CL2018000730A1 - Compuestos heterocíclicos y usos de los mismos - Google Patents

Compuestos heterocíclicos y usos de los mismos

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Publication number
CL2018000730A1
CL2018000730A1 CL2018000730A CL2018000730A CL2018000730A1 CL 2018000730 A1 CL2018000730 A1 CL 2018000730A1 CL 2018000730 A CL2018000730 A CL 2018000730A CL 2018000730 A CL2018000730 A CL 2018000730A CL 2018000730 A1 CL2018000730 A1 CL 2018000730A1
Authority
CL
Chile
Prior art keywords
heterocyclic compounds
compounds
hereerocyclic
compound
preparation
Prior art date
Application number
CL2018000730A
Other languages
English (en)
Inventor
Prabha N Ibrahim
Wayne Spevak
Jiazhong Zhang
Songyuan Shi
Ben Powell
Yan Ma
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57113709&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2018000730(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of CL2018000730A1 publication Critical patent/CL2018000730A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Abstract

<p>AQUÍ SE PROPORCIONAN COMPUESTOS HETEROCÍCLICOS DE FÓRMULA (I), COMPOSICIONES FARMACÉUTICAS QUE CONTIENEN DICHO COMPUESTO Y SUS USOS TERAPÉUTICOS, MÉTODOS PARA SU PREPARACIÓN, COMPUESTOS INTERMEDIOS, COMPOSICIONES FARMACÉUTICAS QUE CONTIENEN DICHO COMPUESTO Y SUS USOS TERAPÉUTICOS.</p>
CL2018000730A 2015-09-21 2018-03-20 Compuestos heterocíclicos y usos de los mismos CL2018000730A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562221508P 2015-09-21 2015-09-21

Publications (1)

Publication Number Publication Date
CL2018000730A1 true CL2018000730A1 (es) 2018-07-27

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
CL2018000730A CL2018000730A1 (es) 2015-09-21 2018-03-20 Compuestos heterocíclicos y usos de los mismos

Country Status (22)

Country Link
US (6) US9771363B2 (es)
EP (2) EP4071149A3 (es)
JP (2) JP6863970B2 (es)
KR (1) KR20180052757A (es)
CN (2) CN113754656A (es)
AU (1) AU2016328619B2 (es)
BR (1) BR112018005497A2 (es)
CA (2) CA3129180A1 (es)
CL (1) CL2018000730A1 (es)
CO (1) CO2018004124A2 (es)
ES (1) ES2913048T3 (es)
HK (1) HK1255102A1 (es)
IL (1) IL258180B (es)
MX (1) MX2018003432A (es)
MY (1) MY195977A (es)
NZ (1) NZ741112A (es)
PE (1) PE20181093A1 (es)
PH (1) PH12018500591A1 (es)
RU (1) RU2744897C2 (es)
SG (1) SG10201912386RA (es)
TW (1) TWI732785B (es)
WO (1) WO2017053243A1 (es)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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