BR0012736A - Processo para a preparação de pirimidinas substituìdas, e, composto - Google Patents

Processo para a preparação de pirimidinas substituìdas, e, composto

Info

Publication number
BR0012736A
BR0012736A BR0012736-1A BR0012736A BR0012736A BR 0012736 A BR0012736 A BR 0012736A BR 0012736 A BR0012736 A BR 0012736A BR 0012736 A BR0012736 A BR 0012736A
Authority
BR
Brazil
Prior art keywords
compound
formula
preparation
substituted pyrimidines
event
Prior art date
Application number
BR0012736-1A
Other languages
English (en)
Inventor
Oliver Meyer
Dieter Gutheil
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of BR0012736A publication Critical patent/BR0012736A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE PIRIMIDINAS SUBSTITUìDAS, E, COMPOSTO". A invenção refere-se a um processo para a preparação de pirimidinas substituidas de fórmula (I): em que R^ 1^, R^ 2^, R^ 3^, R^ 4^ e X são como definidos na reivindicação 1, que compreende reagir uma amidina de fórmula (II): ou um sal da mesma, com um composto de f[fórmula (III): vinilcarbonila 3,3-di-substituído, em que L representa um átomo de halogênio ou um grupo de fórmula -X-R^ 2^, (a) em um solvente inerte, na presença de uma base e um composto de fórmula (IV); H-X-R^ 2^, no evento que L representa um átomo de halogênio, ou (b) em um solvente inerte e na presença de uma base, no evento que L representa um grupo de fórmula -XR^ 2^.
BR0012736-1A 1999-04-15 2000-04-10 Processo para a preparação de pirimidinas substituìdas, e, composto BR0012736A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29244299A 1999-04-15 1999-04-15
US33352899A 1999-06-15 1999-06-15
PCT/US2000/009522 WO2000063183A1 (en) 1999-04-15 2000-04-10 Process for the preparation of substituted pyrimidines

Publications (1)

Publication Number Publication Date
BR0012736A true BR0012736A (pt) 2005-07-05

Family

ID=26967332

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0012736-1A BR0012736A (pt) 1999-04-15 2000-04-10 Processo para a preparação de pirimidinas substituìdas, e, composto

Country Status (22)

