BRPI1013336A2 - novos solvatos de cristais - Google Patents
novos solvatos de cristaisInfo
- Publication number
- BRPI1013336A2 BRPI1013336A2 BRPI1013336A BRPI1013336A BRPI1013336A2 BR PI1013336 A2 BRPI1013336 A2 BR PI1013336A2 BR PI1013336 A BRPI1013336 A BR PI1013336A BR PI1013336 A BRPI1013336 A BR PI1013336A BR PI1013336 A2 BRPI1013336 A2 BR PI1013336A2
- Authority
- BR
- Brazil
- Prior art keywords
- new crystal
- crystal solvates
- solvates
- new
- crystal
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2009109160 | 2009-04-28 | ||
| PCT/JP2010/057404 WO2010126014A1 (ja) | 2009-04-28 | 2010-04-27 | 新規溶媒和物結晶 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI1013336A2 true BRPI1013336A2 (pt) | 2016-03-29 |
| BRPI1013336B1 BRPI1013336B1 (pt) | 2020-02-04 |
Family
ID=43032159
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI1013336A BRPI1013336B1 (pt) | 2009-04-28 | 2010-04-27 | cristais solvatos de acetona, métodos para produção dos referidos cristais e método para produção de olmesartana medoxomila |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US8859600B2 (pt) |
| EP (1) | EP2426127B1 (pt) |
| JP (2) | JP5697593B2 (pt) |
| KR (1) | KR20120006513A (pt) |
| CN (1) | CN102414201B (pt) |
| AU (1) | AU2010242635A1 (pt) |
| BR (1) | BRPI1013336B1 (pt) |
| CA (1) | CA2760031C (pt) |
| CO (1) | CO6470817A2 (pt) |
| ES (1) | ES2753874T3 (pt) |
| IL (1) | IL215965A0 (pt) |
| MX (1) | MX2011011540A (pt) |
| MY (1) | MY158090A (pt) |
| NZ (1) | NZ596326A (pt) |
| RU (1) | RU2563631C2 (pt) |
| SG (2) | SG175296A1 (pt) |
| TW (1) | TWI464162B (pt) |
| WO (1) | WO2010126014A1 (pt) |
| ZA (1) | ZA201107813B (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011021224A2 (en) * | 2009-08-19 | 2011-02-24 | Msn Laboratories Limited | Process for (5-methyl-2-oxo-1,3-dioxolen-4-yl)methyl4-(1-hydroxy-1-methylethyl)-2-propyl-1-[4-[2-tetrazol-5-yl)phenyl]phenyl]methylimidazole-5-carboxylate |
| CN103214469B (zh) * | 2013-04-29 | 2014-12-10 | 孙威 | 一种奥美沙坦酯化合物及其制备方法 |
| CN107474042A (zh) * | 2017-09-07 | 2017-12-15 | 浙江华海致诚药业有限公司 | 一种三苯甲基奥美沙坦酯的晶型h |
| CN110082449B (zh) * | 2019-05-24 | 2020-05-19 | 珠海润都制药股份有限公司 | 一种奥美沙坦酯中三苯基氯甲烷的检测方法 |
| CN113105439A (zh) * | 2021-04-15 | 2021-07-13 | 迪嘉药业集团有限公司 | 一种小粒度奥美沙坦酯的结晶制备方法 |
| CN116217628B (zh) * | 2023-05-08 | 2023-07-14 | 华东理工常熟研究院有限公司 | 奥沙利铂Pt(IV)配合物的共晶及其制备方法 |
Family Cites Families (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0282519A (ja) | 1988-09-19 | 1990-03-23 | Sanyo Electric Co Ltd | 固相エピタキシャル成長方法 |
| US5616599A (en) | 1991-02-21 | 1997-04-01 | Sankyo Company, Limited | Angiotensin II antagosist 1-biphenylmethylimidazole compounds and their therapeutic use |
| IE920540A1 (en) | 1991-02-21 | 1992-08-26 | Sankyo Co | 1-biphenylmethylimidazole derivatives, their preparation and¹their therapetuic use |
| JPH0753489A (ja) * | 1993-06-11 | 1995-02-28 | Sankyo Co Ltd | ビフェニルカルボキサミド誘導体の製造法 |
