BG64213B1 - Глюкокортикоидселективни противовъзпалителни средства - Google Patents
Глюкокортикоидселективни противовъзпалителни средства Download PDFInfo
- Publication number
- BG64213B1 BG64213B1 BG104698A BG10469800A BG64213B1 BG 64213 B1 BG64213 B1 BG 64213B1 BG 104698 A BG104698 A BG 104698A BG 10469800 A BG10469800 A BG 10469800A BG 64213 B1 BG64213 B1 BG 64213B1
- Authority
- BG
- Bulgaria
- Prior art keywords
- carbon atoms
- twelve carbon
- twelve
- alkyl
- aryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/023,913 US6380207B2 (en) | 1998-02-13 | 1998-02-13 | Glucocortiocoid-selective antiinflammatory agents |
| PCT/US1999/003210 WO1999041257A1 (en) | 1998-02-13 | 1999-02-15 | Glucocorticoid-selective antiinflammatory agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG104698A BG104698A (en) | 2001-05-31 |
| BG64213B1 true BG64213B1 (bg) | 2004-05-31 |
Family
ID=21817891
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG104698A BG64213B1 (bg) | 1998-02-13 | 2000-08-17 | Глюкокортикоидселективни противовъзпалителни средства |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6380207B2 (no) |
| EP (1) | EP1053240B1 (no) |
| JP (1) | JP2002503666A (no) |
| KR (1) | KR20010040940A (no) |
| CN (1) | CN1153771C (no) |
| AT (1) | ATE237620T1 (no) |
| AU (1) | AU760511B2 (no) |
| BG (1) | BG64213B1 (no) |
| BR (1) | BR9907847A (no) |
| CA (1) | CA2320911A1 (no) |
| DE (1) | DE69906938T2 (no) |
| DK (1) | DK1053240T3 (no) |
| ES (1) | ES2197618T3 (no) |
| HK (1) | HK1033309A1 (no) |
| HU (1) | HUP0100846A3 (no) |
| IL (1) | IL137509A0 (no) |
| NO (1) | NO20004052L (no) |
| NZ (1) | NZ506012A (no) |
| PL (1) | PL342999A1 (no) |
| PT (1) | PT1053240E (no) |
| SK (1) | SK284076B6 (no) |
| TR (1) | TR200002345T2 (no) |
| WO (1) | WO1999041257A1 (no) |
| ZA (1) | ZA99533B (no) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6566372B1 (en) * | 1999-08-27 | 2003-05-20 | Ligand Pharmaceuticals Incorporated | Bicyclic androgen and progesterone receptor modulator compounds and methods |
| DE60113032T2 (de) | 2000-10-30 | 2006-07-06 | Pfizer Products Inc., Groton | Glukokortikoidrezeptor-Modulatoren |
| US7026484B2 (en) * | 2001-02-23 | 2006-04-11 | Ligand Pharmaceuticals Incorporated | Tricyclic androgen receptor modulator compounds and methods |
| CA2473886C (en) | 2002-01-22 | 2012-08-21 | The Regents Of The University Of California | Non-steroidal ligands for the glucocorticoid receptor, compositions and uses thereof |
| KR100492913B1 (ko) * | 2002-08-23 | 2005-06-03 | 주식회사 태평양 | 피부 감작 및 자극을 완화하는 피부 외용제 조성물 |
| EP2298316A1 (en) | 2002-08-28 | 2011-03-23 | Harbor BioSciences, Inc. | Therapeutic treatment methods |
| US20040220153A1 (en) * | 2002-09-24 | 2004-11-04 | Jost-Price Edward Roydon | Methods and reagents for the treatment of diseases and disorders associated with increased levels of proinflammatory cytokines |
