BR112012012808A2 - método para a produção de 5-(amino-metil)-2-clorotiazol - Google Patents

método para a produção de 5-(amino-metil)-2-clorotiazol

Info

Publication number
BR112012012808A2
BR112012012808A2 BR112012012808A BR112012012808A BR112012012808A2 BR 112012012808 A2 BR112012012808 A2 BR 112012012808A2 BR 112012012808 A BR112012012808 A BR 112012012808A BR 112012012808 A BR112012012808 A BR 112012012808A BR 112012012808 A2 BR112012012808 A2 BR 112012012808A2
Authority
BR
Brazil
Prior art keywords
chlorothiazole
amino
methyl
production
aminomethyl
Prior art date
Application number
BR112012012808A
Other languages
English (en)
Inventor
Kazuyuki Yamagata
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of BR112012012808A2 publication Critical patent/BR112012012808A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

método para a produção de 5-(amino-metil)-2-clorotiazol. a presente invenção refere-se a um método para produzir o 5-(aminometil)-2-clorotiazol, o qual compreende a etapa de misturar um composto representado pela fórmula (2): um ácido mineral e um sal de nitrito conjuntamente.
BR112012012808A 2009-11-30 2010-11-29 método para a produção de 5-(amino-metil)-2-clorotiazol BR112012012808A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2009271482 2009-11-30
PCT/JP2010/071766 WO2011065590A1 (ja) 2009-11-30 2010-11-29 ５－（アミノメチル）－２－クロロチアゾールの製造方法

Publications (1)

Publication Number Publication Date
BR112012012808A2 true BR112012012808A2 (pt) 2015-09-08

Family

ID=44066692

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012012808A BR112012012808A2 (pt) 2009-11-30 2010-11-29 método para a produção de 5-(amino-metil)-2-clorotiazol

Country Status (9)

Country Link
US (1) US8754235B2 (pt)
EP (1) EP2511270A4 (pt)
JP (1) JP5652159B2 (pt)
KR (1) KR20120086744A (pt)
CN (1) CN102648190B (pt)
BR (1) BR112012012808A2 (pt)
IL (1) IL219833A0 (pt)
TW (1) TWI471316B (pt)
WO (1) WO2011065590A1 (pt)

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB850982A (en) * 1957-05-24 1960-10-12 Geigy Ag J R Improvements in and relating to substituted ureas
DE1206914B (de) * 1963-11-26 1965-12-16 Boehringer & Soehne Gmbh Verfahren zur Herstellung von Benzolsulfonylharnstoffen
DE1493672C3 (de) * 1964-08-01 1974-05-02 Farbwerke Hoechst Ag, Vormals Meister Lucius & Bruening, 6000 Frankfurt Verfahren zur Herstellung von Benzolsulfonylharnstoffen
JPS59122444A (ja) * 1982-12-28 1984-07-14 Dai Ichi Pure Chem Co Ltd ４−アミノ酪酸アミド塩酸塩の製造法
DE3511210A1 (de) 1985-03-28 1986-10-02 Bayer Ag, 5090 Leverkusen Verfahren zur inversion der konfiguration sekundaerer alkohole
CA2012716A1 (en) * 1989-03-22 1990-09-22 Akito Tanaka Thiazole compounds, processes for the preparation thereof and pharmaceutical composition comprising the same
JPH03223252A (ja) 1989-12-27 1991-10-02 Nippon Soda Co Ltd 置換メチルアミン類の製造方法
US5180833A (en) 1990-03-16 1993-01-19 Takeda Chemical Industries, Ltd. Process for the preparation of chlorothiazole derivatives
JPH0421674A (ja) 1990-05-15 1992-01-24 Nippon Soda Co Ltd ２―クロロ―５―（アミノメチル）チアゾールの製造方法
JPH05286936A (ja) 1992-04-06 1993-11-02 Takeda Chem Ind Ltd ホルムアミド誘導体の製造法及び新規ホルムアミド誘導体
KR100460828B1 (ko) * 1995-06-23 2005-02-28 스미카 다케다 노야쿠 가부시키가이샤 구아니딘유도체의제조방법,이의중간체및이의제조방법
JP3253245B2 (ja) * 1995-06-23 2002-02-04 武田薬品工業株式会社 グアニジン誘導体の製造法、新規中間体およびその製造法
EP0839153B1 (de) 1995-07-11 2001-08-16 Degussa AG Verfahren zur herstellung von peptiden und n-carbamoyl-geschützten peptiden
JP3413632B2 (ja) * 1995-11-17 2003-06-03 住化武田農薬株式会社 グアニジン誘導体の製造方法
NL1002505C2 (nl) 1996-03-01 1997-09-03 Dijk Food Prod Lopik Zak, alsmede afgifte-inrichting voor het afgeven van een vloeibare substantie uit een zak.
JP3477096B2 (ja) * 1997-12-24 2003-12-10 住化武田農薬株式会社 イソ尿素類の改良された製造方法
CN1125048C (zh) * 1997-12-24 2003-10-22 住化武田农药株式会社 生产异脲的方法
DE19903268A1 (de) * 1999-01-28 2000-08-03 Degussa Verfahren zur Decarbamoylierung von N-carbamoylgeschützten Verbindungen, neue Carbonsäureanhydride und deren Verwendung
BRPI0710204A2 (pt) * 2006-03-16 2011-05-24 Sumitomo Chemical Co processo para a nitração de isouréias

Also Published As

Publication number Publication date
TWI471316B (zh) 2015-02-01
US20120226049A1 (en) 2012-09-06
EP2511270A4 (en) 2013-07-17
JP2011132224A (ja) 2011-07-07
CN102648190A (zh) 2012-08-22
JP5652159B2 (ja) 2015-01-14
CN102648190B (zh) 2014-12-10
KR20120086744A (ko) 2012-08-03
IL219833A0 (en) 2012-07-31
TW201200503A (en) 2012-01-01
US8754235B2 (en) 2014-06-17
WO2011065590A1 (ja) 2011-06-03
EP2511270A1 (en) 2012-10-17

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2386 DE 27-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.