| JPH07121918A (ja) | 1993-08-30 | 1995-05-12 | Tdk Corp | 光磁気記録媒体 |
| JP3671266B2 (ja) | 1996-03-21 | 2005-07-13 | 東洋化成工業株式会社 | ５−置換テトラゾール類の製造方法 |
| JP3521304B2 (ja) | 1996-03-21 | 2004-04-19 | 東洋化成工業株式会社 | １−（テトラゾリルビフェニルメチル）イミダゾール誘導体の製造方法 |
| CO4940418A1 (es) | 1997-07-18 | 2000-07-24 | Novartis Ag | Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso |
| IT1295405B1 (it) * | 1997-09-30 | 1999-05-12 | Merck Sharp & Dohme Italia S P | Uso di un antagonista recettoriale di angiotensina ii per la preparazione di farmaci per aumentare il tasso di sopravvivenza di |
| JP2004217542A (ja) | 2003-01-10 | 2004-08-05 | Fuji Photo Film Co Ltd | ４，５−ジアルコキシカルボニルイミダゾールの製造方法 |
| CN1976926A (zh) * | 2004-09-02 | 2007-06-06 | 特瓦制药工业有限公司 | 奥美沙坦酯的制备 |
| KR100953878B1 (ko) * | 2004-09-02 | 2010-04-22 | 테바 파마슈티컬 인더스트리즈 리미티드 | 올메살탄 메독소밀의 정제 |
| US20070054948A1 (en) | 2004-09-02 | 2007-03-08 | Lilach Hedvati | Purification of olmesartan medoxomil |
| JP2006111586A (ja) | 2004-10-15 | 2006-04-27 | Nippon Petrochemicals Co Ltd | 置換芳香族化合物の酸化方法 |
| CN101094850A (zh) * | 2005-01-03 | 2007-12-26 | 特瓦制药工业有限公司 | 具有较低水平杂质的奥美沙坦酯 |
| EA014026B1 (ru) | 2005-07-29 | 2010-08-30 | Крка, Товарна Здравил, Д.Д., Ново Место | Способ получения олмесартан медоксомила |
| SI22092A (sl) | 2005-07-29 | 2007-02-28 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Postopek za pripravo olmesartan medoksomila |
| WO2007047838A2 (en) * | 2005-10-20 | 2007-04-26 | Dr. Reddy's Laboratories Ltd. | Process for preparing olmesartan medoxomil |
| CZ299902B6 (cs) | 2005-10-27 | 2008-12-29 | Zentiva, A. S | Zpusob odstranování trifenylmethanové chránicí skupiny u prekurzoru antihypertenzních léciv |
| US8048904B2 (en) * | 2006-06-19 | 2011-11-01 | Matrix Laboratories Ltd. | Process for the preparation of olmesartan medoxomil |
| ITMI20061848A1 (it) | 2006-09-27 | 2008-03-28 | Dipharma Spa | Procedimento per la preparazione di composti feniltetrazolici |
| WO2008043996A2 (en) * | 2006-10-09 | 2008-04-17 | Cipla Limited | Process for preparing trityl olmesartan medoxomil and olmesartan medoxomil |
| SI2176253T1 (sl) * | 2007-08-08 | 2012-02-29 | Lek Pharmaceuticals D.D. | Postopek priprave ali čiščenja olmesartan medoksomila ali hidrohalidne soli olmesartan medoksomila |
| EP2036904A1 (en) * | 2007-08-08 | 2009-03-18 | LEK Pharmaceuticals D.D. | A process for the preparation of olmesartan medoxomil |
| HUE025230T2 (en) | 2008-06-09 | 2016-02-29 | Daiichi Sankyo Co Ltd | Process for the preparation of 1-biphenylmethylimidazole compound |
| EP2334668B1 (en) | 2008-09-05 | 2014-04-02 | Krka Tovarna Zdravil, D.D., Novo Mesto | Process for preparing olmesartan medoxomil intermediate |
| KR101676512B1 (ko) * | 2009-04-28 | 2016-11-15 | 다이이찌 산쿄 가부시키가이샤 | 올메살탄메독소밀의 제조 방법 |
| WO2011014611A2 (en) | 2009-07-30 | 2011-02-03 | Dr. Reddy's Laboratories Ltd. | Preparation of olmesartan medoxomil |
| US20130190506A1 (en) | 2010-06-28 | 2013-07-25 | Hetero Research Foundation | Process for olmesartan medoxomil |