| JP2006508076A (ja) * | 2002-10-11 | 2006-03-09 | リガンド・ファーマシューティカルズ・インコーポレイテッド | 選択的プロゲステロン受容体モジュレーター化合物としての５−シクロアルケニル５Ｈ−クロメノ［３，４−ｆ］キノリン誘導体 |
| DE20301728U1 (de) * | 2002-10-11 | 2004-03-11 | Ligand Pharmaceuticals, Inc., San Diego | 5-substituierte 7,9-Difluor-5H-Chromeno(3,4-f) -Chinolin-Verbindungen als selektive Progesteronrezeptormodulator-Verbindungen |
| JP2006504736A (ja) * | 2002-10-11 | 2006-02-09 | リガンド・ファーマシューティカルズ・インコーポレイテッド | 選択的プロゲステロンレセプター調節化合物としての５−（１’，１’−シクロアルキル／アルケニル）メチリデン１，２−ジヒドロ−５Ｈ−クロメノ［３，４−ｆ］キノリン |
| US7235662B2 (en) * | 2003-06-11 | 2007-06-26 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor and method |
| BRPI0413820A (pt) * | 2003-08-22 | 2006-10-24 | Ligand Pharm Inc | derivados de 6-cicloamino-2-quinolinona como compostos moduladores de receptor de androgênio |
| TW200517114A (en) | 2003-10-15 | 2005-06-01 | Combinatorx Inc | Methods and reagents for the treatment of immunoinflammatory disorders |
| JP2007512337A (ja) | 2003-11-21 | 2007-05-17 | コンビナトアールエックス インコーポレーティッド | 炎症性障害の治療のための方法および試薬 |
| US8519158B2 (en) | 2004-03-12 | 2013-08-27 | Ligand Pharmaceuticals Incorporated | Androgen receptor modulator compounds and methods |
| KR101293935B1 (ko) * | 2005-06-17 | 2013-08-08 | 리간드 파마슈티칼스 인코포레이티드 | 안드로겐 수용체 조절 화합물 및 방법 |
| EP1916896A4 (en) | 2005-08-26 | 2010-08-11 | Univ California | NOT STEROID-antiandrogens |
| EP2218442A1 (en) | 2005-11-09 | 2010-08-18 | CombinatoRx, Inc. | Methods, compositions, and kits for the treatment of ophthalmic disorders |
| CN101326155B (zh) * | 2005-12-09 | 2012-06-20 | 霍夫曼-拉罗奇有限公司 | 作为抗炎剂的丙酰胺化合物 |
| KR101023001B1 (ko) * | 2005-12-09 | 2011-03-22 | 에프. 호프만-라 로슈 아게 | 항염증제로서의 글루코코티코이드 수용체 조절제 |
| WO2010021681A2 (en) * | 2008-08-18 | 2010-02-25 | Combinatorx (Singapore) Pte. Ltd. | Compositions and methods for treatment of viral diseases |
| US9908182B2 (en) | 2012-01-30 | 2018-03-06 | Black & Decker Inc. | Remote programming of a power tool |
| US8919456B2 (en) | 2012-06-08 | 2014-12-30 | Black & Decker Inc. | Fastener setting algorithm for drill driver |
| US10011006B2 (en) | 2013-08-08 | 2018-07-03 | Black & Decker Inc. | Fastener setting algorithm for drill driver |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5693646A (en) | 1994-12-22 | 1997-12-02 | Ligand Pharmaceuticals Incorporated | Steroid receptor modulator compounds and methods |
| EP1043326A1 (en) | 1994-12-22 | 2000-10-11 | Ligand Pharmaceuticals Incorporated | Steroid receptor modulator compounds and methods |
| US5693133A (en) | 1995-05-10 | 1997-12-02 | Akzo Nobel Nv | Asbestos free roof coatings |
-
1998
- 1998-02-13 US US09/023,913 patent/US6380207B2/en not_active Expired - Fee Related
-
1999
