CH633291A5 - Verfahren zur herstellung von pyrimido(1,2-a)benzimidazolderivaten. - Google Patents
Verfahren zur herstellung von pyrimido(1,2-a)benzimidazolderivaten. Download PDFInfo
- Publication number
- CH633291A5 CH633291A5 CH1507777A CH1507777A CH633291A5 CH 633291 A5 CH633291 A5 CH 633291A5 CH 1507777 A CH1507777 A CH 1507777A CH 1507777 A CH1507777 A CH 1507777A CH 633291 A5 CH633291 A5 CH 633291A5
- Authority
- CH
- Switzerland
- Prior art keywords
- radical
- carbon atoms
- formula
- hydrogen
- mixture
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB51426/76A GB1585965A (en) | 1976-12-09 | 1976-12-09 | 3,4-dihydropyrimido (1,2 - )benzimidazol - 2(1h) - ones |
| GB3334177 | 1977-08-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH633291A5 true CH633291A5 (de) | 1982-11-30 |
Family
ID=26261828
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH1507777A CH633291A5 (de) | 1976-12-09 | 1977-12-08 | Verfahren zur herstellung von pyrimido(1,2-a)benzimidazolderivaten. |
Country Status (23)
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1157858A (en) | 1979-12-03 | 1983-11-29 | Ikuo Ueda | Quinazoline derivatives |
| IE51802B1 (en) * | 1979-12-03 | 1987-04-01 | Fujisawa Pharmaceutical Co | Quinazoline derivatives,processes for their preparation and pharmaceutical compositions containing them |
| DE3208218A1 (de) * | 1982-03-06 | 1983-09-08 | Basf Ag, 6700 Ludwigshafen | Isoindolinfarbstoffe und deren verwendung |
| RU2453312C1 (ru) * | 2010-11-10 | 2012-06-20 | Федеральное государственное автономное образовательное учреждение высшего профессионального образования "ЮЖНЫЙ ФЕДЕРАЛЬНЫЙ УНИВЕРСИТЕТ" | Средство, проявляющее антиагрегантную и антитромбогенную активности |
| SG11201408617PA (en) | 2012-06-27 | 2015-01-29 | 4Sc Discovery Gmbh | Bifluorodioxalane-amino-benzimidazole kinase inhibitors for the treatment of cancer, autoimmuneinflammation and cns disorders |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3468888A (en) * | 1967-04-11 | 1969-09-23 | Smithkline Corp | 2-substituted pyrimido(1,2-a) benzimidazoles |
| US3988340A (en) * | 1975-01-23 | 1976-10-26 | Bristol-Myers Company | 6-Alkoxymethyl-1,2,3,5-tetrahydroimidazo[2,1-b]quinazolin-2-ones and 7-alkoxymethyl-6-[H]-1,2,3,4-tetrahydropyrimido[2,1-b]quinazolin-2-ones |
| US4072679A (en) * | 1976-06-15 | 1978-02-07 | E. R. Squibb & Sons, Inc. | 1,4- AND 4,10-DIHYDRO-4-OXO-PYRIMIDO (1,2-A)-benzimidazole-3-carboxylic acids, esters and amides |
-
1977
- 1977-11-23 US US05/855,003 patent/US4167569A/en not_active Expired - Lifetime
- 1977-11-28 IE IE2408/77A patent/IE45924B1/en unknown
- 1977-11-29 CA CA291,976A patent/CA1086727A/en not_active Expired
- 1977-11-30 NZ NZ185823A patent/NZ185823A/xx unknown
- 1977-12-01 IL IL53507A patent/IL53507A/xx unknown
- 1977-12-01 AU AU31121/77A patent/AU514427B2/en not_active Expired
- 1977-12-05 HU HU77IE816A patent/HU176540B/hu unknown
- 1977-12-07 DD DD7700202450A patent/DD133330A5/xx unknown
- 1977-12-07 ES ES464862A patent/ES464862A1/es not_active Expired
- 1977-12-07 GR GR54931A patent/GR65298B/el unknown
- 1977-12-08 FR FR7737011A patent/FR2373543A1/fr active Granted
- 1977-12-08 SE SE7713958A patent/SE435385B/sv unknown
- 1977-12-08 PL PL1977202753A patent/PL107142B1/pl unknown
- 1977-12-08 NO NO774216A patent/NO774216L/no unknown
- 1977-12-08 CH CH1507777A patent/CH633291A5/de not_active IP Right Cessation
- 1977-12-09 JP JP14866977A patent/JPS5390296A/ja active Pending
- 1977-12-09 FI FI773724A patent/FI63577C/fi not_active IP Right Cessation
- 1977-12-09 SU SU772552626A patent/SU843751A3/ru active
- 1977-12-09 CS CS778270A patent/CS199696B2/cs unknown
- 1977-12-09 AT AT883677A patent/AT359068B/de not_active IP Right Cessation
- 1977-12-09 DE DE19772754930 patent/DE2754930A1/de not_active Withdrawn
