CN107714994A - 一种治疗玻璃体出血的药物及其制备方法 - Google Patents
一种治疗玻璃体出血的药物及其制备方法 Download PDFInfo
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Abstract
本发明公开了一种治疗玻璃体出血的药物及其制备方法,其主要是由当归、赤芍、川芎、丹参、黄芩、三七、生地黄、金银花、牡丹皮、白术、红花、泽泻、茯苓、青皮、木香、茺蔚子、甘草、竹叶、党参、黄芪、海藻、昆布、夏枯草、香附按一定重量配比制备而成,本发明药物具有清热凉血,散瘀止痛,止血散瘀,消肿定痛,散风明目的功能,用于治疗玻璃体出血见效快、疗效好,不复发。
Description
技术领域
本发明涉及一种治疗玻璃体出血的药物及其制备方法,属中药领域。
背景技术
玻璃体出血是指玻璃体积血,是由血管性、炎症性、肿瘤、视网膜裂孔等原因造成视力下降的一种常见疾病。本病不仅使屈光介质混浊,妨碍光线达到视网膜,而且能对眼部组织产生严重破坏作用。由于西药治疗副作用大,因此人们对有效治疗玻璃体出血的中药药物存在极大的需求,至今为止,还没有发现关于本发明的有关报道。
发明内容
本发明人依据中医理论的研究和临床试验的反复验证,终于找到了有效治疗玻璃体出血的药物,从而完成了本发明。
本发明的目的就是提供一种有效治疗玻璃体出血的中药组合药物。
本发明的另一目的就是提供了该中药组合药物的制备方法。
本发明药物是选择当归、赤芍、川芎、丹参、黄芩、三七、生地黄、金银花、牡丹皮、白术、红花、泽泻、茯苓、刺蒺藜、车前子、枸杞子、石斛、柴胡、青皮、木香、茺蔚子、甘草、竹叶、党参、黄芪、海藻、昆布、夏枯草、香附进行组合制备的,将这些药物组合使得各药物功效产生协同作用,从而能够有效治疗玻璃体出血。其中选用当归是因为其性味甘辛,温,入心、肝、脾经,有补血和血,调经止痛,润燥滑肠的功能,治月经不调,经闭腹痛,癥瘕结聚,崩漏,血虚头痛,眩晕,痿痹,肠燥难便,赤痢后重,痈疽疮疡,金疮,跌扑损伤。选用赤芍是因为其性味苦,微寒,归肝经,有清热凉血,散瘀止痛的功能,治温毒发狂,吐血衄血,目赤肿痛,肝郁胁痛,经闭痛经,癎瘕腹痛,跌扑损伤,痈肿疮疡。选用川芎是因为其性味辛,温,入肝、胆经,有行气开郁,祛风燥湿,活血止痛的功能,治风冷头痛旋晕,胁痛腹疼,寒痹筋挛,经闭,难产,产后瘀阻块痛,痈疽疮疡。选用丹参是因为其性味苦,微温,入心、肝经,有活血祛痰,安神宁心,排脓,止痛的功能,治心绞痛,月经不调,痛经,经闭,血崩带下,癥瘕,积聚,瘀血腹痛,骨节疼痛,惊悸不眠,恶疮肿毒。选用黄芩是因为其性味苦寒,入心肺、胆、大肠经,有泻实火,除湿热,止血安胎的功能,治壮热烦渴,肺热咳嗽。选用三七是因为其性味甘微苦,温,入肝、胃、大肠经,有止血,散瘀,消肿,定痛的功能,治吐血,咳血,衄血,便血,血痢,崩漏,癥瘕,产后血晕,恶露不下,跌扑瘀血,外伤出血,痈肿疼痛。选用生地黄是因为其性味甘,寒,归心、肝、肾经,有清热凉血,养阴,生津的功能,治热病烦渴,阴虚内热,骨蒸劳热,内热消渴,吐血,衄血,发斑发疹。选用金银花是因为其性味甘,寒,入肺、胃经,有清热,解毒的功能,治温病发热,热毒血痢,痈疡,肿毒,瘰疬,痔漏。选用牡丹皮是因为其性味辛苦,凉,入心、肝、肾经,有清热,凉血,和血,消瘀的功能,治热入血分,发斑,惊癎,吐、衄、便血,骨蒸劳热,经闭,癥瘕,痈疡,扑损。选用白术是因为其性味苦甘,温,入脾、胃经,有补脾,益胃,燥湿,和中的功能,治脾胃气弱,不思饮食,倦怠少气,虚胀,泄泻,痰饮,水肿,黄疸,湿痹,小便不利,头晕,自汗,胎气不安。