CS203166B2 - Method of preparing amino-acetamido-oxadethiacephalosporins substituted in position 7 - Google Patents

Method of preparing amino-acetamido-oxadethiacephalosporins substituted in position 7 Download PDF

Info

Publication number
CS203166B2
CS203166B2 CS775642A CS564277A CS203166B2 CS 203166 B2 CS203166 B2 CS 203166B2 CS 775642 A CS775642 A CS 775642A CS 564277 A CS564277 A CS 564277A CS 203166 B2 CS203166 B2 CS 203166B2
Authority
CS
Czechoslovakia
Prior art keywords
group
formula
substituted
phenyl
alkyl
Prior art date
Application number
CS775642A
Other languages
Czech (cs)
English (en)
Inventor
Mosayuki Narisada
Teruji Tsuji
Mitsuru Yoshioka
Hiromu Matsumura
Yoshio Hamashima
Wataru Nagata
Sadao Hayashi
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Priority to CS782436A priority Critical patent/CS203167B2/cs
Priority to CS782437A priority patent/CS203168B2/cs
Priority to CS782438A priority patent/CS203169B2/cs
Publication of CS203166B2 publication Critical patent/CS203166B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS775642A 1976-09-01 1977-08-29 Method of preparing amino-acetamido-oxadethiacephalosporins substituted in position 7 CS203166B2 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
CS782436A CS203167B2 (cs) 1976-09-01 1978-04-14 Způsob přípravy 7-substltuo váných aminoacetamidooxadethia- cefalosporinů
CS782437A CS203168B2 (cs) 1976-09-01 1978-04-14 Způsob přípravy aminoacetmidooxadethiacefalosporinů substituovaných v poloze 7
CS782438A CS203169B2 (cs) 1976-09-01 1978-04-14 Způsob přípravy aminoacetamidooxadetbiacefalosporinů substituovaných v poloze 7

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP10511776A JPS5331690A (en) 1976-09-01 1976-09-01 Oxadithiacephalosporins

Publications (1)

Publication Number Publication Date
CS203166B2 true CS203166B2 (en) 1981-02-27

Family

ID=14398870

Family Applications (1)

Application Number Title Priority Date Filing Date
CS775642A CS203166B2 (en) 1976-09-01 1977-08-29 Method of preparing amino-acetamido-oxadethiacephalosporins substituted in position 7

Country Status (32)

Country Link
US (1) US4226864A (ru)
JP (1) JPS5331690A (ru)
AR (4) AR221583A1 (ru)
AT (1) AT353964B (ru)
AU (1) AU511254B2 (ru)
BE (1) BE858341A (ru)
BG (1) BG34038A3 (ru)
CA (1) CA1079278A (ru)
CH (1) CH636879A5 (ru)
CS (1) CS203166B2 (ru)
DD (1) DD132872A5 (ru)
DE (1) DE2739448A1 (ru)
DK (1) DK388377A (ru)
ES (1) ES462012A1 (ru)
FI (1) FI64599C (ru)
FR (1) FR2375238A1 (ru)
GB (1) GB1551479A (ru)
GR (1) GR69784B (ru)
HU (1) HU177382B (ru)
IE (1) IE45572B1 (ru)
IL (1) IL52841A (ru)
MX (1) MX4451E (ru)
NL (1) NL190267C (ru)
NZ (1) NZ185018A (ru)
PH (1) PH17509A (ru)
PL (2) PL104618B1 (ru)
PT (1) PT66974B (ru)
RO (1) RO77767A (ru)
SE (1) SE441095B (ru)
SU (4) SU786901A3 (ru)
YU (4) YU40172B (ru)
ZA (1) ZA775154B (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5690088A (en) * 1979-11-02 1981-07-21 Meiji Seika Kaisha Ltd Novel cephalosporin analog compound
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
DE3137038A1 (de) * 1981-09-17 1983-03-24 Bayer Ag, 5090 Leverkusen Ss-lactam antibiotika, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
JPS59104389A (ja) * 1982-12-06 1984-06-16 Shionogi & Co Ltd オキサセファム誘導体
JPS59118789A (ja) * 1982-12-27 1984-07-09 Shionogi & Co Ltd オキサセフエム誘導体、その製法および用途
US4645769A (en) * 1985-03-01 1987-02-24 Merck & Co., Inc. 1-oxa-1-dethia-cephalosporin compounds and antibacterial agent comprising the same
US10954231B2 (en) 2006-10-16 2021-03-23 Bionomics Limited Anxiolytic compounds
AU2007312936B2 (en) 2006-10-16 2013-09-26 Bionomics Limited Novel anxiolytic compounds
WO2009049086A1 (en) 2007-10-09 2009-04-16 Larry Sutton Broad spectrum beta-lactamase inhibitors
AU2012253237B2 (en) 2011-05-12 2015-09-24 Bionomics Limited Methods for preparing naphthyridines