- 1977-12-09 IT IT30558/77A patent/IT1143729B/it active
- 1977-12-09 NL NL7713658A patent/NL7713658A/xx not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CA1086727A (en) | 1980-09-30 |
| NZ185823A (en) | 1980-08-26 |
| HU176540B (en) | 1981-03-28 |
| IL53507A0 (en) | 1978-03-10 |
| CS199696B2 (en) | 1980-07-31 |
| AU3112177A (en) | 1979-06-07 |
| FR2373543B1 (US07922777-20110412-C00004.png) | 1980-05-16 |
| DE2754930A1 (de) | 1978-06-15 |
| ATA883677A (de) | 1980-03-15 |
| SE435385B (sv) | 1984-09-24 |
| IE45924B1 (en) | 1982-12-29 |
| GR65298B (en) | 1980-08-01 |
| PL202753A1 (pl) | 1978-10-09 |
| FR2373543A1 (fr) | 1978-07-07 |
| US4167569A (en) | 1979-09-11 |
| JPS5390296A (en) | 1978-08-08 |
| PL107142B1 (pl) | 1980-01-31 |
| FI63577C (fi) | 1983-07-11 |
| IE45924L (en) | 1978-06-09 |
| FI63577B (fi) | 1983-03-31 |
| IT1143729B (it) | 1986-10-22 |
| FI773724A (fi) | 1978-06-10 |
| DD133330A5 (de) | 1978-12-27 |
| AT359068B (de) | 1980-10-27 |
| AU514427B2 (en) | 1981-02-12 |
| IL53507A (en) | 1981-07-31 |
| ES464862A1 (es) | 1979-01-01 |
| NL7713658A (nl) | 1978-06-13 |
| SE7713958L (sv) | 1978-06-10 |
| SU843751A3 (ru) | 1981-06-30 |
| NO774216L (no) | 1978-06-12 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP0682027B1 (de) | Pyrrolopyrimidinderivate mit antiproliferativer Wirkung | |
| DE3724164A1 (de) | Neue 1,4-benzodiazepine, ihre herstellung und verwendung | |
| DE60207759T2 (de) | Pyrimidotriazine als phosphataseinhibitoren | |
| DE69533194T2 (de) | PYRAZOLO(3,4-g)CHINOXALINE ALS PDGF-REZEPTOR PROTEIN TYROSIN-KINASE INHIBITOREN | |
| EP0053767B1 (de) | Tricyclische Cytosinderivate zur Verwendung in Arzneimitteln und Verfahren zu ihrer Herstellung | |
| DE3413489C2 (US07922777-20110412-C00004.png) | ||
| DD266355A5 (de) | Verfahren zur herstellung von neuen 1,4-benzodiozepinen | |
| CH633291A5 (de) | Verfahren zur herstellung von pyrimido(1,2-a)benzimidazolderivaten. | |
| DE1795022B2 (US07922777-20110412-C00004.png) | ||
| DE3447003C2 (de) | 7-Acylamino-9a-methoxymitosane, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Mittel | |
| DE3786865T2 (de) | Aminosäurederivate enthaltende antikonvulsive Zusammensetzungen und Verwendung dieser Aminosäurederivate. | |
| CH500984A (de) | Verfahren zur Herstellung neuartiger Benzomorphan-Derivate | |
| DE1927759A1 (de) | Neue basische Derivate des Benzoxazolin-2-ons und Verfahren zur Herstellung derselben | |
| AT394724B (de) | Verfahren zur herstellung von n7-amidino-substituierten mitomycin-c-derivaten | |
| DD244556A5 (de) | Verfahren zur herstellung von (-)-1beta-aethyl-1alpha-(hydroxymethyl)-1,2,3,4,6,7,12,12b alpha-octahydro-indolo(2,3-a)chinolisin | |
| CH634845A5 (en) | Pharmaceutically useful pyrimido(1,2-a)benzimidazole derivatives and corresponding preparations. | |
| EP0180833A1 (de) | 4-Oxo-pyrido[2,3]pyrimidin-Derivate, Verfahren zur deren Herstellung und diese ethaltende Arzneimittel | |
| DE2949395A1 (de) | Verwendung von substituierten chinazolinen zur behandlung von hochdruck und bradykardie sowie als kardiotone wirkstoffe | |
| DE2901537C2 (US07922777-20110412-C00004.png) | ||
| DE2044666A1 (de) | N substituierte Indoldimere | |
| AT325620B (de) | Verfahren zur herstellung von neuen triazolothienodiazepinverbindungen und deren säureadditionssalzen | |
| AT359074B (de) | Verfahren zur herstellung von neuen pyrimido (1,2-a)benzimidazolderivaten | |
| CH631715A5 (de) | Verfahren zur herstellung von isoxazolo-(3,4-d)-pyrimidinen. | |
| GB1585965A (en) | 3,4-dihydropyrimido (1,2 - )benzimidazol - 2(1h) - ones | |
| CH635842A5 (en) | Process for preparing novel 7H-pyrrolo[3,2-f]quinazoline-1,3-diamines |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PL | Patent ceased |