CN102686571B - 三环杂环化合物 - Google Patents
三环杂环化合物 Download PDFInfo
- Publication number
- CN102686571B CN102686571B CN201080059932.3A CN201080059932A CN102686571B CN 102686571 B CN102686571 B CN 102686571B CN 201080059932 A CN201080059932 A CN 201080059932A CN 102686571 B CN102686571 B CN 102686571B
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- Prior art keywords
- isoxazole
- base
- phenyl
- trifluoromethyl
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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| CN103124727B (zh) | 2010-07-20 | 2015-03-25 | 百时美施贵宝公司 | 取代的3-苯基-1,2,4-噁二唑化合物 |
| JP5869579B2 (ja) | 2010-09-24 | 2016-02-24 | ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company | 置換オキサジアゾール化合物およびそれらのs1p1アゴニストとしての使用 |
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| TWI613182B (zh) | 2013-02-21 | 2018-02-01 | 必治妥美雅史谷比公司 | 雙環化合物 |
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| JP7029445B2 (ja) * | 2016-09-02 | 2022-03-03 | ブリストル-マイヤーズ スクイブ カンパニー | 置換された三環式ヘテロ環化合物 |
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| WO2019032632A1 (en) | 2017-08-09 | 2019-02-14 | Bristol-Myers Squibb Company | ALKYLPHENYL COMPOUNDS |
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| SI2326621T1 (sl) | 2008-07-23 | 2016-10-28 | Arena Pharmaceuticals, Inc. | Substituirani derivati 1,2,3,4-tetrahidrociklopenta(b)indol-3-il)ocetne kisline, uporabni pri zdravljenju avtoimunskih in vnetnih motenj |
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2010
- 2010-10-29 EP EP13154679.8A patent/EP2592071B1/en not_active Not-in-force
- 2010-10-29 US US13/504,541 patent/US9216972B2/en active Active
- 2010-10-29 WO PCT/US2010/054594 patent/WO2011059784A1/en not_active Ceased
- 2010-10-29 ES ES13154679T patent/ES2759949T3/es active Active
- 2010-10-29 AU AU2010319879A patent/AU2010319879A1/en not_active Abandoned
- 2010-10-29 MX MX2012004848A patent/MX336881B/es active IP Right Grant
- 2010-10-29 EP EP13154833.1A patent/EP2597089A1/en not_active Withdrawn
- 2010-10-29 CN CN201080059932.3A patent/CN102686571B/zh not_active Expired - Fee Related
- 2010-10-29 EP EP10774099A patent/EP2493866A1/en not_active Withdrawn
- 2010-10-29 KR KR1020127013598A patent/KR20130036171A/ko not_active Withdrawn
- 2010-10-29 JP JP2012537086A patent/JP5728487B2/ja not_active Expired - Fee Related
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| WO2003027095A1 (en) * | 2001-09-26 | 2003-04-03 | Bayer Pharmaceuticals Corporation | Substituted 3-pyridyl tetrazoles as steroid c17,20 lyase inhibitors |
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| WO2008039520A2 (en) * | 2006-09-26 | 2008-04-03 | Synta Pharmaceuticals Corp. | Fused ring compounds for inflammation and immune-related uses |
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| US20100215741A1 (en) * | 2009-02-25 | 2010-08-26 | Neuroscienze Pharmaness S.C. A.R.L. | Pharmaceutical compounds |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2013509431A (ja) | 2013-03-14 |
| KR20130036171A (ko) | 2013-04-11 |
| MX336881B (es) | 2016-02-04 |
| EP2592071A1 (en) | 2013-05-15 |
| EP2592071B1 (en) | 2019-09-18 |
| US20120214767A1 (en) | 2012-08-23 |
| ES2759949T3 (es) | 2020-05-12 |
| EP2597089A1 (en) | 2013-05-29 |
| JP5728487B2 (ja) | 2015-06-03 |
| CN102686571A (zh) | 2012-09-19 |
| EP2493866A1 (en) | 2012-09-05 |
| AU2010319879A1 (en) | 2012-06-14 |
| MX2012004848A (es) | 2012-05-29 |
| WO2011059784A1 (en) | 2011-05-19 |
| US9216972B2 (en) | 2015-12-22 |
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