CN100341493C - 用于延时和受控释放药物活性成分的微粒口服盖仑制剂 - Google Patents

用于延时和受控释放药物活性成分的微粒口服盖仑制剂 Download PDF

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Publication number
CN100341493C
CN100341493C CNB028200667A CN02820066A CN100341493C CN 100341493 C CN100341493 C CN 100341493C CN B028200667 A CNB028200667 A CN B028200667A CN 02820066 A CN02820066 A CN 02820066A CN 100341493 C CN100341493 C CN 100341493C
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release
active ingredient
microcapsules
form according
active component
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Expired - Lifetime
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Chinese (zh)
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CN1568181A (zh
Inventor
V·勒格朗
C·卡斯唐
R·梅吕埃
G·苏拉
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Flamel Technologies SA
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Flamel Technologies SA
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CNB028200667A 2001-10-09 2002-10-09 用于延时和受控释放药物活性成分的微粒口服盖仑制剂 Expired - Lifetime CN100341493C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR01/12999 2001-10-09
FR0112999A FR2830447B1 (fr) 2001-10-09 2001-10-09 Forme galenique orale microparticulaire pour la liberation retardee et controlee de principes actifs pharmaceutiques

Publications (2)

Publication Number Publication Date
CN1568181A CN1568181A (zh) 2005-01-19
CN100341493C true CN100341493C (zh) 2007-10-10

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CNB028200667A Expired - Lifetime CN100341493C (zh) 2001-10-09 2002-10-09 用于延时和受控释放药物活性成分的微粒口服盖仑制剂

Country Status (14)

Country Link
US (1) US20050037077A1 (enExample)
EP (1) EP1434572B1 (enExample)
JP (1) JP4718116B2 (enExample)
KR (2) KR20100063825A (enExample)
CN (1) CN100341493C (enExample)
AU (1) AU2002362712A1 (enExample)
BR (1) BRPI0213175B8 (enExample)
CA (1) CA2463134C (enExample)
ES (1) ES2661723T3 (enExample)
FR (1) FR2830447B1 (enExample)
IL (2) IL160795A0 (enExample)
MX (1) MXPA04003367A (enExample)
WO (1) WO2003030878A2 (enExample)
ZA (1) ZA200402460B (enExample)

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KR20100063825A (ko) 2010-06-11
BR0213175A (pt) 2004-09-14
MXPA04003367A (es) 2005-01-25
IL160795A (en) 2010-11-30
FR2830447B1 (fr) 2004-04-16
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ZA200402460B (en) 2005-08-31
IL160795A0 (en) 2004-08-31
AU2002362712A1 (en) 2003-04-22
CN1568181A (zh) 2005-01-19
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FR2830447A1 (fr) 2003-04-11
WO2003030878A3 (fr) 2003-12-04
HK1072898A1 (zh) 2005-09-16
US20050037077A1 (en) 2005-02-17
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