CL2008000985A1 - Compuesto derivado de heterociclos de nitrogeno, agonistas del receptor gnrh; composicion farmaceutica que comprende a dicho compuesto; y uso para tratar una afeccion relacionada con las hormonas sexuales, endometriosis, dismenorrea, enfermedad de ov - Google Patents

Compuesto derivado de heterociclos de nitrogeno, agonistas del receptor gnrh; composicion farmaceutica que comprende a dicho compuesto; y uso para tratar una afeccion relacionada con las hormonas sexuales, endometriosis, dismenorrea, enfermedad de ov

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Publication number
CL2008000985A1
CL2008000985A1 CL200800985A CL2008000985A CL2008000985A1 CL 2008000985 A1 CL2008000985 A1 CL 2008000985A1 CL 200800985 A CL200800985 A CL 200800985A CL 2008000985 A CL2008000985 A CL 2008000985A CL 2008000985 A1 CL2008000985 A1 CL 2008000985A1
Authority
CL
Chile
Prior art keywords
compound
dismenorrea
heterocicles
gnrh
endometriosis
Prior art date
Application number
CL200800985A
Other languages
English (en)
Inventor
Chen Graham Beaton Mi
Timothy Richard Coon
Ewing Todd
Jiang Wanlong
Richard Lowe
Willy Moree
Smith Nicole Nicole
Warren Wade
Original Assignee
Neurocrine Biosciences Inc
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Publication date
Application filed by Neurocrine Biosciences Inc filed Critical Neurocrine Biosciences Inc
Publication of CL2008000985A1 publication Critical patent/CL2008000985A1/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
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    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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    • A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Quinoline Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CL200800985A 2007-04-06 2008-04-04 Compuesto derivado de heterociclos de nitrogeno, agonistas del receptor gnrh; composicion farmaceutica que comprende a dicho compuesto; y uso para tratar una afeccion relacionada con las hormonas sexuales, endometriosis, dismenorrea, enfermedad de ov CL2008000985A1 (es)

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CA2683431A1 (en) 2008-10-16
US8481738B2 (en) 2013-07-09
US8084614B2 (en) 2011-12-27
JP2010523593A (ja) 2010-07-15
JP5735799B2 (ja) 2015-06-17
UY31009A1 (es) 2008-11-28
EA017029B1 (ru) 2012-09-28
US20210284653A1 (en) 2021-09-16
AU2008237239B2 (en) 2013-08-29
IL201262A (en) 2016-02-29
BRPI0809931B1 (pt) 2019-10-29
US10941159B2 (en) 2021-03-09
MX2009010828A (es) 2009-10-29
EA200970928A1 (ru) 2010-04-30
KR20090130102A (ko) 2009-12-17
PE20090044A1 (es) 2009-01-23
NZ580457A (en) 2012-03-30
US11713324B2 (en) 2023-08-01
US20140024665A1 (en) 2014-01-23
EP2155194B1 (en) 2015-01-21
ZA200907094B (en) 2011-05-25
EP2155194A1 (en) 2010-02-24
AR065948A1 (es) 2009-07-15
US10336769B2 (en) 2019-07-02
US20100152207A1 (en) 2010-06-17
US20170320888A1 (en) 2017-11-09
AU2008237239A1 (en) 2008-10-16
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US9422310B2 (en) 2016-08-23
IL201262A0 (en) 2010-05-31
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US20120122891A1 (en) 2012-05-17
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CA2683431C (en) 2015-06-09
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US20150183800A1 (en) 2015-07-02
AU2008237239C1 (en) 2014-01-16
PA8775801A1 (es) 2009-05-15
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