CN108884051A - 卤素取代的二酮化合物、吡唑化合物及用于制造吡唑化合物的方法 - Google Patents
卤素取代的二酮化合物、吡唑化合物及用于制造吡唑化合物的方法 Download PDFInfo
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- CN108884051A CN108884051A CN201780019913.XA CN201780019913A CN108884051A CN 108884051 A CN108884051 A CN 108884051A CN 201780019913 A CN201780019913 A CN 201780019913A CN 108884051 A CN108884051 A CN 108884051A
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
- C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP16153112 | 2016-01-28 | ||
| EP16153112.4 | 2016-01-28 | ||
| EP16162487 | 2016-03-25 | ||
| EP16162487.9 | 2016-03-25 | ||
| EP16196175.0 | 2016-10-28 | ||
| EP16196175 | 2016-10-28 | ||
| PCT/EP2017/051797 WO2017129759A1 (en) | 2016-01-28 | 2017-01-27 | Halogen substituted diketones, pyrazole compounds and processes for the manufacture of pyrazole compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN108884051A true CN108884051A (zh) | 2018-11-23 |
Family
ID=57960426
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201780019913.XA Pending CN108884051A (zh) | 2016-01-28 | 2017-01-27 | 卤素取代的二酮化合物、吡唑化合物及用于制造吡唑化合物的方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US10829456B2 (enExample) |
| EP (1) | EP3408259A1 (enExample) |
| JP (1) | JP2019504840A (enExample) |
| KR (1) | KR20180108695A (enExample) |
| CN (1) | CN108884051A (enExample) |
| WO (1) | WO2017129759A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN110461822A (zh) * | 2017-03-27 | 2019-11-15 | Agc株式会社 | 含卤素吡唑羧酸及其中间体的制造方法 |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105541716B (zh) | 2015-03-26 | 2024-02-23 | Agc株式会社 | 吡唑衍生物的制造方法 |
| EP3494107A1 (en) * | 2016-08-02 | 2019-06-12 | Solvay Sa | Manufacture of hydrazinyl compounds useful in the manufacture of pyrazole carboxylic acid and derivatives, hydrazinyl compounds and their use |
| JP2020532524A (ja) | 2017-09-04 | 2020-11-12 | ソルヴェイ(ソシエテ アノニム) | ジフルオロアセチルクロリドの製造方法及び製造中間体 |
| CN107987021A (zh) * | 2017-11-24 | 2018-05-04 | 上海应用技术大学 | 一种3-二氟甲基-1-甲基-1h-吡唑-4-羧酸的制备方法 |
| EP3495351A1 (en) * | 2017-12-08 | 2019-06-12 | Solvay Sa | Oxidation of a pyrazolyl ketone compound to the corresponding carboxylic acid |
| EP3728195A1 (en) * | 2017-12-22 | 2020-10-28 | Solvay Sa | Process for the manufacture of pyrazole compounds |
| KR20200103744A (ko) * | 2017-12-22 | 2020-09-02 | 솔베이(소시에떼아노님) | 이미늄 화합물의 제조 방법 및 피라졸 유도체 제조에서의 이의 응용 |
| US20210171468A1 (en) | 2017-12-22 | 2021-06-10 | Solvay Sa | Process for the manufacture of pyrazole carboxylic derivatives and precursors thereof |
| CN110526810A (zh) * | 2018-05-25 | 2019-12-03 | 浙江蓝天环保高科技股份有限公司 | 一种1,1,1-三氟-4-乙氧基戊-3-烯-2-酮的制备方法 |
| EP3605699A1 (en) | 2018-07-31 | 2020-02-05 | Solvay Sa | New components for electrolyte compositions |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0569912A1 (de) * | 1992-05-15 | 1993-11-18 | Hoechst Schering AgrEvo GmbH | 4-Alkyl-substituierte Pyrimidin-5-carboxanilide, Verfahren zu deren Herstellung, diese enthaltende Mittel und deren Verwendung als Fungizide |
| US20050020564A1 (en) * | 2003-05-01 | 2005-01-27 | Atkinson Robert N. | Pyrazole-amides and sulfonamides as sodium channel modulators |
| JP2006273844A (ja) * | 2005-02-17 | 2006-10-12 | Shionogi & Co Ltd | 新規ベンゾジアゼピン類 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4342601A1 (de) | 1993-08-13 | 1995-02-16 | Solvay Fluor & Derivate | Verfahren zur Herstellung von Poly- und Perfluorcarbonsäurechloriden |
| ES2119952T3 (es) | 1993-12-23 | 1998-10-16 | Solvay Fluor & Derivate | Procedimiento para la preparacion de cloruros de acidos polifluoroclorocarboxilicos y perfluorocarboxilicos bajo adicion de cloro. |
| JP3632243B2 (ja) | 1994-07-28 | 2005-03-23 | 旭硝子株式会社 | ジフルオロ酢酸フルオリドおよびジフルオロ酢酸エステルの製造方法 |
| US5905169A (en) | 1995-03-20 | 1999-05-18 | E. I. Du Pont De Nemours And Company | Process for producing polyfluoroacyl compositions |
| US6248923B1 (en) | 1999-09-03 | 2001-06-19 | Eastman Chemical Company | Process for the production of fluorocarboxylic acid anhydrides |
| DE10215292A1 (de) | 2002-02-19 | 2003-08-28 | Bayer Cropscience Ag | Disubstitutierte Pyrazolylcarbocanilide |
| GB0224316D0 (en) | 2002-10-18 | 2002-11-27 | Syngenta Participations Ag | Chemical compounds |
| MXPA05011775A (es) * | 2003-05-01 | 2006-02-17 | Abbott Lab | Sulfonamidas y pirazolamidas como moduladores de canal de sodio. |
