ES482420A1 - Un procedimiento para la preparacion de 4-desoxi-4-acilamino-derivados de eritromicilamina. - Google Patents

Un procedimiento para la preparacion de 4-desoxi-4-acilamino-derivados de eritromicilamina.

Info

Publication number
ES482420A1
ES482420A1 ES482420A ES482420A ES482420A1 ES 482420 A1 ES482420 A1 ES 482420A1 ES 482420 A ES482420 A ES 482420A ES 482420 A ES482420 A ES 482420A ES 482420 A1 ES482420 A1 ES 482420A1
Authority
ES
Spain
Prior art keywords
erythromycin
oleandomycin
carbonate
deoxy
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES482420A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES482420A1 publication Critical patent/ES482420A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

1. Un procedimiento para la preparación de 4¿¿-desoxy-4¿¿- acilamino-derivados de eritromicilamina de Fórmula-01 (C): **(Fórmula-01)** donde Z es Fórmula-02: **(Fórmula-02)** cuyo procedimiento consiste en reducir un compuesto de Fórmula-01 (C): **(Fórmula-01)** donde R1 es hidrógeno o hidroxi y Z es el definido anteriormente y, si se desea, formar una sal de adición de ácido farmacéuticamente aceptable.
ES482420A 1978-01-03 1979-07-11 Un procedimiento para la preparacion de 4-desoxi-4-acilamino-derivados de eritromicilamina. Expired ES482420A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86672278A 1978-01-03 1978-01-03
US05/937,640 US4180654A (en) 1978-01-03 1978-08-29 4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate

Publications (1)

Publication Number Publication Date
ES482420A1 true ES482420A1 (es) 1980-09-01

Family

ID=27127966

Family Applications (2)

Application Number Title Priority Date Filing Date
ES476544A Expired ES476544A1 (es) 1978-01-03 1979-01-02 Un procedimiento para la preparacion de 4Ÿ-desoxi-4Ÿ-acila- mino-derivados de oleandomicinaeritromicina y carbonato de eritromicina.
ES482420A Expired ES482420A1 (es) 1978-01-03 1979-07-11 Un procedimiento para la preparacion de 4-desoxi-4-acilamino-derivados de eritromicilamina.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES476544A Expired ES476544A1 (es) 1978-01-03 1979-01-02 Un procedimiento para la preparacion de 4Ÿ-desoxi-4Ÿ-acila- mino-derivados de oleandomicinaeritromicina y carbonato de eritromicina.

Country Status (28)

Country Link
US (1) US4180654A (es)
JP (1) JPS5495585A (es)
AT (1) AT364457B (es)
AU (1) AU506684B2 (es)
CH (1) CH639972A5 (es)
CS (1) CS204042B2 (es)
DD (1) DD141026A5 (es)
DE (2) DE2900118A1 (es)
DK (1) DK147943C (es)
ES (2) ES476544A1 (es)
FI (1) FI68058C (es)
FR (1) FR2413403A1 (es)
GB (1) GB2013181B (es)
GR (1) GR72779B (es)
HU (1) HU180276B (es)
IE (1) IE47642B1 (es)
IL (1) IL56363A (es)
IN (1) IN150395B (es)
IT (1) IT1109925B (es)
LU (1) LU80747A1 (es)
NL (1) NL176461C (es)
NO (2) NO146711C (es)
NZ (1) NZ189274A (es)
PH (4) PH14745A (es)
PL (2) PL117603B1 (es)
PT (1) PT69014A (es)
SE (2) SE447118B (es)
YU (2) YU312278A (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6211669Y2 (es) * 1980-10-06 1987-03-19
JPS5848285U (ja) * 1981-09-26 1983-04-01 コナミ工業株式会社 テ−ブル型テレビゲ−ム機
US4429116A (en) * 1982-12-27 1984-01-31 Pfizer Inc. Alkylated oleandomycin containing compounds
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
JPS62240086A (ja) * 1986-04-12 1987-10-20 株式会社　エ−ス電研 遊技機の前面構造
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
SI9010556B (sl) * 1990-03-21 1998-10-31 Pliva Oleandomicin oksimi in postopek za njihovo pripravo
GB0310984D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310992D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310980D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
PL1628989T3 (pl) * 2003-05-13 2007-05-31 Glaxo Group Ltd Nowe związki o 14- i 15- członowym pierścieniu

