BR9714215A - Derivados de benzoato de 1,4-diazabiciclo[2.2.2]oct-2-ilmetila, seu preparo e sua aplicação em terapêutica - Google Patents
Derivados de benzoato de 1,4-diazabiciclo[2.2.2]oct-2-ilmetila, seu preparo e sua aplicação em terapêuticaInfo
- Publication number
- BR9714215A BR9714215A BR9714215-8A BR9714215A BR9714215A BR 9714215 A BR9714215 A BR 9714215A BR 9714215 A BR9714215 A BR 9714215A BR 9714215 A BR9714215 A BR 9714215A
- Authority
- BR
- Brazil
- Prior art keywords
- oct
- preparation
- application
- diazabicyclo
- therapy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Patente de Invenção: <B>"DERIVADOS DE BENZOATO DE 1,4-DIAZABICICLO[2.2.2]OCT-2-ILMETILA, SEU PREPARO E SUA APLICAçãO EM TERAPêUTICA"<D>. Compostos correspondentes à fórmula geral (I) na qual R~ 1~ representa um grupo metila, X~ 1~ representa um átomo de hidrogênio, ou bem OR~ 1~ e X~ 1~ formam juntos um grupo de fórmula -O(CH~ 2~)~ 2~-, -O(CH~ 2~)~ 3~-, -O(CH~ 2~)~ 2~O- ou -O(CH~ 2~)~ 3~O-. X~ 2~ representa um átomo de hidrogênio ou um grupo amino, e X~ 3~ representa um átomo de halogênio. Os compostos da invenção são ligadas dos receptores serotoninérgicos de tipos 5-HT~ 3~ e/ou 5-HT~ 4~, e que agem como agonistas 5-HT~ 4~ e/ou como antagonistas 5-HT~ 3~.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9614847A FR2756563B1 (fr) | 1996-12-04 | 1996-12-04 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-yl- methyle, leur preparation et leur application en therapeutique |
| PCT/FR1997/002174 WO1998024790A1 (fr) | 1996-12-04 | 1997-12-02 | Derives de benzoate de 1,4-diazabicyclo[2.2.2]oct-2-ylmethyle, leur preparation et leur application en therapeutique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9714215A true BR9714215A (pt) | 2000-04-18 |
Family
ID=9498306
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9714215-8A BR9714215A (pt) | 1996-12-04 | 1997-12-02 | Derivados de benzoato de 1,4-diazabiciclo[2.2.2]oct-2-ilmetila, seu preparo e sua aplicação em terapêutica |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6057321A (pt) |
| EP (1) | EP0942910A1 (pt) |
| JP (1) | JP2001504855A (pt) |
| KR (1) | KR20000069283A (pt) |
| CN (1) | CN1239962A (pt) |
| AU (1) | AU7624598A (pt) |
| BG (1) | BG103432A (pt) |
| BR (1) | BR9714215A (pt) |
| CA (1) | CA2271072A1 (pt) |
| CZ (1) | CZ193799A3 (pt) |
| EE (1) | EE9900218A (pt) |
| FR (1) | FR2756563B1 (pt) |
| HU (1) | HUP9904206A3 (pt) |
| IL (1) | IL129927A0 (pt) |
| NO (1) | NO992676L (pt) |
| NZ (1) | NZ336044A (pt) |
| SK (1) | SK74199A3 (pt) |
| TR (1) | TR199901068T2 (pt) |
| WO (1) | WO1998024790A1 (pt) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH11506744A (ja) | 1995-06-07 | 1999-06-15 | ノウブン ファーマシューティカルズ インク． | 室温で液体である低分子量薬を含む経皮組成物 |
| CN1802409A (zh) * | 2003-04-08 | 2006-07-12 | 西巴特殊化学品控股有限公司 | 颜料分散体中的光稳定聚合物分散剂 |
| US7880683B2 (en) * | 2004-08-18 | 2011-02-01 | Ruckus Wireless, Inc. | Antennas with polarization diversity |
| JP5278312B2 (ja) | 2007-04-16 | 2013-09-04 | ダイキン工業株式会社 | 含フッ素エラストマー組成物およびそれからなるシール材 |
| US20100204438A1 (en) * | 2007-09-03 | 2010-08-12 | Basf Se | Method for producing teda derivatives |
| US20110077376A1 (en) * | 2008-05-30 | 2011-03-31 | Katsumi Tokumoto | Process for producing hydroxyalkyltriethylenediamine, and catalyst composition for the production of polyurethane resin using it |
| PL2295438T3 (pl) * | 2008-05-30 | 2015-06-30 | Tosoh Corp | Sposób wytwarzania kompozycji zawierającej hydroksyalkilotrietylenodiaminę i kompozycja katalizatora do wytwarzania żywicy poliuretanowej z zastosowaniem kompozycji hydroksyalkilotrietylenodiaminy |