选用红花是因为其性味辛,温,入心、肝经,有活血通经,去瘀止痛的功能,治经闭,癥瘕,难产,死胎,产后恶露不行,瘀血作痛,痈肿,跌扑损伤。选用泽泻是因为其性味甘,寒,入膀胱经,有利水,渗湿,泄热的功能,治小便不利,水肿肛满,呕吐,泻痢,痰饮,脚气,淋病,尿血。选用茯苓是因为其性味甘淡,平,入心、脾、肺经,有渗湿利水,益脾和胃,宁心安神的功能,治小便不利水肿胀痛,痰饮咳逆,呕哕,泄泻,遗精,淋浊,惊悸,健忘。选用刺蒺藜是因为其性味苦辛,温,入肝、肺经,有散风,明目,下气,行血的功能,治头痛,身痒,目赤肿翳,胸满,咳逆,癥瘕,乳难,痈疽,瘰疬。选用车前子是因为其性味甘,寒,入肾、膀胱经,有利水,清热,明目,祛痰的功能,治小便不通,淋浊,带下,尿血,暑湿泻痢,咳嗽多痰,湿痹,目赤障翳。选用枸杞子是因为其性味甘,平,有滋肾,润肺,补肝,明目的功能,治肝肾阴亏,腰膝酸软,头晕目眩,目昏多泪,虚劳咳嗽,消渴,遗精。选用石斛是因为其性味甘淡微咸,寒,入有、肺、肾经,有生津益胃,清热养阴的功能,治热病伤津,口干烦喝,病后虚热,阴伤目暗。选用柴胡是因为其性味苦,凉,入肝、胆经,有和解表里,疏肝,升阳的功能,治寒热往来,胸满胁痛,口苦耳聋,头痛目眩,疟疾,下利脱肛,月经不调,子宫下垂。选用青皮是因为其性味苦辛,微温,入肝、胆经,有疏肝破气,散结消痰的功能,治胸胁胃脘疼痛,疝气,食积,乳肿,乳核,久疟癖块。选用木香是因为其性味辛苦,温,入肺、肝、脾经,有行气止痛,温中和胃的功能,治中寒气滞,胸腹胀痛,呕吐,泄泻,下痢里急后重,寒疝。选用茺蔚子是因为其性味甘辛,凉,入心胞、肝经,有活血调经,疏风清热的功能,治妇女月经不调,崩中带下,产后瘀血作痛,肝热头痛,目赤肿痛,或生翳膜。选用甘草是因为其性味甘平,入脾、胃、肺经,有和中缓急,润肺,解毒,调和诸药的功能,炙用治脾胃虚弱,食少,腹痛便溏,劳倦发热,肺痿咳嗽,心悸,惊痈,生用治咽喉肿痛,消化性溃疡,痈疽疮疡,解药毒及食物中毒。选用竹叶是因为其性味甘淡,寒,入心、肺、胆、胃经,有清热除烦,生津利尿的功能,治热病烦喝,小儿惊癎,咳逆吐衄,面赤,小便短赤,口糜舌疮。选用党参是因为其性味甘,平,入手、足太阴经气分,有补中益气,生津的功能,治脾胃虚弱,气血两亏,体倦无力,食少,口渴,久泻,脱肛。选用黄芪是因为其性味甘,微温,入肺、脾经,生用有益卫固表,利水消肿,托毒,生肌的功能,治自汗,盗汗,血痹,浮肿,痈疽不溃或溃久敛;炙用有补中益的功能,治内伤劳倦,脾虚泄泻,脱肛,气虚血脱,崩带及一切气衰血虚之症。选用海藻是因为其性味苦咸,寒,入肺、脾、肾经,有软坚,消痰,利水,泄热的功能,治瘰疬,瘿瘤,积聚,水肿,脚气,睾丸肿痛。选用昆布是因为其性味咸,寒,入胃经,有软坚,行水的功能,治瘰疬,瘿瘤,噎膈,水肿,睾丸肿痛,带下。选用夏枯草是因为其性味苦辛,寒,入肝、胆经,有清肝,散结的功能,治瘰疬,瘿瘤,乳痈,乳癌,目珠夜痛,羞明流泪,头目眩晕,口眼歪斜,筋骨疼痛,肺结核,急性黄疸型传染性肝炎,血崩,带下。选用香附是因为其性味辛微苦干,平,入肝、三焦经,有理气解郁,止痛调经的功能,治肝胃不和,气郁不舒,胸腹胁肋胀痛,痰饮痞满,月经不调,崩漏带下。
具体实施方式
本发明组分的药物用量也是发明人经过大量摸索总结得出的,各组分的用量在下述重量范围内都具有较好的疗效:
当归10-14克,赤芍10-14克,川芎10-14克,丹参10-14克,黄芩10-14克,三七15-25克,生地黄10-20克,金银花10-20克,牡丹皮10-20克,白术10-20克,红花10-20克,泽泻5-15克,茯苓5-15克,刺蒺藜5-15克,车前子5-15克,枸杞子15-20克,石斛5-15克,柴胡5-15克,青皮5-15克,木香4-8克,茺蔚子5-15克,甘草10-15克,竹叶5-15克,党参5-15克,黄芪5-15克,海藻5-15克,昆布5-15克,夏枯草5-15克,香附5-15克。