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3869445A (en) * 1973-05-03 1975-03-04 Abbott Lab 4{41 -O-sulfonyl erythromycin-9-O-oxime derivatives
US3884902A (en) * 1973-05-04 1975-05-20 Abbott Lab Sulfonyl derivatives of erythromycin
US3884903A (en) * 1973-06-21 1975-05-20 Abbott Lab 4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
US4063014A (en) * 1975-06-12 1977-12-13 Abbott Laboratories 4"-O-sulfonyl erythromycin-9-O-oxime derivatives
IE44509B1 (en) * 1976-03-03 1981-12-30 Pfizer Semi-synthetic oleandomycins
US4069379A (en) * 1976-07-08 1978-01-17 Pfizer Inc. Semi-synthetic oleandomycins
US4085119A (en) * 1977-02-04 1978-04-18 Pfizer Inc. 4-Substituted amino derivatives of oleandomycin
US4090017A (en) * 1977-02-04 1978-05-16 Pfizer Inc. 4-Deoxy-4-substituted amino derivatives of oleandomycin

Also Published As

Publication number Publication date
FI68058C (fi) 1985-07-10
JPS5734280B2 (es) 1982-07-22
IE47642B1 (en) 1984-05-16
ATA2979A (de) 1981-03-15
PL117603B1 (en) 1981-08-31
FI68058B (fi) 1985-03-29
NL7900006A (nl) 1979-07-05
DE2900118C2 (es) 1987-09-17
IE790005L (en) 1979-07-03
SE447118B (sv) 1986-10-27
NO146711C (no) 1982-11-24
FI790004A (fi) 1979-07-04
IL56363A0 (en) 1979-03-12
DK147943B (da) 1985-01-14
SE8304417D0 (sv) 1983-08-15
IL56363A (en) 1982-12-31
AT364457B (de) 1981-10-27
FR2413403B1 (es) 1982-07-23
NO147716C (no) 1983-06-01
DK507778A (da) 1979-07-04
IT1109925B (it) 1985-12-23
LU80747A1 (fr) 1979-09-07
GR72779B (es) 1983-12-05
YU312278A (en) 1983-01-21
PL212593A1 (pl) 1979-08-27
NL176461C (nl) 1985-04-16
DE2953969C2 (es) 1987-09-03
FR2413403A1 (fr) 1979-07-27
GB2013181A (en) 1979-08-08
NZ189274A (en) 1982-03-23
SE8304417L (sv) 1983-08-15
ES476544A1 (es) 1979-12-01
NO147716B (no) 1983-02-21
AU4298578A (en) 1979-07-12
GB2013181B (en) 1982-06-03
DE2900118A1 (de) 1979-07-05
DK147943C (da) 1985-08-05
PH15752A (en) 1983-03-18
PH15626A (en) 1983-03-11
CH639972A5 (de) 1983-12-15
AU506684B2 (en) 1980-01-17
NO146711B (no) 1982-08-16
IT7919013A0 (it) 1979-01-02
HU180276B (en) 1983-02-28
PT69014A (en) 1979-02-01
NO790006L (no) 1979-07-04
SE7900028L (sv) 1979-07-04
CS204042B2 (en) 1981-03-31
SE448385B (sv) 1987-02-16
PH15439A (en) 1983-01-18
JPS5495585A (en) 1979-07-28
PH14745A (en) 1981-11-20
PL118573B1 (en) 1981-10-31
NO820613L (no) 1979-07-04
DD141026A5 (de) 1980-04-09
IN150395B (es) 1982-09-25
US4180654A (en) 1979-12-25
YU213982A (en) 1983-02-28

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970505