CS204042B2 - Process for preparing derivatives of oleandomycine and erythromycine - Google Patents

Process for preparing derivatives of oleandomycine and erythromycine Download PDF

Info

Publication number
CS204042B2
CS204042B2 CS79100A CS10079A CS204042B2 CS 204042 B2 CS204042 B2 CS 204042B2 CS 79100 A CS79100 A CS 79100A CS 10079 A CS10079 A CS 10079A CS 204042 B2 CS204042 B2 CS 204042B2
Authority
CS
Czechoslovakia
Prior art keywords
group
deoxy
formula
acid
mixture
Prior art date
Application number
CS79100A
Other languages
Czech (cs)
English (en)
Inventor
Framk Ch Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS204042B2 publication Critical patent/CS204042B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS79100A 1978-01-03 1979-01-03 Process for preparing derivatives of oleandomycine and erythromycine CS204042B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86672278A 1978-01-03 1978-01-03
US05/937,640 US4180654A (en) 1978-01-03 1978-08-29 4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate

Publications (1)

Publication Number Publication Date
CS204042B2 true CS204042B2 (en) 1981-03-31

Family

ID=27127966

Family Applications (1)

Application Number Title Priority Date Filing Date
CS79100A CS204042B2 (en) 1978-01-03 1979-01-03 Process for preparing derivatives of oleandomycine and erythromycine

Country Status (28)

Country Link
US (1) US4180654A (fi)
JP (1) JPS5495585A (fi)
AT (1) AT364457B (fi)
AU (1) AU506684B2 (fi)
CH (1) CH639972A5 (fi)
CS (1) CS204042B2 (fi)
DD (1) DD141026A5 (fi)
DE (2) DE2900118A1 (fi)
DK (1) DK147943C (fi)
ES (2) ES476544A1 (fi)
FI (1) FI68058C (fi)
FR (1) FR2413403A1 (fi)
GB (1) GB2013181B (fi)
GR (1) GR72779B (fi)
HU (1) HU180276B (fi)
IE (1) IE47642B1 (fi)
IL (1) IL56363A (fi)
IN (1) IN150395B (fi)
IT (1) IT1109925B (fi)
LU (1) LU80747A1 (fi)
NL (1) NL176461C (fi)
NO (2) NO146711C (fi)
NZ (1) NZ189274A (fi)
PH (4) PH14745A (fi)
PL (2) PL118573B1 (fi)
PT (1) PT69014A (fi)
SE (2) SE447118B (fi)
YU (2) YU312278A (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6211669Y2 (fi) * 1980-10-06 1987-03-19
JPS5848285U (ja) * 1981-09-26 1983-04-01 コナミ工業株式会社 テ−ブル型テレビゲ−ム機
US4429116A (en) * 1982-12-27 1984-01-31 Pfizer Inc. Alkylated oleandomycin containing compounds
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
JPS62240086A (ja) * 1986-04-12 1987-10-20 株式会社　エ−ス電研 遊技機の前面構造
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
SI9010556B (sl) * 1990-03-21 1998-10-31 Pliva Oleandomicin oksimi in postopek za njihovo pripravo
CA2525455A1 (en) * 2003-05-13 2004-11-25 Glaxo Group Limited Novel 14 and 15 membered-ring compounds
GB0310980D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310992D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310984D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3869445A (en) * 1973-05-03 1975-03-04 Abbott Lab 4{41 -O-sulfonyl erythromycin-9-O-oxime derivatives
US3884902A (en) * 1973-05-04 1975-05-20 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
US4063014A (en) * 1975-06-12 1977-12-13 Abbott Laboratories 4"-O-sulfonyl erythromycin-9-O-oxime derivatives
IE44509B1 (en) * 1976-03-03 1981-12-30 Pfizer Semi-synthetic oleandomycins
US4069379A (en) * 1976-07-08 1978-01-17 Pfizer Inc. Semi-synthetic oleandomycins
US4090017A (en) * 1977-02-04 1978-05-16 Pfizer Inc. 4-Deoxy-4-substituted amino derivatives of oleandomycin
US4085119A (en) * 1977-02-04 1978-04-18 Pfizer Inc. 4-Substituted amino derivatives of oleandomycin

Also Published As

Publication number Publication date
PH15439A (en) 1983-01-18
IT7919013A0 (it) 1979-01-02
NO790006L (no) 1979-07-04
GB2013181A (en) 1979-08-08
HU180276B (en) 1983-02-28
AU506684B2 (en) 1980-01-17
DE2900118A1 (de) 1979-07-05
DK147943C (da) 1985-08-05
FI68058B (fi) 1985-03-29
PT69014A (en) 1979-02-01
IN150395B (fi) 1982-09-25
DK507778A (da) 1979-07-04
AT364457B (de) 1981-10-27
JPS5734280B2 (fi) 1982-07-22
SE8304417L (sv) 1983-08-15
PL118573B1 (en) 1981-10-31
DE2900118C2 (fi) 1987-09-17
IE790005L (en) 1979-07-03
FR2413403B1 (fi) 1982-07-23
DK147943B (da) 1985-01-14
GR72779B (fi) 1983-12-05
YU312278A (en) 1983-01-21
FI68058C (fi) 1985-07-10
IL56363A (en) 1982-12-31
NO147716C (no) 1983-06-01
NO820613L (no) 1979-07-04
AU4298578A (en) 1979-07-12
ES476544A1 (es) 1979-12-01
FR2413403A1 (fr) 1979-07-27
NL176461C (nl) 1985-04-16
NZ189274A (en) 1982-03-23
SE448385B (sv) 1987-02-16
GB2013181B (en) 1982-06-03
ATA2979A (de) 1981-03-15
PH14745A (en) 1981-11-20
NO146711B (no) 1982-08-16
JPS5495585A (en) 1979-07-28
PL212593A1 (pl) 1979-08-27
IT1109925B (it) 1985-12-23
LU80747A1 (fr) 1979-09-07
ES482420A1 (es) 1980-09-01
CH639972A5 (de) 1983-12-15
PH15626A (en) 1983-03-11
US4180654A (en) 1979-12-25
SE7900028L (sv) 1979-07-04
DE2953969C2 (fi) 1987-09-03
FI790004A (fi) 1979-07-04
PL117603B1 (en) 1981-08-31
PH15752A (en) 1983-03-18
SE447118B (sv) 1986-10-27
SE8304417D0 (sv) 1983-08-15
DD141026A5 (de) 1980-04-09
NL7900006A (nl) 1979-07-05
YU213982A (en) 1983-02-28
NO147716B (no) 1983-02-21
NO146711C (no) 1982-11-24
IL56363A0 (en) 1979-03-12
IE47642B1 (en) 1984-05-16

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