CN107743481A - 用于治疗癌症的吲哚胺2,3‑双加氧酶抑制剂 - Google Patents

用于治疗癌症的吲哚胺2,3‑双加氧酶抑制剂 Download PDF

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CN107743481A
CN107743481A CN201680032102.9A CN201680032102A CN107743481A CN 107743481 A CN107743481 A CN 107743481A CN 201680032102 A CN201680032102 A CN 201680032102A CN 107743481 A CN107743481 A CN 107743481A
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optionally substituted
alkyl
mmol
cancer
solvent
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Chinese (zh)
Inventor
J.A.巴罗
E.C.彻尔尼
J.A.马克沃尔德
S.P.塞茨
单伟芳
D.K.威廉斯
S.J.纳拉
S.罗伊
S.桑加维尔
R.K.西斯特拉
S.彻鲁库
S.桑加蒂鲁帕希
Y.肯亚博伊纳
N.普利查拉
A.黄
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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CN109608334A (zh) * 2019-01-11 2019-04-12 盐城通海生物科技有限公司 一种合成4-甲氧基巴豆酸甲酯的方法
WO2021104186A1 (en) * 2019-11-25 2021-06-03 InventisBio Co., Ltd. Novel salts of indoleamine 2,3-dioxygenase inhibitors
CN113214138A (zh) * 2020-02-04 2021-08-06 中国医学科学院药物研究所 苯丙酸类衍生物、及其制法和药物组合物与用途

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SI3105218T1 (sl) 2014-02-13 2019-11-29 Incyte Corp Ciklopropilamini kot inhibitorji LSD1
TWI687419B (zh) 2014-07-10 2020-03-11 美商英塞特公司 作為lsd1抑制劑之咪唑并吡啶及咪唑并吡嗪
TW201613925A (en) 2014-07-10 2016-04-16 Incyte Corp Imidazopyrazines as LSD1 inhibitors
WO2016007722A1 (en) 2014-07-10 2016-01-14 Incyte Corporation Triazolopyridines and triazolopyrazines as lsd1 inhibitors
EP3277689B1 (en) 2015-04-03 2019-09-04 Incyte Corporation Heterocyclic compounds as lsd1 inhibitors
KR20170134980A (ko) * 2015-04-03 2017-12-07 브리스톨-마이어스 스큅 컴퍼니 암의 치료를 위한 인돌아민-2,3-디옥시게나제의 억제제
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