| CN101671336B (zh) * | 2009-09-23 | 2013-11-13 | 辽宁利锋科技开发有限公司 | 芳杂环并嘧啶衍生物和类似物及其制备方法和用途 |
| JP5504835B2 (ja) * | 2009-11-13 | 2014-05-28 | 東ソー株式会社 | ヒドロキシアルキルピペラジン類及び／又はヒドロキシメチルトリエチレンジアミン類の製造方法 |
| JP5549847B2 (ja) * | 2009-11-16 | 2014-07-16 | 東ソー株式会社 | Ｎ−（２−アルコキシメチル）トリエチレンジアミン類の製造法 |
| JP5707912B2 (ja) * | 2010-12-08 | 2015-04-30 | 東ソー株式会社 | Ｎ−（ジヒドロキシアルキル）ジエチレントリアミン類の組成物、及びそれを用いた２−ヒドロキシ（アルキル）トリエチレンジアミン類の製造方 |
| JP6393959B2 (ja) | 2012-05-31 | 2018-09-26 | 東ソー株式会社 | ポリウレタン樹脂製造用触媒組成物及びそれを用いたポリウレタン樹脂の製造方法 |
| JP6252152B2 (ja) * | 2013-12-11 | 2017-12-27 | 東ソー株式会社 | 二環式アミン化合物の製造方法 |
| KR20220055152A (ko) | 2020-10-26 | 2022-05-03 | 인하대학교 산학협력단 | 급성 융모양막염 진단용 조성물 및 이를 이용한 급성 융모양막염 진단방법 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4772459A (en) * | 1986-09-09 | 1988-09-20 | Erbamont, Inc. | Method for controlling emesis caused by chemotherapeutic agents and antiemetic agents useful therein |
| TW282460B (pt) * | 1993-12-28 | 1996-08-01 | Yamanouchi Pharma Co Ltd | |
| FR2735475B1 (fr) * | 1995-06-13 | 1997-07-11 | Synthelabo | Derives de n-((1,4-diazabicyclo(2.2.2)oct-2-yl)methyl) benzamide, leur preparation et leur application en therapeutique |
-
1996
- 1996-12-04 FR FR9614847A patent/FR2756563B1/fr not_active Expired - Fee Related
-
1997
- 1997-12-02 US US09/319,413 patent/US6057321A/en not_active Expired - Fee Related
- 1997-12-02 JP JP52527298A patent/JP2001504855A/ja active Pending
- 1997-12-02 CZ CZ991937A patent/CZ193799A3/cs unknown
- 1997-12-02 KR KR1019997004915A patent/KR20000069283A/ko not_active Application Discontinuation
- 1997-12-02 EE EEP199900218A patent/EE9900218A/xx unknown
- 1997-12-02 AU AU76245/98A patent/AU7624598A/en not_active Abandoned
- 1997-12-02 CA CA002271072A patent/CA2271072A1/fr not_active Abandoned
- 1997-12-02 HU HU9904206A patent/HUP9904206A3/hu unknown
- 1997-12-02 EP EP97948976A patent/EP0942910A1/fr not_active Withdrawn
- 1997-12-02 TR TR1999/01068T patent/TR199901068T2/xx unknown
- 1997-12-02 CN CN97180353A patent/CN1239962A/zh active Pending
- 1997-12-02 IL IL12992797A patent/IL129927A0/xx unknown
- 1997-12-02 NZ NZ336044A patent/NZ336044A/xx unknown
- 1997-12-02 BR BR9714215-8A patent/BR9714215A/pt not_active Application Discontinuation
- 1997-12-02 WO PCT/FR1997/002174 patent/WO1998024790A1/fr not_active Application Discontinuation
- 1997-12-02 SK SK741-99A patent/SK74199A3/sk unknown
-
1999
- 1999-05-26 BG BG103432A patent/BG103432A/xx unknown
- 1999-06-02 NO NO992676A patent/NO992676L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20000069283A (ko) | 2000-11-25 |
| EE9900218A (et) | 1999-12-15 |
| CZ193799A3 (cs) | 1999-09-15 |
| EP0942910A1 (fr) | 1999-09-22 |
| IL129927A0 (en) | 2000-02-29 |
| AU7624598A (en) | 1998-06-29 |
| SK74199A3 (en) | 2000-02-14 |
| FR2756563A1 (fr) | 1998-06-05 |
| NO992676L (no) | 1999-07-29 |
| NO992676D0 (no) | 1999-06-02 |
| HUP9904206A2 (hu) | 2000-06-28 |
| US6057321A (en) | 2000-05-02 |
| TR199901068T2 (xx) | 1999-07-21 |
| FR2756563B1 (fr) | 1998-12-24 |
| WO1998024790A1 (fr) | 1998-06-11 |
| HUP9904206A3 (en) | 2000-07-28 |
| CN1239962A (zh) | 1999-12-29 |
| BG103432A (en) | 2000-06-30 |
| NZ336044A (en) | 2000-03-27 |
| JP2001504855A (ja) | 2001-04-10 |
| CA2271072A1 (fr) | 1998-06-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA10 | Dismissal: dismissal - article 33 of industrial property law | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |