SG11201707948WA - Inhibitors of indoleamine 2,3-dioxygenase for the treatment of cancer - Google Patents

Inhibitors of indoleamine 2,3-dioxygenase for the treatment of cancer

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Publication number
SG11201707948WA
SG11201707948WA SG11201707948WA SG11201707948WA SG11201707948WA SG 11201707948W A SG11201707948W A SG 11201707948WA SG 11201707948W A SG11201707948W A SG 11201707948WA SG 11201707948W A SG11201707948W A SG 11201707948WA SG 11201707948W A SG11201707948W A SG 11201707948WA
Authority
SG
Singapore
Prior art keywords
indoleamine
dioxygenase
inhibitors
cancer
treatment
Prior art date
Application number
SG11201707948WA
Inventor
James Aaron Balog
Emily Charlotte Cherney
Jay A Markwalder
Steven P Seitz
Weifang Shan
David K Williams
Susheel Jethanand Nara
Saumya Roy
Soodamani Thangavel
Ramesh Kumar Sistla
Srinivas Cheruku
Srinivasan Thangathirupathy
Yadagiri Kanyaboina
Nagalakshmi Pulicharla
Audris Huang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55702190&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201707948W(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of SG11201707948WA publication Critical patent/SG11201707948WA/en

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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/40—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/42—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino groups bound to carbon atoms of at least one six-membered aromatic ring and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton with carboxyl groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by saturated carbon chains
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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