CN101827844B - 可用作ALK抑制剂的咪唑并[1,2-a]吡啶衍生物 - Google Patents

可用作ALK抑制剂的咪唑并[1,2-a]吡啶衍生物 Download PDF

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Publication number
CN101827844B
CN101827844B CN2008801122032A CN200880112203A CN101827844B CN 101827844 B CN101827844 B CN 101827844B CN 2008801122032 A CN2008801122032 A CN 2008801122032A CN 200880112203 A CN200880112203 A CN 200880112203A CN 101827844 B CN101827844 B CN 101827844B
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pyridin
imidazo
phenyl
pyridine
pyrazol
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CN101827844A (zh
Inventor
D·肖
C·勒布朗
D·利佐斯
C·里奇
V·弗明格尔
S·刘易斯
B·霍恩斯佩格尔
N·J·施蒂夫尔
S·韦勒
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Novartis AG
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Novartis AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Virology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Urology & Nephrology (AREA)
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  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
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CN2008801122032A 2007-10-17 2008-10-15 可用作ALK抑制剂的咪唑并[1,2-a]吡啶衍生物 Expired - Fee Related CN101827844B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP07118726 2007-10-17
EP07118726.4 2007-10-17
EP08151336.8 2008-02-12
EP08151336 2008-02-12
PCT/EP2008/063841 WO2009050183A2 (en) 2007-10-17 2008-10-15 Imidazo [1, 2-a] pyridine derivatives useful as alk inhibitors

Publications (2)

Publication Number Publication Date
CN101827844A CN101827844A (zh) 2010-09-08
CN101827844B true CN101827844B (zh) 2013-08-14

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CN2008801122032A Expired - Fee Related CN101827844B (zh) 2007-10-17 2008-10-15 可用作ALK抑制剂的咪唑并[1,2-a]吡啶衍生物

Country Status (23)

Country Link
US (1) US8367662B2 (enExample)
EP (1) EP2212323B1 (enExample)
JP (1) JP5456681B2 (enExample)
KR (1) KR20100076022A (enExample)
CN (1) CN101827844B (enExample)
AR (1) AR068877A1 (enExample)
AU (1) AU2008313773B2 (enExample)
BR (1) BRPI0817434A2 (enExample)
CA (1) CA2703037A1 (enExample)
CL (1) CL2008003056A1 (enExample)
CO (1) CO6270321A2 (enExample)
EA (1) EA201000615A1 (enExample)
ES (1) ES2393430T3 (enExample)
IL (1) IL204720A0 (enExample)
MA (1) MA31766B1 (enExample)
MX (1) MX2010004244A (enExample)
PE (1) PE20091383A1 (enExample)
PL (1) PL2212323T3 (enExample)
PT (1) PT2212323E (enExample)
TN (1) TN2010000167A1 (enExample)
TW (1) TW200922570A (enExample)
WO (1) WO2009050183A2 (enExample)
ZA (1) ZA201002334B (enExample)

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