- 1999-01-25 ZA ZA9900533A patent/ZA99533B/xx unknown
- 1999-02-15 PT PT99905971T patent/PT1053240E/pt unknown
- 1999-02-15 PL PL99342999A patent/PL342999A1/xx unknown
- 1999-02-15 TR TR2000/02345T patent/TR200002345T2/xx unknown
- 1999-02-15 CA CA002320911A patent/CA2320911A1/en not_active Abandoned
- 1999-02-15 KR KR1020007008857A patent/KR20010040940A/ko not_active Application Discontinuation
- 1999-02-15 IL IL13750999A patent/IL137509A0/xx unknown
- 1999-02-15 AU AU26003/99A patent/AU760511B2/en not_active Ceased
- 1999-02-15 AT AT99905971T patent/ATE237620T1/de not_active IP Right Cessation
- 1999-02-15 WO PCT/US1999/003210 patent/WO1999041257A1/en not_active Application Discontinuation
- 1999-02-15 BR BR9907847-3A patent/BR9907847A/pt not_active IP Right Cessation
- 1999-02-15 CN CNB998050342A patent/CN1153771C/zh not_active Expired - Fee Related
- 1999-02-15 SK SK1196-2000A patent/SK284076B6/sk unknown
- 1999-02-15 JP JP2000531450A patent/JP2002503666A/ja not_active Withdrawn
- 1999-02-15 NZ NZ506012A patent/NZ506012A/xx unknown
- 1999-02-15 DK DK99905971T patent/DK1053240T3/da active
- 1999-02-15 DE DE69906938T patent/DE69906938T2/de not_active Expired - Fee Related
- 1999-02-15 HU HU0100846A patent/HUP0100846A3/hu unknown
- 1999-02-15 EP EP99905971A patent/EP1053240B1/en not_active Expired - Lifetime
- 1999-02-15 ES ES99905971T patent/ES2197618T3/es not_active Expired - Lifetime
-
2000
- 2000-08-11 NO NO20004052A patent/NO20004052L/no not_active Application Discontinuation
- 2000-08-17 BG BG104698A patent/BG64213B1/bg unknown
-
2001
- 2001-04-19 HK HK01102795A patent/HK1033309A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| SK11962000A3 (sk) | 2001-03-12 |
| DK1053240T3 (da) | 2003-08-11 |
| DE69906938T2 (de) | 2004-02-26 |
| NZ506012A (en) | 2003-03-28 |
| SK284076B6 (sk) | 2004-09-08 |
| EP1053240B1 (en) | 2003-04-16 |
| PL342999A1 (en) | 2001-07-16 |
| EP1053240A1 (en) | 2000-11-22 |
| CA2320911A1 (en) | 1999-08-19 |
| NO20004052D0 (no) | 2000-08-11 |
| US20010049377A1 (en) | 2001-12-06 |
| US6380207B2 (en) | 2002-04-30 |
| HK1033309A1 (en) | 2001-08-24 |
| HUP0100846A2 (hu) | 2001-09-28 |
| CN1153771C (zh) | 2004-06-16 |
| ZA99533B (en) | 1999-07-26 |
| DE69906938D1 (de) | 2003-05-22 |
| CN1297451A (zh) | 2001-05-30 |
| BR9907847A (pt) | 2001-01-09 |
| JP2002503666A (ja) | 2002-02-05 |
| PT1053240E (pt) | 2003-09-30 |
| WO1999041257A1 (en) | 1999-08-19 |
| ES2197618T3 (es) | 2004-01-01 |
| NO20004052L (no) | 2000-10-12 |
| BG104698A (en) | 2001-05-31 |
| TR200002345T2 (tr) | 2000-11-21 |
| HUP0100846A3 (en) | 2003-03-28 |
| AU2600399A (en) | 1999-08-30 |
| KR20010040940A (ko) | 2001-05-15 |
| AU760511B2 (en) | 2003-05-15 |
| ATE237620T1 (de) | 2003-05-15 |
| IL137509A0 (en) | 2001-07-24 |
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