BG107604A - Тартаратна сол на тиазолидиндионово производно - Google Patents

Тартаратна сол на тиазолидиндионово производно Download PDF

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Publication number
BG107604A
BG107604A BG107604A BG10760403A BG107604A BG 107604 A BG107604 A BG 107604A BG 107604 A BG107604 A BG 107604A BG 10760403 A BG10760403 A BG 10760403A BG 107604 A BG107604 A BG 107604A
Authority
BG
Bulgaria
Prior art keywords
tartrate
solvate
accordance
compound according
pyridyl
Prior art date
Application number
BG107604A
Other languages
Bulgarian (bg)
English (en)
Inventor
Andrew Craig
Tim HO
Original Assignee
Smithkline Beecham P.L.C.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham P.L.C. filed Critical Smithkline Beecham P.L.C.
Publication of BG107604A publication Critical patent/BG107604A/bg

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/08Antibacterial agents for leprosy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
BG107604A 2000-08-04 2003-02-28 Тартаратна сол на тиазолидиндионово производно BG107604A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0019224.5A GB0019224D0 (en) 2000-08-04 2000-08-04 Novel pharmaceutical
PCT/GB2001/003511 WO2002012232A1 (en) 2000-08-04 2001-08-03 Tartrate salt of thiazolidinedione derivative

Publications (1)

Publication Number Publication Date
BG107604A true BG107604A (bg) 2003-09-30

Family

ID=9897026

Family Applications (1)

Application Number Title Priority Date Filing Date
BG107604A BG107604A (bg) 2000-08-04 2003-02-28 Тартаратна сол на тиазолидиндионово производно

Country Status (37)

Country Link
US (1) US20040014790A1 (da)
EP (1) EP1305311B1 (da)
JP (1) JP2004505970A (da)
KR (1) KR100755174B1 (da)
CN (1) CN1455778A (da)
AP (1) AP1785A (da)
AT (1) ATE384059T1 (da)
AU (1) AU2001276506A1 (da)
BG (1) BG107604A (da)
BR (1) BR0112982A (da)
CA (1) CA2417827A1 (da)
CY (1) CY1107252T1 (da)
CZ (1) CZ2003313A3 (da)
DE (1) DE60132461T2 (da)
DK (1) DK1305311T3 (da)
DZ (1) DZ3418A1 (da)
EA (1) EA005408B1 (da)
EC (1) ECSP034467A (da)
ES (1) ES2296772T3 (da)
GB (1) GB0019224D0 (da)
HK (1) HK1057358A1 (da)
HR (1) HRP20030068B1 (da)
HU (1) HUP0300778A3 (da)
IL (2) IL154275A0 (da)
MA (1) MA25832A1 (da)
MX (1) MXPA03001085A (da)
NO (1) NO324596B1 (da)
NZ (1) NZ524030A (da)
OA (1) OA12354A (da)
PL (1) PL360662A1 (da)
PT (1) PT1305311E (da)
SI (1) SI1305311T1 (da)
SK (1) SK1462003A3 (da)
UA (1) UA76720C2 (da)
WO (1) WO2002012232A1 (da)
YU (1) YU14603A (da)
ZA (1) ZA200300961B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE39384E1 (en) 1993-09-01 2006-11-07 Smithkline Beecham P.L.C. Substituted thiazolidinedione derivatives
DE102005034406A1 (de) * 2005-07-22 2007-02-01 Ratiopharm Gmbh Neue Salze von Rosiglitazon
US7435741B2 (en) * 2006-05-09 2008-10-14 Teva Pharmaceutical Industries, Ltd. 2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
CN108348292B (zh) 2015-10-27 2021-04-27 纳诺帕斯技术有限公司 具有机械性导引的微针装置

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds

Also Published As

Publication number Publication date
ES2296772T3 (es) 2008-05-01
EA005408B1 (ru) 2005-02-24
PL360662A1 (en) 2004-09-20
DE60132461D1 (de) 2008-03-06
ZA200300961B (en) 2004-04-01
MXPA03001085A (es) 2003-05-27
HUP0300778A2 (hu) 2003-11-28
KR20030022355A (ko) 2003-03-15
IL154275A0 (en) 2003-09-17
HUP0300778A3 (en) 2005-04-28
SI1305311T1 (sl) 2008-04-30
YU14603A (sh) 2006-05-25
DK1305311T3 (da) 2008-05-19
MA25832A1 (fr) 2003-07-01
AP2003002736A0 (en) 2003-03-31
NZ524030A (en) 2004-07-30
GB0019224D0 (en) 2000-09-27
HRP20030068B1 (en) 2008-07-31
HRP20030068A2 (en) 2005-02-28
JP2004505970A (ja) 2004-02-26
BR0112982A (pt) 2003-08-26
KR100755174B1 (ko) 2007-09-03
NO20030530L (no) 2003-02-03
ECSP034467A (es) 2003-03-31
CY1107252T1 (el) 2012-11-21
DE60132461T2 (de) 2008-12-24
WO2002012232A1 (en) 2002-02-14
EA200300230A1 (ru) 2003-06-26
UA76720C2 (uk) 2006-09-15
NO324596B1 (no) 2007-11-26
DZ3418A1 (fr) 2002-02-14
EP1305311A1 (en) 2003-05-02
PT1305311E (pt) 2008-04-07
EP1305311B1 (en) 2008-01-16
OA12354A (en) 2004-03-19
HK1057358A1 (en) 2004-04-02
IL154275A (en) 2009-02-11
ATE384059T1 (de) 2008-02-15
CA2417827A1 (en) 2002-02-14
AU2001276506A1 (en) 2002-02-18
US20040014790A1 (en) 2004-01-22
CZ2003313A3 (cs) 2004-02-18
SK1462003A3 (en) 2004-06-08
NO20030530D0 (no) 2003-02-03
AP1785A (en) 2007-10-04
CN1455778A (zh) 2003-11-12

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