CO6801756A2 - Derivas de tieno [2,3-d] pirimidina y su uso para el tratamiento de la arritimia - Google Patents

Derivas de tieno [2,3-d] pirimidina y su uso para el tratamiento de la arritimia

Info

Publication number
CO6801756A2
CO6801756A2 CO13252150A CO13252150A CO6801756A2 CO 6801756 A2 CO6801756 A2 CO 6801756A2 CO 13252150 A CO13252150 A CO 13252150A CO 13252150 A CO13252150 A CO 13252150A CO 6801756 A2 CO6801756 A2 CO 6801756A2
Authority
CO
Colombia
Prior art keywords
thieno
drifts
arrhythmia
pyrimidine
treatment
Prior art date
Application number
CO13252150A
Other languages
English (en)
Spanish (es)
Inventor
Derek Eward John
John Ford
Original Assignee
Xention Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44071904&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6801756(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Xention Ltd filed Critical Xention Ltd
Publication of CO6801756A2 publication Critical patent/CO6801756A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CO13252150A 2011-04-01 2013-10-24 Derivas de tieno [2,3-d] pirimidina y su uso para el tratamiento de la arritimia CO6801756A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1105659.5A GB201105659D0 (en) 2011-04-01 2011-04-01 Compounds

Publications (1)

Publication Number Publication Date
CO6801756A2 true CO6801756A2 (es) 2013-11-29

Family

ID=44071904

Family Applications (1)

Application Number Title Priority Date Filing Date
CO13252150A CO6801756A2 (es) 2011-04-01 2013-10-24 Derivas de tieno [2,3-d] pirimidina y su uso para el tratamiento de la arritimia

Country Status (42)

Country Link
US (1) US9249155B2 (enExample)
EP (1) EP2694518B1 (enExample)
JP (1) JP5826374B2 (enExample)
KR (1) KR20140023332A (enExample)
CN (1) CN103492392B (enExample)
AP (1) AP2013007198A0 (enExample)
AR (1) AR088735A1 (enExample)
AU (1) AU2012235882B2 (enExample)
BR (1) BR112013025236A2 (enExample)
CA (1) CA2831493A1 (enExample)
CL (1) CL2013002789A1 (enExample)
CO (1) CO6801756A2 (enExample)
CR (1) CR20130488A (enExample)
CU (1) CU24173B1 (enExample)
CY (1) CY1117025T1 (enExample)
DK (1) DK2694518T3 (enExample)
EA (1) EA201301111A1 (enExample)
EC (1) ECSP13012988A (enExample)
ES (1) ES2558563T3 (enExample)
GB (1) GB201105659D0 (enExample)
GT (1) GT201300225A (enExample)
HR (1) HRP20151340T1 (enExample)
HU (1) HUE028438T2 (enExample)
IL (1) IL228555A0 (enExample)
MA (1) MA35064B1 (enExample)
ME (1) ME02314B (enExample)
MX (1) MX335937B (enExample)
NI (1) NI201300100A (enExample)
PE (1) PE20141021A1 (enExample)
PH (1) PH12013501952A1 (enExample)
PL (1) PL2694518T3 (enExample)
PT (1) PT2694518E (enExample)
RS (1) RS54458B1 (enExample)
RU (1) RU2013148627A (enExample)
SG (1) SG193578A1 (enExample)
SI (1) SI2694518T1 (enExample)
SM (1) SMT201500322B (enExample)
TN (1) TN2013000377A1 (enExample)
TW (1) TWI516265B (enExample)
UA (1) UA110131C2 (enExample)
WO (1) WO2012131379A1 (enExample)
ZA (1) ZA201307085B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2922858A4 (en) * 2012-11-20 2016-06-15 Univ Mcgill THIENOPYRIMIDININHIBITORS OF FARNESYL AND / OR GERANYL GERANYL PYROPHOSPHATE SYNTHASE
CN109311868B (zh) 2015-12-22 2022-04-01 尚医治疗有限责任公司 用于治疗癌症和炎性疾病的化合物
CN106727587A (zh) * 2016-11-28 2017-05-31 李娜 一种治疗心律失常的药物组合物
BR112019027640A2 (pt) 2017-06-21 2020-07-07 SHY Therapeutics LLC composto, método para testar a capacidade de um ou mais compostos, método para inibir a função de ras, método para inibir a função de rho, método para inibir a função de rac, composição farmacêutica
US12391705B2 (en) 2018-12-19 2025-08-19 Shy Therapeutics, Llc Compounds that interact with the Ras superfamily for the treatment of cancers, inflammatory diseases, rasopathies, and fibrotic disease

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Also Published As

Publication number Publication date
CU24173B1 (es) 2016-04-25
JP5826374B2 (ja) 2015-12-02
TW201244720A (en) 2012-11-16
RU2013148627A (ru) 2015-05-10
TN2013000377A1 (en) 2015-01-20
IL228555A0 (en) 2013-12-31
BR112013025236A2 (pt) 2019-09-24
US20140206703A1 (en) 2014-07-24
TWI516265B (zh) 2016-01-11
UA110131C2 (ru) 2015-11-25
JP2014509637A (ja) 2014-04-21
EP2694518B1 (en) 2015-10-07
CA2831493A1 (en) 2012-10-04
EA201301111A1 (ru) 2014-02-28
PT2694518E (pt) 2016-02-05
SG193578A1 (en) 2013-10-30
CR20130488A (es) 2013-12-06
HK1193806A1 (zh) 2014-10-03
AU2012235882B2 (en) 2015-08-06
CL2013002789A1 (es) 2014-07-18
WO2012131379A1 (en) 2012-10-04
HRP20151340T1 (hr) 2016-02-26
SI2694518T1 (sl) 2016-02-29
HUE028438T2 (en) 2017-02-28
EP2694518A1 (en) 2014-02-12
PH12013501952A1 (en) 2018-04-11
AU2012235882A1 (en) 2013-05-02
CU20130124A7 (es) 2014-01-29
US9249155B2 (en) 2016-02-02
AP2013007198A0 (en) 2013-10-31
HK1193096A1 (zh) 2014-09-12
CN103492392A (zh) 2014-01-01
PE20141021A1 (es) 2014-08-30
ZA201307085B (en) 2015-04-29
RS54458B1 (sr) 2016-06-30
MX335937B (es) 2016-01-04
AR088735A1 (es) 2014-07-02
NZ615621A (en) 2015-01-30
ME02314B (me) 2016-06-20
SMT201500322B (it) 2016-02-25
NI201300100A (es) 2014-01-07
DK2694518T3 (en) 2015-11-09
CY1117025T1 (el) 2017-04-05
ES2558563T3 (es) 2016-02-05
GT201300225A (es) 2014-12-30
CN103492392B (zh) 2015-11-25
PL2694518T3 (pl) 2016-03-31
GB201105659D0 (en) 2011-05-18
MX2013011301A (es) 2014-04-16
ECSP13012988A (es) 2013-12-31
KR20140023332A (ko) 2014-02-26
MA35064B1 (fr) 2014-04-03

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