BG61694B1 - Хинуклидинови производни - Google Patents

Хинуклидинови производни Download PDF

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Publication number
BG61694B1
BG61694B1 BG98248A BG9824893A BG61694B1 BG 61694 B1 BG61694 B1 BG 61694B1 BG 98248 A BG98248 A BG 98248A BG 9824893 A BG9824893 A BG 9824893A BG 61694 B1 BG61694 B1 BG 61694B1
Authority
BG
Bulgaria
Prior art keywords
compound
formula
methyl
azabicyclo
diphenylmethyl
Prior art date
Application number
BG98248A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG98248A (bg
Inventor
Fumitaka Ito
Hiroshi Kondo
Kaoru Shimada
Masami Nakane
John A. Lowe Iii
Terry J. Rosen
Bingwei V. Yang
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24845673&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG61694(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of BG98248A publication Critical patent/BG98248A/bg
Publication of BG61694B1 publication Critical patent/BG61694B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG98248A 1991-05-31 1993-11-26 Хинуклидинови производни BG61694B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70840491A 1991-05-31 1991-05-31
PCT/US1992/003317 WO1992021677A1 (en) 1991-05-31 1992-04-28 bibNUCLIDINE DERIVATIVES

Publications (2)

Publication Number Publication Date
BG98248A BG98248A (bg) 1994-07-29
BG61694B1 true BG61694B1 (bg) 1998-03-31

Family

ID=24845673

Family Applications (1)

Application Number Title Priority Date Filing Date
BG98248A BG61694B1 (bg) 1991-05-31 1993-11-26 Хинуклидинови производни

Country Status (41)

Country Link
US (3) US5807867A (enExample)
EP (1) EP0587723B1 (enExample)
JP (2) JPH0733386B2 (enExample)
KR (1) KR100214905B1 (enExample)
CN (1) CN1048492C (enExample)
AP (1) AP299A (enExample)
AT (1) ATE135006T1 (enExample)
AU (1) AU657552B2 (enExample)
BG (1) BG61694B1 (enExample)
BR (1) BR9206073A (enExample)
CA (1) CA2102179C (enExample)
CZ (1) CZ281403B6 (enExample)
DE (4) DE9290063U1 (enExample)
DK (1) DK0587723T3 (enExample)
EG (1) EG19944A (enExample)
ES (1) ES2084361T3 (enExample)
FI (1) FI114475B (enExample)
GR (1) GR3019687T3 (enExample)
GT (1) GT199200028A (enExample)
HU (1) HU217548B (enExample)
IE (1) IE72473B1 (enExample)
IL (1) IL102008A (enExample)
IS (1) IS1611B (enExample)
LU (1) LU91293I2 (enExample)
MA (1) MA22539A1 (enExample)
MX (1) MX9202554A (enExample)
NL (1) NL300250I2 (enExample)
NO (2) NO302701B1 (enExample)
NZ (2) NZ270673A (enExample)
OA (1) OA09867A (enExample)
PL (1) PL171379B1 (enExample)
PT (1) PT100546B (enExample)
RO (1) RO110499B1 (enExample)
RU (1) RU2103269C1 (enExample)
SK (1) SK278788B6 (enExample)
TW (1) TW204349B (enExample)
UA (1) UA27776C2 (enExample)
UY (1) UY23422A1 (enExample)
WO (1) WO1992021677A1 (enExample)
YU (1) YU48995B (enExample)
ZA (1) ZA923942B (enExample)

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IL116249A (en) * 1994-12-12 2003-07-06 Pfizer Nk-1 receptor antagonists for the treatment of neuronal damage and stroke
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TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
IL123740A0 (en) * 1997-03-28 1998-10-30 Pfizer NK-1 receptor antagonists for the treatment of delayed emesis
NZ329807A (en) * 1997-04-23 2000-07-28 Pfizer NK-1 receptor antagonists and P receptor antagonists 2-Diarylmethyl-3-amino-1-azabicyclo[2.2.2]octane derivatives and amino substituted N-containing rings as agents for treating irritable bowel syndrome
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US6255320B1 (en) * 1999-06-01 2001-07-03 Pfizer Inc. Polymorphs of a crystalline azo-bicyclo (2,2,2) octan-3-amine citrate and their pharmaceutical compositions
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Also Published As

Publication number Publication date
CN1048492C (zh) 2000-01-19
ES2084361T3 (es) 1996-05-01
US5939433A (en) 1999-08-17
JP2645225B2 (ja) 1997-08-25
ZA923942B (en) 1993-11-29
HUT70151A (en) 1995-09-28
HU217548B (hu) 2000-02-28
IS1611B (is) 1996-10-18
GT199200028A (es) 1993-11-20
US6222038B1 (en) 2001-04-24
US5807867A (en) 1998-09-15
IS3871A (is) 1992-12-02
DE69208877T2 (de) 1996-07-25
AP299A (en) 1994-01-14
PT100546B (pt) 1999-12-31
PT100546A (pt) 1993-08-31
IE921729A1 (en) 1992-12-02
IE72473B1 (en) 1997-04-23
YU56492A (sh) 1995-03-27
JPH06504292A (ja) 1994-05-19
LU91293I2 (fr) 2007-02-06
OA09867A (en) 1994-08-15
NL300250I2 (nl) 2007-03-01
RO110499B1 (ro) 1996-01-30
KR100214905B1 (ko) 1999-08-02
FI935297A0 (fi) 1993-11-29
GR3019687T3 (en) 1996-07-31
MX9202554A (es) 1992-11-01
NL300250I1 (nl) 2007-02-01
CZ281403B6 (cs) 1996-09-11
RU2103269C1 (ru) 1998-01-27
IL102008A (en) 1995-12-08
PL171379B1 (en) 1997-04-30
ATE135006T1 (de) 1996-03-15
DE122006000066I2 (de) 2007-12-06
UY23422A1 (es) 1992-11-12
NO2007003I2 (no) 2011-04-18
DE9290063U1 (de) 1994-02-24
EP0587723A1 (en) 1994-03-23
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FI935297L (fi) 1993-11-29
YU48995B (sh) 2003-04-30
WO1992021677A1 (en) 1992-12-10
JPH07285965A (ja) 1995-10-31
DE69208877D1 (de) 1996-04-11
FI114475B (fi) 2004-10-29
NZ242956A (en) 1995-06-27
BR9206073A (pt) 1994-12-06
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AU657552B2 (en) 1995-03-16
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BG98248A (bg) 1994-07-29
NO302701B1 (no) 1998-04-14
MA22539A1 (fr) 1992-12-31
JPH0733386B2 (ja) 1995-04-12
AP9200384A0 (en) 1992-07-31
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NO934312L (no) 1993-11-29
CN1067428A (zh) 1992-12-30
AU1990192A (en) 1993-01-08
CZ390692A3 (en) 1994-02-16
NZ270673A (en) 1997-07-27
EP0587723B1 (en) 1996-03-06
NO2007003I1 (no) 2007-03-26
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DK0587723T3 (da) 1996-04-01
UA27776C2 (uk) 2000-10-16

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