优选为:
当归12克,赤芍12克,川芎12克,丹参12克,黄芩12克,三七20克,生地黄15克,金银花15克,牡丹皮15克,白术15克,红花15克,泽泻10克,茯苓10克,刺蒺藜10克,车前子10克,枸杞子15克,石斛10克,柴胡10克,青皮10克,木香6克,茺蔚子10克,甘草12克,竹叶10克,党参10克,黄芪10克,海藻10克,昆布10克,夏枯草10克,香附10克。
本发明药物的制备方法如下
一、备料
1、当归:拣去杂质,洗净,闷润,稍晾至内外湿度适宜时,切片晒干;
2、赤芍:取原药材,除去杂质,大小分档,洗净,润透,切薄片,干燥,筛去碎屑;
3、川芎:拣去杂质,分开大、小个,用水浸泡,晒晾,闷润后切片,干燥;
4、丹参:拣净杂质,除去根茎,洗净,捞出,润透后切片,晾干;
5、黄芩:拣去杂质,除去残茎,用凉水浸润或置开水中稍浸捞出,切片,晒干;
6、三七:拣净杂质,捣碎,研末或润透后切片晒干;
7、生地黄:除去杂质,洗净,稍润,切厚片,干燥,筛去碎屑;
8、金银花:筛去泥沙,拣净杂质;
9、牡丹皮:拣去杂质,除去木心,洗净,润透,切片,晾干;
10、白术:拣净杂质,用水浸泡,泡后捞出,润透,切片,晒干;
11、红花:拣净杂质,除去茎叶、蒂头,晒干;
12、泽泻:拣去杂质,大小分档,用水浸泡至八成透,捞出,晒凉,闷润至内外湿度均匀,切片,晒干;
13、茯苓:用水浸泡,洗净捞出,闷透后,切片,晒干;
14、刺蒺藜:漂去泥沙,除净残留的硬刺;
15、车前子:拣去杂质,筛去泥屑,空粒;
16、枸杞子:簸净杂质,摘去残留的梗和蒂;
17、石斛:取干燥的石斛,用水泡约至八成透,焖润,除去残根及黑枝,切段,撞去薄膜,晒干;
18、柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,随即晒干;
19、青皮:拣净杂质,用水浸泡,捞出,润透,切片,晒干;
20、木香:将原生药放清水内洗净,捞出,闷润12—24小时使软,切片,晒干;
21、茺蔚子:果实成熟时割取全株,晒干,打下果实,拣去枝叶,筛净杂质;
22、甘草:拣去杂质,洗净,用水浸泡至八成透时,捞出,润透,切片,晾干;
23、竹叶:拣净杂质,除去梗叶,晾干;
24、党参:洗净泥沙后润透去芦,切片或切段,晒干;
25、黄芪:拣净杂质,除去残留的根头和空心较大的根,用水浸泡,捞出,润透后及时切片,晒干;
26、海藻:拣去杂质,用水略漂,稍晾,切段,晒干;
27、昆布:拣去杂质,用水漂净,切成宽丝,晾干;
28、夏枯草:取原药材,除去枝梗、叶片及杂质,筛去灰屑;
29、香附:拣去杂质,碾成碎粒,簸去细毛及细末。
二、制备
1、将所述重量的当归、赤芍、川芎、丹参、黄芩、三七、生地黄、金银花、牡丹皮、白术、红花、泽泻、茯苓、刺蒺藜、车前子、枸杞子、石斛、柴胡、青皮、木香、茺蔚子、甘草、竹叶、党参、黄芪、海藻、昆布、夏枯草、香附放入煎药容器内,加水6倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
2、将过滤的药渣加水4倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
3、将两次煎煮液混合搅拌均匀,分为2剂服用。
