AU518147B2 - Derivatives of thiazolidine, thiazine and morpholine carboxylic acids - Google Patents

Derivatives of thiazolidine, thiazine and morpholine carboxylic acids

Info

Publication number
AU518147B2
AU518147B2 AU30379/77A AU3037977A AU518147B2 AU 518147 B2 AU518147 B2 AU 518147B2 AU 30379/77 A AU30379/77 A AU 30379/77A AU 3037977 A AU3037977 A AU 3037977A AU 518147 B2 AU518147 B2 AU 518147B2
Authority
AU
Australia
Prior art keywords
thiazine
thiazolidine
derivatives
carboxylic acids
morpholine carboxylic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU30379/77A
Other languages
English (en)
Other versions
AU3037977A (en
Inventor
MA Ondetti
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of AU3037977A publication Critical patent/AU3037977A/en
Application granted granted Critical
Publication of AU518147B2 publication Critical patent/AU518147B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU30379/77A 1976-12-03 1977-11-07 Derivatives of thiazolidine, thiazine and morpholine carboxylic acids Expired AU518147B2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
USUS747281 1976-12-03
US83610777A 1977-09-23 1977-09-23
USUS836107 1977-09-23

Publications (2)

Publication Number Publication Date
AU3037977A AU3037977A (en) 1979-05-17
AU518147B2 true AU518147B2 (en) 1981-09-17

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
AU30379/77A Expired AU518147B2 (en) 1976-12-03 1977-11-07 Derivatives of thiazolidine, thiazine and morpholine carboxylic acids

Country Status (28)

Country Link
JP (1) JPS5382778A (el)
AR (1) AR220689A1 (el)
AT (1) AT363467B (el)
AU (1) AU518147B2 (el)
BG (1) BG32269A3 (el)
CA (1) CA1146940A (el)
CH (1) CH634062A5 (el)
DD (1) DD133798A5 (el)
DE (1) DE2752719C2 (el)
DK (1) DK152494C (el)
EG (1) EG13037A (el)
ES (1) ES464555A1 (el)
FI (1) FI67378C (el)
FR (1) FR2372817A1 (el)
GB (1) GB1578940A (el)
GR (1) GR72453B (el)
HK (1) HK55881A (el)
IE (1) IE46169B1 (el)
IL (1) IL53352A0 (el)
IN (1) IN146945B (el)
IT (1) IT1092179B (el)
NL (3) NL171055C (el)
NO (1) NO148416C (el)
NZ (1) NZ185800A (el)
PT (1) PT67352B (el)
RO (2) RO78013A (el)
SE (1) SE441267B (el)
YU (1) YU41823B (el)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1105731B (it) * 1977-06-29 1985-11-04 Yoshitomi Pharmaceutical Composti di tiazolidina
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
US4430344A (en) * 1978-04-08 1984-02-07 Santen Pharmaceutical Co., Ltd. Antihypertensive 4-thiazolidinecarboxylic acids
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (el) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (ja) * 1978-10-05 1983-06-25 ウェルファイド株式会社 環状イミノカルボン酸誘導体およびその塩類
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (de) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd Heterocyclic 5-membered ring compounds
JPH0662529B2 (ja) * 1984-07-13 1994-08-17 三共株式会社 アミノ酸誘導体
DE3685829T2 (de) * 1985-02-04 1992-12-17 Searle & Co Heterocyclische amide.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (de) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkancarbonsäureamide von Thiazolidincarbonsäuren, Verfahren zu ihrer Herstellung und Arzneimittel
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
ATA857677A (de) 1981-01-15
JPS618834B2 (el) 1986-03-18
CH634062A5 (en) 1983-01-14
DD133798A5 (de) 1979-01-24
NL7713274A (nl) 1978-06-06
HK55881A (en) 1981-11-20
RO72596A (ro) 1983-08-03
ES464555A1 (es) 1978-09-01
PT67352B (fr) 1979-05-15
FR2372817A1 (fr) 1978-06-30
FR2372817B1 (el) 1981-06-19
EG13037A (en) 1980-12-31
IN146945B (el) 1979-10-20
IE46169B1 (en) 1983-03-09
FI773640A (fi) 1978-06-04
FI67378B (fi) 1984-11-30
FI67378C (fi) 1985-03-11
IE46169L (en) 1978-06-03
DE2752719A1 (de) 1978-06-08
NO148416C (no) 1983-10-12
NO148416B (no) 1983-06-27
DK152494C (da) 1988-07-25
NL8201145A (nl) 1982-07-01
DE2752719C2 (de) 1982-03-25
IL53352A0 (en) 1978-01-31
RO72596B (ro) 1983-07-30
GR72453B (el) 1983-11-09
NL171055C (nl) 1983-02-01
DK152494B (da) 1988-03-07
RO78013A (ro) 1981-12-25
NL8201146A (nl) 1982-07-01
DK538277A (da) 1978-06-04
NZ185800A (en) 1980-04-28
SE441267B (sv) 1985-09-23
JPS5382778A (en) 1978-07-21
SE7713722L (sv) 1978-06-04
IT1092179B (it) 1985-07-06
AT363467B (de) 1981-08-10
CA1146940A (en) 1983-05-24
BG32269A3 (en) 1982-06-15
AU3037977A (en) 1979-05-17
PT67352A (fr) 1978-01-01
YU41823B (en) 1988-02-29
GB1578940A (en) 1980-11-12
NO774126L (no) 1978-06-06
YU283777A (en) 1983-01-21
AR220689A1 (es) 1980-11-28

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