown
-
1996
- 1996-07-17 GR GR960401929T patent/GR3020560T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ237431A (en) | 1993-09-27 |
| CA2078429A1 (en) | 1991-09-17 |
| GR3020560T3 (en) | 1996-10-31 |
| AU7576791A (en) | 1991-10-10 |
| AU652560B2 (en) | 1994-09-01 |
| IE910685A1 (en) | 1991-09-25 |
| WO1991013878A1 (en) | 1991-09-19 |
| ES2089204T3 (es) | 1996-10-01 |
| EP0520024A1 (en) | 1992-12-30 |
| NO179949C (no) | 1997-01-15 |
| PT97047A (pt) | 1991-10-31 |
| HU9202953D0 (en) | 1992-12-28 |
| HUT62274A (en) | 1993-04-28 |
| FI924118A0 (fi) | 1992-09-15 |
| NO179949B (no) | 1996-10-07 |
| ATE139530T1 (de) | 1996-07-15 |
| NO923586D0 (no) | 1992-09-15 |
| PT97047B (pt) | 1998-07-31 |
| IL97405A (en) | 1995-12-08 |
| IL97405A0 (en) | 1992-06-21 |
| NO923586L (no) | 1992-09-15 |
| FI924118L (fi) | 1992-09-15 |
| EP0520024B1 (en) | 1996-06-19 |
| DK69790D0 (da) | 1990-03-16 |
| DE69120400D1 (de) | 1996-07-25 |
| ZA911779B (en) | 1991-12-24 |
| US5166155A (en) | 1992-11-24 |
| DE69120400T2 (de) | 1996-12-19 |
| DK0520024T3 (da) | 1996-10-14 |
| FI924118A7 (fi) | 1992-09-15 |
| JPH05505810A (ja) | 1993-08-26 |
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