CA2550540A1 - Isothiazole dioxides as cxc- and cc- chemokine receptor ligands - Google Patents

Isothiazole dioxides as cxc- and cc- chemokine receptor ligands Download PDF

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Publication number
CA2550540A1
CA2550540A1 CA002550540A CA2550540A CA2550540A1 CA 2550540 A1 CA2550540 A1 CA 2550540A1 CA 002550540 A CA002550540 A CA 002550540A CA 2550540 A CA2550540 A CA 2550540A CA 2550540 A1 CA2550540 A1 CA 2550540A1
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Prior art keywords
compound
group
pharmaceutically acceptable
substituted
acceptable salt
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CA002550540A
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English (en)
French (fr)
Inventor
Arthur G. Taveras
Junying Zheng
Purakkattle J. Biju
Younong Yu
Jianhua Chao
Jay Fine
Daniel Lundell
Tony Priestley
Angelo Reggiani
J. Robert Merritt
John J. Baldwin
Gaifa Lai
Minglang Wu
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Merck Sharp and Dohme LLC
Pharmacopeia LLC
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Individual
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    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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