BR9803173A - Processos para a preparação de amidas e ésteres hero) ariloxi-heteroarilcarboxìlico, e, composto. - Google Patents

Processos para a preparação de amidas e ésteres hero) ariloxi-heteroarilcarboxìlico, e, composto.

Info

Publication number
BR9803173A
BR9803173A BR9803173A BR9803173A BR9803173A BR 9803173 A BR9803173 A BR 9803173A BR 9803173 A BR9803173 A BR 9803173A BR 9803173 A BR9803173 A BR 9803173A BR 9803173 A BR9803173 A BR 9803173A
Authority
BR
Brazil
Prior art keywords
compound
aryloxy
formula
group
hero
Prior art date
Application number
BR9803173A
Other languages
English (en)
Inventor
Marcus Knell
Monika Brink
Jan Hendrik Wevers
Willi Heinz
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of BR9803173A publication Critical patent/BR9803173A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/26—Radicals substituted by halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

ERO)ARILOXI-HETEROARILCARBOXìLICO, E, COMPOSTO". A invenção diz respeito a um processo para a prepar fórmula I em que A^ 1^ até A^ 5^, R^ 1^, Hal e X um ou dois dos grupos A^ 1^, A^ 2^, A^ 3^, A^ 4^ e A^ 5^ representam um átomo de nitrogênio e os outros grupos, cada um independentemente, representam CR^ 3^, Hal representa um átomo de halogênio, X representa oxigênio ou NR^ 2^, R^ 1^ representa um grupo opcionalmente substituído de alquila, arila, heteroarila ou cicloalquila, R^ 2^ representa um átomo de hidrogênio ou um grupo alquila, ou R^ 1^ e R^ 2^ juntos com o anel interjacente formam um grupo heterocíclico, e R^ 3^, cada um independentemente, representa um átomo de hidrogênio ou um gruptura consistindo essencialmente de um composto heteroariltriclorometano de fórmula II, em que A^ 1^ até A^ 5^ são como mais acima definidos, e 1,0 a 1,5 equivalente de ácido sulfúrico concentrado, e reação do produto intermediário resultante com um álcool ou amina de fórmula III HXR^ 1^ III opcionalmente na presença de um diluente e/ou uma base.
BR9803173A 1997-08-19 1998-08-18 Processos para a preparação de amidas e ésteres hero) ariloxi-heteroarilcarboxìlico, e, composto. BR9803173A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP97114250 1997-08-19

Publications (1)

Publication Number Publication Date
BR9803173A true BR9803173A (pt) 2000-03-21

Family

ID=8227235

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9803173A BR9803173A (pt) 1997-08-19 1998-08-18 Processos para a preparação de amidas e ésteres hero) ariloxi-heteroarilcarboxìlico, e, composto.

Country Status (23)

Country Link
EP (1) EP0899262B1 (pt)
JP (1) JPH11130752A (pt)
KR (1) KR100519420B1 (pt)
CN (1) CN1132817C (pt)
AR (1) AR015420A1 (pt)
AT (1) ATE292624T1 (pt)
AU (1) AU746709B2 (pt)
BR (1) BR9803173A (pt)
CA (1) CA2245080C (pt)
CZ (2) CZ294125B6 (pt)
DE (1) DE69829613T2 (pt)
DK (1) DK0899262T3 (pt)
ES (1) ES2241102T3 (pt)
HK (1) HK1018060A1 (pt)
HU (1) HU222621B1 (pt)
IL (3) IL125787A (pt)
PL (1) PL190872B1 (pt)
PT (1) PT899262E (pt)
SG (1) SG65781A1 (pt)
SI (1) SI0899262T1 (pt)
SK (1) SK284614B6 (pt)
TW (1) TW575563B (pt)
ZA (1) ZA987326B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2341130T3 (es) * 2005-11-07 2010-06-15 Basf Se Proceso para la preparacion de amidas piridilcarboxilicas y esteres.
TWI594975B (zh) 2013-04-24 2017-08-11 第一三共股份有限公司 二羧酸化合物
CN103450125B (zh) * 2013-07-18 2016-01-13 嘉兴中科化学有限公司 一种5-取代苯丙呋喃-2-羧酸及其衍生物的合成方法
CN107074793B (zh) 2014-09-26 2019-08-23 第一三共株式会社 二羧酸化合物的盐
CN104402814A (zh) * 2014-12-01 2015-03-11 南通嘉禾化工有限公司 一锅法合成2-氯-n-(2,4-二氟苯基)烟酰胺的方法
CN107382847A (zh) * 2017-07-21 2017-11-24 南通嘉禾化工有限公司 一种氟吡草胺的合成方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3317549A (en) * 1963-03-25 1967-05-02 Dow Chemical Co Picolinic acid compounds
GB2005667B (en) * 1977-10-03 1982-03-17 Hooker Chemicals Plastics Corp Process for the preparation of benzoyl halide and halosulftonylbenzoul halide
CA2245055C (en) * 1989-02-28 2003-03-25 F. Hoffmann-La Roche Ag Amidation of pyridines
GB9005965D0 (en) * 1990-03-16 1990-05-09 Shell Int Research Herbicidal carboxamide derivatives
BR9406630A (pt) * 1993-05-27 1996-02-06 Shell Int Research Compostos herbicidas
ZA947672B (en) * 1993-10-05 1995-06-29 Shell Internationale Researchm Process for the preparation of acid chloride compounds.
HUP0001957A3 (en) * 1997-02-03 2000-12-28 Dow Agrosciences Llc 2-methoxyimino-2-(pyridinyloxymethyl)phenyl acetamides with carboxylic acid derivatives on the pyridine ring as fungicides, intermediates, preparation and use thereof

Also Published As

Publication number Publication date
SG65781A1 (en) 1999-06-22
EP0899262B1 (en) 2005-04-06
CA2245080C (en) 2009-06-23
CZ294184B6 (cs) 2004-10-13
KR19990023640A (ko) 1999-03-25
AU8080998A (en) 1999-03-04
IL125787A (en) 2003-06-24
DE69829613T2 (de) 2005-09-15
CN1132817C (zh) 2003-12-31
SI0899262T1 (en) 2005-10-31
HU9801890D0 (en) 1998-10-28
PL328053A1 (en) 1999-03-01
DK0899262T3 (da) 2005-06-20
IL148976A (en) 2003-07-31
AR015420A1 (es) 2001-05-02
PT899262E (pt) 2005-08-31
ZA987326B (en) 2000-02-14
JPH11130752A (ja) 1999-05-18
HUP9801890A2 (hu) 1999-05-28
TW575563B (en) 2004-02-11
EP0899262A2 (en) 1999-03-03
SK284614B6 (sk) 2005-07-01
CZ294125B6 (cs) 2004-10-13
CA2245080A1 (en) 1999-02-19
SK113598A3 (en) 1999-08-06
CZ259498A3 (cs) 1999-05-12
CN1210856A (zh) 1999-03-17
IL148976A0 (en) 2002-11-10
AU746709B2 (en) 2002-05-02
IL125787A0 (en) 1999-04-11
HK1018060A1 (en) 1999-12-10
KR100519420B1 (ko) 2006-04-28
ATE292624T1 (de) 2005-04-15
EP0899262A3 (en) 2000-02-02
DE69829613D1 (de) 2005-05-12
HUP9801890A3 (en) 2000-04-28
HU222621B1 (hu) 2003-09-29
ES2241102T3 (es) 2005-10-16
PL190872B1 (pl) 2006-02-28

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE PATENTE COM BASE NOS ARTIGOS 8O E 13 DA LPI NO 9.279 DE 14/05/96.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.