组方中赤芍有清热凉血,散瘀止痛的功能为君药;三七有止血,散瘀,消肿,定痛的功能;刺蒺藜有散风,明目,下气,行血的功能,二者为臣药,三味药共同发挥清热凉血,散瘀止痛,止血散瘀,消肿定痛,散风明目的作用,治疗玻璃体出血效力全面,且以清热凉血,止血散瘀,散风明目为主可治本,枸杞子有滋肾,润肺,补肝,明目的功能为佐药,夏枯草有清肝,散结的功能为使药,与下余诸药是治标。
本发明药物具有清热凉血,散瘀止痛,止血散瘀,消肿定痛,散风明目的功能,用于治疗玻璃体出血,疗程短、见效快、治愈后不复发。
以下通过试验例来进一步阐述本发明所述药物的有益效果,这些试验例包括本发明药物的动物毒性试验报告和临床疗效观察资料。
[试验例1]本发明药物的动物毒性试验报告:
取家兔30只,雌雄兼用,体重2.0—2.5kg,分两组,每组15只,其中一组为超剂量试验组,另一组为正常量试验组。超常量组为20ml/kg,正常量为10ml/kg,给药方式为灌胃法给药,每天两次,连服7天,每天观察给药反应,结果表明二组家兔活动、饮食正常,药物无不良毒副作用。
[试验例2]本发明药物的临床疗效观察
1、一般资料
收治玻璃体出血门诊患者共37例。
2、诊断标准
本病的症状、体征、预后和并发症主要取决于引起疾病的原发病和出血量的多少,出血的次数等因素。自发性积血常突然发作,可以是很少量的积血,多者形成浓密的血块。少量积血时,患者可能不自察觉,或仅有“飞蚊症”;较多的积血发生时,患者发觉眼前暗影飘动,或似有红玻璃片遮挡,反复出血的患者可自觉“冒烟”,视力明显下降。眼科检查,在积血较少,不致影响裂隙灯观察时,可以看到红细胞聚集于玻璃体凝胶的支架中,呈柠檬色尘状。中等量的新鲜积血可呈致密的黑色条状混浊。大量积血致眼底无红光反射。
3、治疗方法
选用上述药剂,给患者服用,每次服用1剂,每天早、晚各服1次,10天为一个疗程,连续服用3个疗程。
4、疗效评定标准
显效:玻璃体出血症状消失,体质恢复正常,痊愈;
好转:飞蚊症消失,视力明显好转,逐步恢复正常;
无效:达不到好转标准者。
5、治疗结果(见下表)
在上述治疗中,用本发明药物治疗玻璃体出血患者37例,结果显效30例,显效率为81.1%,好转5例,好转率为13.5%,无效2例,总有效率为94.6%。
Claims (3)
1.一种治疗玻璃体出血的药物,其特征在于:它是由下列重量范围内的原料药制成:
当归10-14克,赤芍10-14克,川芎10-14克,丹参10-14克,黄芩10-14克,三七15-25克,生地黄10-20克,金银花10-20克,牡丹皮10-20克,白术10-20克,红花10-20克,泽泻5-15克,茯苓5-15克,刺蒺藜5-15克,车前子5-15克,枸杞子15-20克,石斛5-15克,柴胡5-15克,青皮5-15克,木香4-8克,茺蔚子5-15克,甘草10-15克,竹叶5-15克,党参5-15克,黄芪5-15克,海藻5-15克,昆布5-15克,夏枯草5-15克,香附5-15克。
2.根据权利要求1所述的药物,其中各原料药的用量为:
当归12克,赤芍12克,川芎12克,丹参12克,黄芩12克,三七20克,生地黄15克,金银花15克,牡丹皮15克,白术15克,红花15克,泽泻10克,茯苓10克,刺蒺藜10克,车前子10克,枸杞子15克,石斛10克,柴胡10克,青皮10克,木香6克,茺蔚子10克,甘草12克,竹叶10克,党参10克,黄芪10克,海藻10克,昆布10克,夏枯草10克,香附10克。
3.根据权利要求1或2所述药物的制备方法,它包括下列步骤:
(一)备料
(1)当归:拣去杂质,洗净,闷润,稍晾至内外湿度适宜时,切片晒干;
(2)赤芍:取原药材,除去杂质,大小分档,洗净,润透,切薄片,干燥,筛去碎屑;
(3)川芎:拣去杂质,分开大、小个,用水浸泡,晒晾,闷润后切片,干燥;