| DE10325715A1 (de) | 2003-06-06 | 2004-12-23 | Solvay Fluor Und Derivate Gmbh | Vereinfachte Herstellung von Alkenonen |
| GB0418048D0 (en) | 2004-08-12 | 2004-09-15 | Syngenta Participations Ag | Method for protecting useful plants or plant propagation material |
| DE102005007160A1 (de) | 2005-02-16 | 2006-08-24 | Basf Ag | Pyrazolcarbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen |
| JP2009501742A (ja) | 2005-07-18 | 2009-01-22 | シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト | 殺微生物剤としてのピラゾール−4−カルボキサミド誘導体 |
| BRPI0616238B1 (pt) | 2005-09-16 | 2016-01-19 | Syngenta Ltd | processo para a produção de amidas |
| AU2006308128B2 (en) | 2005-10-25 | 2011-07-28 | Syngenta Crop Protection Ag | Heterocyclic amide derivatives useful as microbiocides |
| BRPI0812958A2 (pt) | 2007-06-15 | 2014-12-09 | Basf Se | Processo para preparar compostos, uso de compostos, e, compostos |
| CN101801906A (zh) | 2007-08-16 | 2010-08-11 | 索尔维公司 | 制备4-氟取代的3-氧代-烷酸酯的方法 |
| CN102015653B (zh) | 2008-05-02 | 2013-09-11 | 巴斯夫欧洲公司 | 制备卤素取代的2-(氨基亚甲基)-3-氧代丁酸酯的方法 |
| CA2729362C (en) | 2008-07-04 | 2016-09-27 | Solvay Sa | Process for the manufacture of alkenones |
| JP2010030970A (ja) | 2008-07-31 | 2010-02-12 | Bayer Cropscience Ag | 殺虫性ベンゼンジカルボキサミド誘導体 |
| EP2184273A1 (de) | 2008-11-05 | 2010-05-12 | Bayer CropScience AG | Halogen-substituierte Verbindungen als Pestizide |
| CN103068805A (zh) | 2010-07-23 | 2013-04-24 | 索尔维公司 | 1-取代-3-氟烷基-吡唑-4-羧酸酯的制备方法 |
| US8987470B2 (en) | 2010-10-27 | 2015-03-24 | Solvay Sa | Process for the preparation of pyrazole-4-carboxamides |
| EP2810931B1 (en) | 2013-06-06 | 2018-04-25 | Solvay SA | Process for the preparation of halogenated carboxylic anhydrides |
| ITMI20132201A1 (it) | 2013-12-23 | 2015-06-24 | Isagro Spa | Processo per la sintesi regioselettiva di pirazoli |
-
2017
- 2017-01-27 JP JP2018539274A patent/JP2019504840A/ja active Pending
- 2017-01-27 KR KR1020187024272A patent/KR20180108695A/ko not_active Withdrawn
- 2017-01-27 EP EP17702825.5A patent/EP3408259A1/en not_active Withdrawn
- 2017-01-27 US US16/071,677 patent/US10829456B2/en not_active Expired - Fee Related
- 2017-01-27 CN CN201780019913.XA patent/CN108884051A/zh active Pending
- 2017-01-27 WO PCT/EP2017/051797 patent/WO2017129759A1/en not_active Ceased
-
2020
- 2020-10-23 US US17/078,555 patent/US20210040043A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0569912A1 (de) * | 1992-05-15 | 1993-11-18 | Hoechst Schering AgrEvo GmbH | 4-Alkyl-substituierte Pyrimidin-5-carboxanilide, Verfahren zu deren Herstellung, diese enthaltende Mittel und deren Verwendung als Fungizide |
| US20050020564A1 (en) * | 2003-05-01 | 2005-01-27 | Atkinson Robert N. | Pyrazole-amides and sulfonamides as sodium channel modulators |
| JP2006273844A (ja) * | 2005-02-17 | 2006-10-12 | Shionogi & Co Ltd | 新規ベンゾジアゼピン類 |
Non-Patent Citations (3)
| Title |
|---|
| ETSUJI OKADA等: "FACILE SYNTHETIC METHODS FOR 3- AND 5-TRIFLUOROMETHY-4-TRIFLUOROACETYL PYRAZOLES AND THEIR CONVERSION INTO PYRAZOLE-4-CARBOXYLIC ACIDS", 《HETEROCYCLES》 * |
| FERNANDA A ROSA等: "N- and C-acylation in β-enamino ketones: structural effects on regiocontrol", 《SYNLETT》 * |
| NORIO OTA等: "A CONVENIENT SYNTHESIS OF FLUORINE-CONTAINING DIHYDROBENZO[b][1,4]DIAZEPINOLS AND ITS APPLICATION TO A SYNTHESIS OF NOVEL N-SULFINYLANILINES", 《HETEROCYCLES》 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN110461822A (zh) * | 2017-03-27 | 2019-11-15 | Agc株式会社 | 含卤素吡唑羧酸及其中间体的制造方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| US10829456B2 (en) | 2020-11-10 |
| WO2017129759A1 (en) | 2017-08-03 |
| KR20180108695A (ko) | 2018-10-04 |
| EP3408259A1 (en) | 2018-12-05 |
| JP2019504840A (ja) | 2019-02-21 |
| US20190031616A1 (en) | 2019-01-31 |
| US20210040043A1 (en) | 2021-02-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PB01 | Publication | ||
| PB01 | Publication | ||
| SE01 | Entry into force of request for substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| WD01 | Invention patent application deemed withdrawn after publication |
Application publication date: 20181123 |
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| WD01 | Invention patent application deemed withdrawn after publication |