Country Link
EP (1) EP1200414B1 (pt)
JP (1) JP2002542233A (pt)
KR (1) KR100781851B1 (pt)
CN (1) CN1161342C (pt)
AR (1) AR023506A1 (pt)
AT (1) ATE293608T1 (pt)
AU (1) AU780907B2 (pt)
BR (1) BR0012736A (pt)
CA (1) CA2370285A1 (pt)
CO (1) CO4970700A1 (pt)
CZ (1) CZ20013691A3 (pt)
DE (1) DE60019606T2 (pt)
ES (1) ES2240093T3 (pt)
HU (1) HUP0200830A3 (pt)
IL (2) IL145888A0 (pt)
MX (1) MXPA01010390A (pt)
PL (1) PL351088A1 (pt)
PT (1) PT1200414E (pt)
SK (1) SK285728B6 (pt)
UA (1) UA73735C2 (pt)
WO (1) WO2000063183A1 (pt)
ZA (1) ZA200108392B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001090080A1 (en) * 2000-05-19 2001-11-29 Basf Aktiengesellschaft Method of combating undesired plant growth on cereals
DE502005003473D1 (de) * 2004-05-19 2008-05-08 Basf Se 2-substituierte pyrimidine und ihre verwendung als pestizide
KR100746582B1 (ko) * 2005-04-19 2007-08-06 주식회사 에이스 디지텍 디스플레이 장치용 광학필터, 이를 포함하는 디스플레이장치, 및 디스플레이 장치용 광학필터의 제조방법
KR100711858B1 (ko) * 2005-04-25 2007-04-30 주식회사 미래건설 세탁물도어를 포함하는 지능형 도어 시스템
ZA200707975B (en) 2005-05-06 2008-11-26 Du Pont Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids
PL1888536T3 (pl) 2005-05-16 2010-09-30 Du Pont Sposób otrzymywania podstawionych pirymidyn
CN101253158B (zh) 2005-09-01 2013-07-10 弗·哈夫曼-拉罗切有限公司 合成芳氧基二氨基嘧啶类化合物的方法
JP2009514876A (ja) * 2005-11-03 2009-04-09 アイアールエム・リミテッド・ライアビリティ・カンパニー タンパク質キナーゼのための化合物および組成物
CN106496127B (zh) * 2016-10-21 2019-09-27 苏州大学 一种多取代嘧啶的制备方法
CN106831603B (zh) * 2017-01-09 2019-07-02 辽宁大学 一种含氟嘧啶化合物的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH660589A5 (de) * 1983-01-28 1987-05-15 Lonza Ag Verfahren zur herstellung von 2-substituierten 5-nitroso-4,6-diamino-pyrimidinen.
DE3642832A1 (de) * 1986-12-16 1988-06-30 Hoechst Ag Verfahren zur herstellung von aminopyrimidinen
DE3642830A1 (de) * 1986-12-16 1988-07-07 Hoechst Ag Verfahren zur herstellung von pyrimidinen
DK160270C (da) * 1988-12-16 1991-08-05 Cheminova Agro As Fremgangsmaade til fremstilling af 2,4- eller 2,4,5-substituerede 6-hydroxypyrimidiner
CZ290330B6 (cs) * 1995-01-26 2002-07-17 American Cyanamid Company 2,6-Disubstituované pyridinové a 2,4-disubstituované pyrimidinové deriváty, způsob a meziprodukty pro jejich výrobu, jejich pouľití a herbicidní prostředky na jejich bázi a způsob potlačování růstu neľádoucích rostlin
PT802193E (pt) * 1996-04-09 2002-04-29 Lonza Ag Processo para a fabricacao de pirimidinas substituidas
DE59801768D1 (de) * 1997-01-13 2001-11-22 Lonza Ag Visp Verfahren zur herstellung von substituierten pyrimidinderivaten
EP0970072A1 (en) * 1997-03-11 2000-01-12 E.I. Dupont De Nemours And Company Heteroaryl azole herbicides
AU7831398A (en) * 1997-06-10 1998-12-30 E.I. Du Pont De Nemours And Company Pyrimidinyl azole herbicides

Also Published As

Publication number Publication date
WO2000063183A1 (en) 2000-10-26
SK285728B6 (sk) 2007-07-06
EP1200414A1 (en) 2002-05-02
EP1200414B1 (en) 2005-04-20
AR023506A1 (es) 2002-09-04
AU780907B2 (en) 2005-04-21
HUP0200830A3 (en) 2003-04-28
CZ20013691A3 (cs) 2002-04-17
PL351088A1 (en) 2003-03-24
CN1355792A (zh) 2002-06-26
AU4337100A (en) 2000-11-02
HUP0200830A2 (hu) 2002-07-29
IL145888A0 (en) 2002-07-25
SK14752001A3 (sk) 2002-05-09
UA73735C2 (en) 2005-09-15
CO4970700A1 (es) 2000-11-07
ZA200108392B (en) 2002-12-24
CN1161342C (zh) 2004-08-11
CA2370285A1 (en) 2000-10-26
PT1200414E (pt) 2005-09-30
JP2002542233A (ja) 2002-12-10
ATE293608T1 (de) 2005-05-15
KR20020000167A (ko) 2002-01-04
DE60019606D1 (de) 2005-05-25
MXPA01010390A (es) 2002-03-27
IL145888A (en) 2006-08-20
DE60019606T2 (de) 2005-08-18
ES2240093T3 (es) 2005-10-16
KR100781851B1 (ko) 2007-12-03

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Legal Events

Date Code Title Description
B15V Prolongation of time limit allowed
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements