CO2018004124A2 - Compuestos heterocíclicos - Google Patents

Compuestos heterocíclicos

Info

Publication number
CO2018004124A2
CO2018004124A2 CONC2018/0004124A CO2018004124A CO2018004124A2 CO 2018004124 A2 CO2018004124 A2 CO 2018004124A2 CO 2018004124 A CO2018004124 A CO 2018004124A CO 2018004124 A2 CO2018004124 A2 CO 2018004124A2
Authority
CO
Colombia
Prior art keywords
heterocyclic compounds
compound
pharmaceutical compositions
compositions containing
therapeutic uses
Prior art date
Application number
CONC2018/0004124A
Other languages
English (en)
Spanish (es)
Inventor
Prabha N Ibrahim
Wayne Spevak
Jiazhong Zhang
Songyuan Shi
Ben Powell
Yan Ma
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57113709&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO2018004124(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of CO2018004124A2 publication Critical patent/CO2018004124A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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  • Diabetes (AREA)
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CONC2018/0004124A 2015-09-21 2018-04-18 Compuestos heterocíclicos CO2018004124A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562221508P 2015-09-21 2015-09-21
PCT/US2016/052538 WO2017053243A1 (en) 2015-09-21 2016-09-19 Heterocyclic compounds and uses thereof

Publications (1)

Publication Number Publication Date
CO2018004124A2 true CO2018004124A2 (es) 2018-08-10

Family

ID=57113709

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2018/0004124A CO2018004124A2 (es) 2015-09-21 2018-04-18 Compuestos heterocíclicos

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US (6) US9771363B2 (https=)
EP (2) EP3353179B1 (https=)
JP (2) JP6863970B2 (https=)
KR (1) KR20180052757A (https=)
CN (2) CN113754656A (https=)
AU (1) AU2016328619B2 (https=)
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US20220356183A1 (en) 2022-11-10
EP3353179A1 (en) 2018-08-01
US20170081326A1 (en) 2017-03-23
RU2018111459A3 (https=) 2020-01-27
US20170362231A1 (en) 2017-12-21
JP2018527398A (ja) 2018-09-20

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