CN1578659A - 过氧化物酶体增殖剂激活的受体(ppar)的调节剂 - Google Patents

过氧化物酶体增殖剂激活的受体(ppar)的调节剂 Download PDF

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Publication number
CN1578659A
CN1578659A CNA028154533A CN02815453A CN1578659A CN 1578659 A CN1578659 A CN 1578659A CN A028154533 A CNA028154533 A CN A028154533A CN 02815453 A CN02815453 A CN 02815453A CN 1578659 A CN1578659 A CN 1578659A
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methyl
alkyl
aryl
phenyl
chemical compound
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Chinese (zh)
Inventor
L·S·戈塞特
J·E·格林
J·R·亨利
W·D·小琼斯
D·P·马休斯
Q·R·沈
D·L·史密斯
J·A·范斯
A·M·瓦肖斯基
M·R·冈萨雷斯－加西亚
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Eli Lilly and Co
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Eli Lilly and Co
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Publication of CN1578659A publication Critical patent/CN1578659A/zh
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    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
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    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Optical Modulation, Optical Deflection, Nonlinear Optics, Optical Demodulation, Optical Logic Elements (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
CNA028154533A 2001-06-07 2002-05-24 过氧化物酶体增殖剂激活的受体(ppar)的调节剂 Pending CN1578659A (zh)

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US29670101P 2001-06-07 2001-06-07
US60/296,701 2001-06-07

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CN1578659A true CN1578659A (zh) 2005-02-09

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US (2) US7282501B2 (https=)
EP (1) EP1401434B1 (https=)
JP (1) JP2005502600A (https=)
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