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR208171A1 (es) * 1972-09-29 1976-12-09 Ciba Geigy Ag Procedimiento para la obtencion de nuevos derivados del acido cef-3-em-4-carboxilico
NL178005C (nl) * 1972-11-06 1986-01-02 Merck & Co Inc Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
US4032521A (en) * 1972-12-29 1977-06-28 Merck & Co., Inc. Cephalosporin phosphonic acid, sulfonic acid and sulfonamide compounds
JPS49133593A (ru) * 1973-05-04 1974-12-21
GB1449420A (en) * 1973-11-26 1976-09-15 Sankyo Co 7alpha-methoxycephalosporing derivatives
IL47168A (en) * 1974-05-09 1979-07-25 Toyama Chemical Co Ltd Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
US4110327A (en) * 1974-05-09 1978-08-29 Toyama Chemical Co., Ltd. 2,3 Diketo-piperazinocarbonylamino alkanoic acids and derivatives
US4087424A (en) * 1974-05-09 1978-05-02 Toyama Chemical Co., Ltd. Novel penicillins and cephalosporins and process for producing the same
GB1510794A (en) * 1974-08-06 1978-05-17 Univ Kingston 1-oxacephems and intermediates therefor
GB1486349A (en) * 1974-11-28 1977-09-21 Bayer Ag Beta-lactam antibiotics process for their preparation and their use as medicaments
DE2528077A1 (de) * 1975-06-24 1977-01-20 Bayer Ag Beta-lactamantibiotika, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
US3996218A (en) * 1975-09-08 1976-12-07 E. R. Squibb & Sons, Inc. Oxopyridazinylthiomethyl derivatives of ureidocephalosporins
US4103008A (en) * 1976-04-07 1978-07-25 Ishimaru Toshiyasu 7[2(2,3 Dioxopiperazin-1-yl-carbonylamino)substituted 2 phenylacetamido]-3-2'-thiadiazolyl cephalosporanic acid derivatives
JPS609515B2 (ja) * 1976-08-09 1985-03-11 塩野義製薬株式会社 ３′−ノルオキサセファロスポリン類