-
2010
- 2010-04-27 US US13/266,967 patent/US8859600B2/en active Active
- 2010-04-27 MX MX2011011540A patent/MX2011011540A/es active IP Right Grant
- 2010-04-27 EP EP10769712.0A patent/EP2426127B1/en active Active
- 2010-04-27 RU RU2011148101/04A patent/RU2563631C2/ru not_active IP Right Cessation
- 2010-04-27 JP JP2011511396A patent/JP5697593B2/ja active Active
- 2010-04-27 NZ NZ596326A patent/NZ596326A/en not_active IP Right Cessation
- 2010-04-27 AU AU2010242635A patent/AU2010242635A1/en not_active Abandoned
- 2010-04-27 SG SG2011077146A patent/SG175296A1/en unknown
- 2010-04-27 KR KR1020117025160A patent/KR20120006513A/ko active Search and Examination
- 2010-04-27 CA CA2760031A patent/CA2760031C/en active Active
- 2010-04-27 CN CN201080018900.9A patent/CN102414201B/zh active Active
- 2010-04-27 WO PCT/JP2010/057404 patent/WO2010126014A1/ja active Application Filing
- 2010-04-27 BR BRPI1013336A patent/BRPI1013336B1/pt active IP Right Grant
- 2010-04-27 SG SG10201501131SA patent/SG10201501131SA/en unknown
- 2010-04-27 MY MYPI2011005182A patent/MY158090A/en unknown
- 2010-04-27 TW TW099113167A patent/TWI464162B/zh active
- 2010-04-27 ES ES10769712T patent/ES2753874T3/es active Active
-
2011
- 2011-10-25 ZA ZA2011/07813A patent/ZA201107813B/en unknown
- 2011-10-26 IL IL215965A patent/IL215965A0/en unknown
- 2011-11-24 CO CO11161167A patent/CO6470817A2/es not_active Application Discontinuation
-
2014
- 2014-10-14 US US14/513,984 patent/US20160102079A1/en not_active Abandoned
-
2015
- 2015-01-08 JP JP2015002227A patent/JP5944539B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP2426127A1 (en) | 2012-03-07 |
| AU2010242635A1 (en) | 2011-12-01 |
| US20120059172A1 (en) | 2012-03-08 |
| IL215965A0 (en) | 2012-01-31 |
| CA2760031C (en) | 2015-03-10 |
| RU2563631C2 (ru) | 2015-09-20 |
| SG10201501131SA (en) | 2015-04-29 |
| EP2426127B1 (en) | 2019-09-04 |
| SG175296A1 (en) | 2011-11-28 |
| TW201043616A (en) | 2010-12-16 |
| CN102414201B (zh) | 2015-10-14 |
| CN102414201A (zh) | 2012-04-11 |
| RU2011148101A (ru) | 2013-06-10 |
| KR20120006513A (ko) | 2012-01-18 |
| ZA201107813B (en) | 2012-07-25 |
| BRPI1013336B1 (pt) | 2020-02-04 |
| TWI464162B (zh) | 2014-12-11 |
| MX2011011540A (es) | 2012-04-30 |
| US8859600B2 (en) | 2014-10-14 |
| US20160102079A1 (en) | 2016-04-14 |
| JP2015071647A (ja) | 2015-04-16 |
| WO2010126014A1 (ja) | 2010-11-04 |
| MY158090A (en) | 2016-08-30 |
| AU2010242635A2 (en) | 2014-08-07 |
| EP2426127A4 (en) | 2012-10-03 |
| CA2760031A1 (en) | 2010-11-04 |
| NZ596326A (en) | 2014-02-28 |
| JPWO2010126014A1 (ja) | 2012-11-01 |
| JP5944539B2 (ja) | 2016-07-05 |
| ES2753874T3 (es) | 2020-04-14 |
| JP5697593B2 (ja) | 2015-04-08 |
| CO6470817A2 (es) | 2012-06-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] | ||
| B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 27/04/2010, OBSERVADAS AS CONDICOES LEGAIS. |