CH634062A5 - Process for preparing substituted thiazolidinecarboxylic, oxazanecarboxylic and thiazanecarboxylic acids and their esters - Google Patents

Process for preparing substituted thiazolidinecarboxylic, oxazanecarboxylic and thiazanecarboxylic acids and their esters Download PDF

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Publication number
CH634062A5
CH634062A5 CH1480077A CH1480077A CH634062A5 CH 634062 A5 CH634062 A5 CH 634062A5 CH 1480077 A CH1480077 A CH 1480077A CH 1480077 A CH1480077 A CH 1480077A CH 634062 A5 CH634062 A5 CH 634062A5
Authority
CH
Switzerland
Prior art keywords
value
group
atom
acid
formula
Prior art date
Application number
CH1480077A
Other languages
German (de)
English (en)
Inventor
Miguel Angel Ondetti
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of CH634062A5 publication Critical patent/CH634062A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
CH1480077A 1976-12-03 1977-12-02 Process for preparing substituted thiazolidinecarboxylic, oxazanecarboxylic and thiazanecarboxylic acids and their esters CH634062A5 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
US83610777A 1977-09-23 1977-09-23

Publications (1)

Publication Number Publication Date
CH634062A5 true CH634062A5 (en) 1983-01-14

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1480077A CH634062A5 (en) 1976-12-03 1977-12-02 Process for preparing substituted thiazolidinecarboxylic, oxazanecarboxylic and thiazanecarboxylic acids and their esters

Country Status (28)

Country Link
JP (1) JPS5382778A (el)
AR (1) AR220689A1 (el)
AT (1) AT363467B (el)
AU (1) AU518147B2 (el)
BG (1) BG32269A3 (el)
CA (1) CA1146940A (el)
CH (1) CH634062A5 (el)
DD (1) DD133798A5 (el)
DE (1) DE2752719C2 (el)
DK (1) DK152494C (el)
EG (1) EG13037A (el)
ES (1) ES464555A1 (el)
FI (1) FI67378C (el)
FR (1) FR2372817A1 (el)
GB (1) GB1578940A (el)
GR (1) GR72453B (el)
HK (1) HK55881A (el)
IE (1) IE46169B1 (el)
IL (1) IL53352A0 (el)
IN (1) IN146945B (el)
IT (1) IT1092179B (el)
NL (3) NL171055C (el)
NO (1) NO148416C (el)
NZ (1) NZ185800A (el)
PT (1) PT67352B (el)
RO (2) RO78013A (el)
SE (1) SE441267B (el)
YU (1) YU41823B (el)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1105731B (it) * 1977-06-29 1985-11-04 Yoshitomi Pharmaceutical Composti di tiazolidina
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
US4430344A (en) * 1978-04-08 1984-02-07 Santen Pharmaceutical Co., Ltd. Antihypertensive 4-thiazolidinecarboxylic acids
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (el) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (ja) * 1978-10-05 1983-06-25 ウェルファイド株式会社 環状イミノカルボン酸誘導体およびその塩類
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (de) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd Heterocyclic 5-membered ring compounds
JPH0662529B2 (ja) * 1984-07-13 1994-08-17 三共株式会社 アミノ酸誘導体
DE3685829T2 (de) * 1985-02-04 1992-12-17 Searle & Co Heterocyclische amide.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (de) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkancarbonsäureamide von Thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und Arzneimittel
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
ATA857677A (de) 1981-01-15
JPS618834B2 (el) 1986-03-18
DD133798A5 (de) 1979-01-24
NL7713274A (nl) 1978-06-06
HK55881A (en) 1981-11-20
RO72596A (ro) 1983-08-03
ES464555A1 (es) 1978-09-01
PT67352B (fr) 1979-05-15
FR2372817A1 (fr) 1978-06-30
FR2372817B1 (el) 1981-06-19
EG13037A (en) 1980-12-31
IN146945B (el) 1979-10-20
IE46169B1 (en) 1983-03-09
FI773640A (fi) 1978-06-04
FI67378B (fi) 1984-11-30
FI67378C (fi) 1985-03-11
IE46169L (en) 1978-06-03
DE2752719A1 (de) 1978-06-08
NO148416C (no) 1983-10-12
NO148416B (no) 1983-06-27
DK152494C (da) 1988-07-25
NL8201145A (nl) 1982-07-01
DE2752719C2 (de) 1982-03-25
IL53352A0 (en) 1978-01-31
RO72596B (ro) 1983-07-30
GR72453B (el) 1983-11-09
NL171055C (nl) 1983-02-01
DK152494B (da) 1988-03-07
RO78013A (ro) 1981-12-25
NL8201146A (nl) 1982-07-01
DK538277A (da) 1978-06-04
AU518147B2 (en) 1981-09-17
NZ185800A (en) 1980-04-28
SE441267B (sv) 1985-09-23
JPS5382778A (en) 1978-07-21
SE7713722L (sv) 1978-06-04
IT1092179B (it) 1985-07-06
AT363467B (de) 1981-08-10
CA1146940A (en) 1983-05-24
BG32269A3 (en) 1982-06-15
AU3037977A (en) 1979-05-17
PT67352A (fr) 1978-01-01
YU41823B (en) 1988-02-29
GB1578940A (en) 1980-11-12
NO774126L (no) 1978-06-06
YU283777A (en) 1983-01-21
AR220689A1 (es) 1980-11-28

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