CS215064B2 - Method of making the derivatives of the thiadiazolotetrahydro-isochiline - Google Patents
Method of making the derivatives of the thiadiazolotetrahydro-isochiline Download PDFInfo
- Publication number
- CS215064B2 CS215064B2 CS804525A CS452580A CS215064B2 CS 215064 B2 CS215064 B2 CS 215064B2 CS 804525 A CS804525 A CS 804525A CS 452580 A CS452580 A CS 452580A CS 215064 B2 CS215064 B2 CS 215064B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- acid
- chloride
- mixture
- derivatives
- mol
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/04—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/06—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with the ring nitrogen atom acylated by carboxylic or carbonic acids, or with sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS81908A CS215065B2 (cs) | 1979-07-02 | 1981-02-06 | Způsob výroby derivátů oxadiazolotetrahydroisochinolinu |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5434379A | 1979-07-02 | 1979-07-02 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS215064B2 true CS215064B2 (en) | 1982-07-30 |
Family
ID=21990408
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS804525A CS215064B2 (en) | 1979-07-02 | 1980-06-25 | Method of making the derivatives of the thiadiazolotetrahydro-isochiline |
Country Status (30)
| Country | Link |
|---|---|
| EP (1) | EP0023761B1 (ko) |
| JP (1) | JPS5610192A (ko) |
| KR (1) | KR840000396B1 (ko) |
| AR (1) | AR225925A1 (ko) |
| AT (1) | ATE6515T1 (ko) |
| AU (1) | AU531641B2 (ko) |
| BG (1) | BG51250A3 (ko) |
| CA (1) | CA1129415A (ko) |
| CS (1) | CS215064B2 (ko) |
| DD (1) | DD151750A5 (ko) |
| DE (1) | DE3066826D1 (ko) |
| DK (1) | DK151029C (ko) |
| ES (1) | ES492971A0 (ko) |
| FI (1) | FI67221C (ko) |
| GR (1) | GR69206B (ko) |
| HU (1) | HU179382B (ko) |
| IE (1) | IE50290B1 (ko) |
| IL (1) | IL60426A (ko) |
| IN (1) | IN160542B (ko) |
| MX (1) | MX6317E (ko) |
| NO (1) | NO801951L (ko) |
| NZ (1) | NZ194156A (ko) |
| PH (1) | PH17042A (ko) |
| PL (2) | PL230619A1 (ko) |
| PT (1) | PT71458A (ko) |
| RO (1) | RO79707A (ko) |
| SU (1) | SU1072809A3 (ko) |
| YU (1) | YU171180A (ko) |
| ZA (1) | ZA802987B (ko) |
| ZW (1) | ZW14680A1 (ko) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4352809A (en) * | 1981-09-04 | 1982-10-05 | Smithkline Corporation | Method of producing alpha2 antagonism |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3988339A (en) * | 1974-02-08 | 1976-10-26 | Smithkline Corporation | Pharmaceutical compositions and methods of inhibiting phenylethanolamine N-methyltransferase |
| US3939164A (en) * | 1974-02-08 | 1976-02-17 | Smithkline Corporation | 7 AND 8-Halo substituted 1,2,3,4-tetrahydroisoquinoline compounds |
-
1980
- 1980-05-20 ZA ZA00802987A patent/ZA802987B/xx unknown
- 1980-06-25 CS CS804525A patent/CS215064B2/cs unknown
- 1980-06-25 CA CA354,710A patent/CA1129415A/en not_active Expired
- 1980-06-25 PH PH24191A patent/PH17042A/en unknown
- 1980-06-25 JP JP8720980A patent/JPS5610192A/ja active Pending
- 1980-06-26 NZ NZ194156A patent/NZ194156A/xx unknown
- 1980-06-26 PT PT71458A patent/PT71458A/pt unknown
- 1980-06-26 EP EP80302140A patent/EP0023761B1/en not_active Expired
- 1980-06-26 AT AT80302140T patent/ATE6515T1/de not_active IP Right Cessation
- 1980-06-26 AU AU59677/80A patent/AU531641B2/en not_active Ceased
- 1980-06-26 IN IN485/DEL/80A patent/IN160542B/en unknown
- 1980-06-26 DE DE8080302140T patent/DE3066826D1/de not_active Expired
- 1980-06-26 DK DK274280A patent/DK151029C/da not_active IP Right Cessation
- 1980-06-27 IL IL60426A patent/IL60426A/xx unknown
- 1980-06-27 NO NO801951A patent/NO801951L/no unknown
- 1980-06-27 ZW ZW146/80A patent/ZW14680A1/xx unknown
- 1980-06-28 KR KR1019800002551A patent/KR840000396B1/ko active
- 1980-06-30 AR AR281587A patent/AR225925A1/es active
- 1980-06-30 DD DD80222268A patent/DD151750A5/de unknown
- 1980-06-30 IE IE1352/80A patent/IE50290B1/en unknown
- 1980-06-30 RO RO80101552A patent/RO79707A/ro unknown
- 1980-07-01 PL PL23061980A patent/PL230619A1/xx unknown
- 1980-07-01 HU HU80801631A patent/HU179382B/hu unknown
- 1980-07-01 BG BG48339(A patent/BG51250A3/xx unknown
- 1980-07-01 YU YU01711/80A patent/YU171180A/xx unknown
- 1980-07-01 FI FI802112A patent/FI67221C/fi not_active IP Right Cessation
- 1980-07-01 GR GR62330A patent/GR69206B/el unknown
- 1980-07-01 PL PL1980225377A patent/PL127098B1/pl unknown
- 1980-07-01 ES ES492971A patent/ES492971A0/es active Granted
- 1980-07-01 SU SU802942953A patent/SU1072809A3/ru active
- 1980-07-02 MX MX808900U patent/MX6317E/es unknown
Also Published As
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