HK1255102A1 - 雜環化合物及其應用 - Google Patents

雜環化合物及其應用

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Publication number
HK1255102A1
HK1255102A1 HK18114256.0A HK18114256A HK1255102A1 HK 1255102 A1 HK1255102 A1 HK 1255102A1 HK 18114256 A HK18114256 A HK 18114256A HK 1255102 A1 HK1255102 A1 HK 1255102A1
Authority
HK
Hong Kong
Prior art keywords
heterocyclic compounds
heterocyclic
compounds
Prior art date
Application number
HK18114256.0A
Other languages
English (en)
Inventor
Prabha N Ibrahim
Wayne Spevak
Jiazhong Zhang
Songyuan Shi
Ben Powell
Yan Ma
Original Assignee
Plexxikon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57113709&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1255102(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Plexxikon Inc filed Critical Plexxikon Inc
Publication of HK1255102A1 publication Critical patent/HK1255102A1/zh

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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HK18114256.0A 2015-09-21 2018-11-08 雜環化合物及其應用 HK1255102A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562221508P 2015-09-21 2015-09-21
PCT/US2016/052538 WO2017053243A1 (en) 2015-09-21 2016-09-19 Heterocyclic compounds and uses thereof

Publications (1)

Publication Number Publication Date
HK1255102A1 true HK1255102A1 (zh) 2019-08-02

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HK18114256.0A HK1255102A1 (zh) 2015-09-21 2018-11-08 雜環化合物及其應用

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US (6) US9771363B2 (zh)
EP (2) EP3353179B1 (zh)
JP (2) JP6863970B2 (zh)
KR (1) KR20180052757A (zh)
CN (2) CN113754656A (zh)
AU (1) AU2016328619B2 (zh)
BR (1) BR112018005497A2 (zh)
CA (2) CA2999253C (zh)
CL (1) CL2018000730A1 (zh)
CO (1) CO2018004124A2 (zh)
ES (1) ES2913048T3 (zh)
HK (1) HK1255102A1 (zh)
IL (1) IL258180B (zh)
MX (1) MX2018003432A (zh)
MY (1) MY195977A (zh)
NZ (1) NZ741112A (zh)
PE (1) PE20181093A1 (zh)
PH (1) PH12018500591A1 (zh)
RU (1) RU2744897C2 (zh)
SG (1) SG10201912386RA (zh)
TW (1) TWI732785B (zh)
WO (1) WO2017053243A1 (zh)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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