Also Published As

Publication number Publication date
SU786901A3 (ru) 1980-12-07
IE45572L (en) 1978-03-01
DK388377A (da) 1978-03-02
FI64599B (fi) 1983-08-31
GR69784B (ru) 1982-07-07
SE441095B (sv) 1985-09-09
GB1551479A (en) 1979-08-30
FR2375238A1 (fr) 1978-07-21
PL104617B1 (pl) 1979-08-31
BG34038A3 (en) 1983-06-15
JPS612672B2 (ru) 1986-01-27
US4226864A (en) 1980-10-07
FR2375238B1 (ru) 1980-07-25
SU812183A3 (ru) 1981-03-07
ES462012A1 (es) 1978-06-01
SU799665A3 (ru) 1981-01-23
AR221583A1 (es) 1981-02-27
CA1079278A (en) 1980-06-10
PH17509A (en) 1984-09-07
IL52841A0 (en) 1977-10-31
PL200534A1 (pl) 1978-05-22
IE45572B1 (en) 1982-10-06
NL190267B (nl) 1993-08-02
DD132872A5 (de) 1978-11-15
AU511254B2 (en) 1980-08-07
FI772582A (fi) 1978-03-02
JPS5331690A (en) 1978-03-25
DE2739448A1 (de) 1978-03-02
CH636879A5 (de) 1983-06-30
AR218951A1 (es) 1980-07-15
NL7709611A (nl) 1978-03-03
SU831079A3 (ru) 1981-05-15
NL190267C (nl) 1994-01-03
ZA775154B (en) 1978-07-26
ATA628177A (de) 1979-05-15
HU177382B (en) 1981-09-28
YU206777A (en) 1982-10-31
BE858341A (fr) 1978-03-01
NZ185018A (en) 1980-05-08
RO77767A (ro) 1981-11-24
FI64599C (fi) 1983-12-12
AR227270A1 (es) 1982-10-15
YU160782A (en) 1983-01-21
AR221609A1 (es) 1981-02-27
MX4451E (es) 1982-05-11
AU2823377A (en) 1979-03-01
YU40172B (en) 1985-08-31
YU160882A (en) 1983-01-21
SE7709736L (sv) 1978-03-02
PL104618B1 (pl) 1979-08-31
AT353964B (de) 1979-12-10
PT66974A (en) 1977-09-01
PT66974B (en) 1979-02-13
IL52841A (en) 1980-10-26
YU160682A (en) 1983-01-21

Similar Documents

Publication Publication Date Title
US3935204A (en) Cephalosporin and pharmaceutical preparations containing the same
US4015000A (en) 6-Acylamino-penam-3-carboxylic and 7-acylamino-3-cephem-4-carboxylic acids
US3954733A (en) Naphthyridine-3-carboxamido-benzylpenicillins and salts thereof
US4396619A (en) Cephalosporin betaines
CS203166B2 (en) Method of preparing amino-acetamido-oxadethiacephalosporins substituted in position 7
US3929779A (en) Aminopyridinium acetyl cephalosporanes
US3719673A (en) Derivatives of 7-aminocephalosporanic acid
US4312982A (en) α-Acylureidocephalosporins and salts and esters thereof
US4758557A (en) Cephalosporin derivatives and bactericides containing the same
US3956292A (en) 7-(α-FUROYLUREIDOARYL AND CYCLOHEXADIENYLACETAMIDO) CEPHALOSPORIN ANTIBIOTICS
JPH0633281B2 (ja) 新規セファロスポリン化合物及び抗菌剤
US3217000A (en) 7-thienylmercaptoacetamido-cephalo-sporanic acid derivatives
JPS5934197B2 (ja) 抗バクテリア剤中間体の合成法
US3928336A (en) 7-{8 D-({60 -amino{60 -phenyl-, 2-thienyl- and 3-thienyl-acetamido){9 -3-(3-methyl-1,2,5-oxadiazol-4-yl)carbonylthiomethyl-3-cephem-4-carboxylic acids
CS232743B2 (en) Method of cephalosporine preparation
JP3363157B2 (ja) 抗菌性の置換７−アシルアミノ−３−（メチルヒドラゾノ）メチルセファロスポリンおよび中間体
CA1137976A (en) Substituted-imidazolidinyl-3-chloro-3- cephem-4-carboxylic acids
KR810000979B1 (ko) 7-치환 아미노 아세타미도 옥사데티아-세팔로스포린류의 제조방법
KR810000893B1 (ko) 7-치환 아미노 아세타미도 옥사데티아-세팔로스포린류의 제조방법
US4160829A (en) Antibacterial 1,2,4-oxadiazolylacetamido cephalosporins
EP0117143A2 (en) Cephalosporin hydroxamic acids, their preparation, antibacterial formulations comprising the same, and their use in combating bacteria
US3879381A (en) 7-(2-Carbamoy L-1-oxaspiro(2,x)alkane-carboxamido) penicillanic acids
US4025509A (en) Aminopyridinium acetyl cephalosporanes
US3734907A (en) 7-(d-(alpha-amino-alpha-phenylacetamido))-3-(5-methyl-1,3,4-oxadiazol7-2-ylthiomethyl)-3-cephem-4-carboxylic acid and salts thereof
US4198503A (en) 3-Carbamoyl substituted-7-ureido substituted cephalosporins