(4)丹参:拣净杂质,除去根茎,洗净,捞出,润透后切片,晾干;
(5)黄芩:拣去杂质,除去残茎,用凉水浸润或置开水中稍浸捞出,切片,晒干;
(6)三七:拣净杂质,捣碎,研末或润透后切片晒干;
(7)生地黄:除去杂质,洗净,稍润,切厚片,干燥,筛去碎屑;
(8)金银花:筛去泥沙,拣净杂质;
(9)牡丹皮:拣去杂质,除去木心,洗净,润透,切片,晾干;
(10)白术:拣净杂质,用水浸泡,泡后捞出,润透,切片,晒干;
(11)红花:拣净杂质,除去茎叶、蒂头,晒干;
(12)泽泻:拣去杂质,大小分档,用水浸泡至八成透,捞出,晒凉,闷润至内外湿度均匀,切片,晒干;
(13)茯苓:用水浸泡,洗净捞出,闷透后,切片,晒干;
(14)刺蒺藜:漂去泥沙,除净残留的硬刺;
(15)车前子:拣去杂质,筛去泥屑,空粒;
(16)枸杞子:簸净杂质,摘去残留的梗和蒂;
(17)石斛:取干燥的石斛,用水泡约至八成透,焖润,除去残根及黑枝,切段,撞去薄膜,晒干;
(18)柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,随即晒干;
(19)青皮:拣净杂质,用水浸泡,捞出,润透,切片,晒干;
(20)木香:将原生药放清水内洗净,捞出,闷润12—24小时使软,切片,晒干;
(21)茺蔚子:果实成熟时割取全株,晒干,打下果实,拣去枝叶,筛净杂质;
(22)甘草:拣去杂质,洗净,用水浸泡至八成透时,捞出,润透,切片,晾干;
(23)竹叶:拣净杂质,除去梗叶,晾干;
(24)党参:洗净泥沙后润透去芦,切片或切段,晒干;
(25)黄芪:拣净杂质,除去残留的根头和空心较大的根,用水浸泡,捞出,润透后及时切片,晒干;
(26)海藻:拣去杂质,用水略漂,稍晾,切段,晒干;
(27)昆布:拣去杂质,用水漂净,切成宽丝,晾干;
(28)夏枯草:取原药材,除去枝梗、叶片及杂质,筛去灰屑;
(29)香附:拣去杂质,碾成碎粒,簸去细毛及细末;
(二)制备
(1)将所述重量的当归、赤芍、川芎、丹参、黄芩、三七、生地黄、金银花、牡丹皮、白术、红花、泽泻、茯苓、刺蒺藜、车前子、枸杞子、石斛、柴胡、青皮、木香、茺蔚子、甘草、竹叶、党参、黄芪、海藻、昆布、夏枯草、香附放入煎药容器内,加水6倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
(2)将过滤的药渣加水4倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
(3)将两次煎煮液混合搅拌均匀,分为2剂服用。
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CN1273851A (zh) * | 1999-05-18 | 2000-11-22 | 宋敏 | 治疗眼内出血的中药 |
CN106728705A (zh) * | 2017-03-19 | 2017-05-31 | 郝振昌 | 一种治疗视网膜色素变性的药物及其制备方法 |
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CN1273851A (zh) * | 1999-05-18 | 2000-11-22 | 宋敏 | 治疗眼内出血的中药 |
CN106728705A (zh) * | 2017-03-19 | 2017-05-31 | 郝振昌 | 一种治疗视网膜色素变性的药物及其制备方法 |
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