BG107652A - Алфа-арил етаноламини и използването им като бета-3 адренергични рецепторни агонисти - Google Patents

Алфа-арил етаноламини и използването им като бета-3 адренергични рецепторни агонисти

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Publication number
BG107652A
BG107652A BG107652A BG10765203A BG107652A BG 107652 A BG107652 A BG 107652A BG 107652 A BG107652 A BG 107652A BG 10765203 A BG10765203 A BG 10765203A BG 107652 A BG107652 A BG 107652A
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BG
Bulgaria
Prior art keywords
prodrugs
stereoisomers
compounds
receptor agonists
adrenergic receptor
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Application number
BG107652A
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English (en)
Inventor
Robert Day
Jennifer LAFONTAINE
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Pfizer Products Inc.
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Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG107652A publication Critical patent/BG107652A/bg

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
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  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Neurosurgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
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  • Endocrinology (AREA)
  • AIDS & HIV (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
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  • Molecular Biology (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Child & Adolescent Psychology (AREA)
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Abstract

Изобретението се отнася до бета-3 адренергични рецепторни агонисти със структурна формула@@в която Ar e пиридил, оксазолил, тиазолил или фенил; R5 е 5- или 6-членен хетероцикъл; Х е директна връзка или кислород и Y е директна връзка, алкилен, OCH2, CH2O или кислород. Изобретението се отнася до техни стереоизомери и пролекарствени средства, до фармацевтично приемливи соли на съединенията, стереоизомерите и пролекарствените средства, както и до междинни съединения, които се използват за получаване на съединенията с формула I и техни комбинации,до техни стереоизомери и пролекарствени средства и до фармацевтично приемливи соли на съединенията,стереоизомерите и пролекарствените средства.
BG107652A 2000-10-20 2003-03-20 Алфа-арил етаноламини и използването им като бета-3 адренергични рецепторни агонисти BG107652A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24227400P 2000-10-20 2000-10-20
PCT/IB2001/001847 WO2002032897A1 (en) 2000-10-20 2001-10-04 Alpha-aryl ethanolamines and their use as beta-3 adrenergic receptor agonists

Publications (1)

Publication Number Publication Date
BG107652A true BG107652A (bg) 2003-11-28

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Country Status (34)

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US (2) US6566377B2 (bg)
EP (1) EP1326861A1 (bg)
JP (1) JP2004511555A (bg)
KR (1) KR20030044013A (bg)
CN (1) CN1469876A (bg)
AP (1) AP2001002307A0 (bg)
AR (1) AR035716A1 (bg)
AU (1) AU2001292161A1 (bg)
BG (1) BG107652A (bg)
BR (1) BR0114836A (bg)
CA (1) CA2423792A1 (bg)
CR (1) CR6935A (bg)
CZ (1) CZ20031012A3 (bg)
DO (1) DOP2001000270A (bg)
EA (1) EA200300305A1 (bg)
EC (1) ECSP034562A (bg)
EE (1) EE200300191A (bg)
GT (1) GT200100210A (bg)
HR (1) HRP20030297A2 (bg)
HU (1) HUP0301382A2 (bg)
IL (1) IL154911A0 (bg)
IS (1) IS6748A (bg)
MA (1) MA26954A1 (bg)
MX (1) MXPA03003455A (bg)
NO (1) NO20031573L (bg)
PA (1) PA8530401A1 (bg)
PE (1) PE20020541A1 (bg)
PL (1) PL362076A1 (bg)
SK (1) SK4612003A3 (bg)
SV (1) SV2003000697A (bg)
TN (1) TNSN01148A1 (bg)
UY (1) UY26974A1 (bg)
WO (1) WO2002032897A1 (bg)
ZA (1) ZA200302191B (bg)

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