AR023506A1 - Proceso para la preparacion de pirimidinas sustituidas. - Google Patents

Proceso para la preparacion de pirimidinas sustituidas.

Info

Publication number
AR023506A1
AR023506A1 ARP000101750A ARP000101750A AR023506A1 AR 023506 A1 AR023506 A1 AR 023506A1 AR P000101750 A ARP000101750 A AR P000101750A AR P000101750 A ARP000101750 A AR P000101750A AR 023506 A1 AR023506 A1 AR 023506A1
Authority
AR
Argentina
Prior art keywords
formula
preparation
pyrimidins
replaced
group
Prior art date
Application number
ARP000101750A
Other languages
English (en)
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of AR023506A1 publication Critical patent/AR023506A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Un proceso para la preparacion de pirimidinas sustituidas de formula 1 en donde R1, R2, R3, R4 y X se definen como en la reivindicacion 1 que comprendehacer reaccionar una amidina de formula 2 o una sal de la misma, con un compuesto de vinilcarbonilo3,3-disustituido de formula 3 en donde L representa unátomo de halogeno o un grupo de formula -X-R2, (a)en un solvente inerte, en presencia de una base y un compuesto de formula H-X-R2 en el caso que L representaun átomo de halogeno o (b)en un solvente inerte y en presencia de una base, en el caso que L represente un grupo de formula -X-R2.
ARP000101750A 1999-04-15 2000-04-14 Proceso para la preparacion de pirimidinas sustituidas. AR023506A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29244299A 1999-04-15 1999-04-15
US33352899A 1999-06-15 1999-06-15

Publications (1)

Publication Number Publication Date
AR023506A1 true AR023506A1 (es) 2002-09-04

Family

ID=26967332

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000101750A AR023506A1 (es) 1999-04-15 2000-04-14 Proceso para la preparacion de pirimidinas sustituidas.

Country Status (22)

Country Link
EP (1) EP1200414B1 (es)
JP (1) JP2002542233A (es)
KR (1) KR100781851B1 (es)
CN (1) CN1161342C (es)
AR (1) AR023506A1 (es)
AT (1) ATE293608T1 (es)
AU (1) AU780907B2 (es)
BR (1) BR0012736A (es)
CA (1) CA2370285A1 (es)
CO (1) CO4970700A1 (es)
CZ (1) CZ20013691A3 (es)
DE (1) DE60019606T2 (es)
ES (1) ES2240093T3 (es)
HU (1) HUP0200830A3 (es)
IL (2) IL145888A0 (es)
MX (1) MXPA01010390A (es)
PL (1) PL351088A1 (es)
PT (1) PT1200414E (es)
SK (1) SK285728B6 (es)
UA (1) UA73735C2 (es)
WO (1) WO2000063183A1 (es)
ZA (1) ZA200108392B (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2408604A1 (en) * 2000-05-19 2001-11-29 Basf Aktiengesellschaft Method of combating undesired plant growth on cereals
WO2005113538A1 (de) * 2004-05-19 2005-12-01 Basf Aktiengesellschaft 2-substituierte pyrimidine und ihre verwendung als pestizide
KR100746582B1 (ko) * 2005-04-19 2007-08-06 주식회사 에이스 디지텍 디스플레이 장치용 광학필터, 이를 포함하는 디스플레이장치, 및 디스플레이 장치용 광학필터의 제조방법
KR100711858B1 (ko) * 2005-04-25 2007-04-30 주식회사 미래건설 세탁물도어를 포함하는 지능형 도어 시스템
AU2006246374B2 (en) 2005-05-06 2012-03-29 Corteva Agriscience Llc Method for preparation of optionally 2-substituted 1,6-dihydro-6-oxo-4-pyrimidinecarboxylic acids
US8013155B2 (en) 2005-05-16 2011-09-06 E. I. Du Pont De Nemours And Company Method for preparing substituted pyrimidines
CN101253158B (zh) * 2005-09-01 2013-07-10 弗·哈夫曼-拉罗切有限公司 合成芳氧基二氨基嘧啶类化合物的方法
CN101300234A (zh) * 2005-11-03 2008-11-05 Irm责任有限公司 蛋白激酶抑制剂
CN106496127B (zh) * 2016-10-21 2019-09-27 苏州大学 一种多取代嘧啶的制备方法
CN106831603B (zh) * 2017-01-09 2019-07-02 辽宁大学 一种含氟嘧啶化合物的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH660589A5 (de) * 1983-01-28 1987-05-15 Lonza Ag Verfahren zur herstellung von 2-substituierten 5-nitroso-4,6-diamino-pyrimidinen.
DE3642832A1 (de) * 1986-12-16 1988-06-30 Hoechst Ag Verfahren zur herstellung von aminopyrimidinen
DE3642830A1 (de) * 1986-12-16 1988-07-07 Hoechst Ag Verfahren zur herstellung von pyrimidinen
DK160270C (da) * 1988-12-16 1991-08-05 Cheminova Agro As Fremgangsmaade til fremstilling af 2,4- eller 2,4,5-substituerede 6-hydroxypyrimidiner
CZ290330B6 (cs) * 1995-01-26 2002-07-17 American Cyanamid Company 2,6-Disubstituované pyridinové a 2,4-disubstituované pyrimidinové deriváty, způsob a meziprodukty pro jejich výrobu, jejich pouľití a herbicidní prostředky na jejich bázi a způsob potlačování růstu neľádoucích rostlin
PT802193E (pt) * 1996-04-09 2002-04-29 Lonza Ag Processo para a fabricacao de pirimidinas substituidas
CA2275400C (en) * 1997-01-13 2008-07-15 Beat Schmidt Process for the preparation of substituted pyrimidine desrivatives
AU725548B2 (en) * 1997-03-11 2000-10-12 E.I. Du Pont De Nemours And Company Heteroaryl azole herbicides
WO1998056789A1 (en) * 1997-06-10 1998-12-17 E.I. Du Pont De Nemours And Company Pyrimidinyl azole herbicides

Also Published As

Publication number Publication date
PL351088A1 (en) 2003-03-24
IL145888A0 (en) 2002-07-25
CO4970700A1 (es) 2000-11-07
UA73735C2 (en) 2005-09-15
MXPA01010390A (es) 2002-03-27
EP1200414B1 (en) 2005-04-20
ZA200108392B (en) 2002-12-24
CZ20013691A3 (cs) 2002-04-17
WO2000063183A1 (en) 2000-10-26
HUP0200830A3 (en) 2003-04-28
IL145888A (en) 2006-08-20
KR20020000167A (ko) 2002-01-04
JP2002542233A (ja) 2002-12-10
HUP0200830A2 (hu) 2002-07-29
DE60019606T2 (de) 2005-08-18
ES2240093T3 (es) 2005-10-16
BR0012736A (pt) 2005-07-05
AU780907B2 (en) 2005-04-21
CN1355792A (zh) 2002-06-26
PT1200414E (pt) 2005-09-30
CN1161342C (zh) 2004-08-11
KR100781851B1 (ko) 2007-12-03
ATE293608T1 (de) 2005-05-15
EP1200414A1 (en) 2002-05-02
AU4337100A (en) 2000-11-02
SK14752001A3 (sk) 2002-05-09
DE60019606D1 (de) 2005-05-25
CA2370285A1 (en) 2000-10-26
SK285728B6 (sk) 2007-07-06

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