BG106734A - Pyrazolo[1,5-d][1,2,4]triazines for enhancing cognition - Google Patents
Pyrazolo[1,5-d][1,2,4]triazines for enhancing cognitionInfo
- Publication number
- BG106734A BG106734A BG106734A BG10673402A BG106734A BG 106734 A BG106734 A BG 106734A BG 106734 A BG106734 A BG 106734A BG 10673402 A BG10673402 A BG 10673402A BG 106734 A BG106734 A BG 106734A
- Authority
- BG
- Bulgaria
- Prior art keywords
- optionally substituted
- heteroaromatic ring
- alkyl
- compounds
- membered heteroaromatic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Psychiatry (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hospice & Palliative Care (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9927874.9A GB9927874D0 (en) | 1999-11-25 | 1999-11-25 | Therapeutic agents |
| GB0009602A GB0009602D0 (en) | 2000-04-18 | 2000-04-18 | Therapeutic agents |
| GB0018651A GB0018651D0 (en) | 2000-07-28 | 2000-07-28 | Therapeutic agents |
| PCT/GB2000/004450 WO2001038331A2 (en) | 1999-11-25 | 2000-11-22 | Pyrazolo[1,5-d][1,2,4]triazines for enhancing cognition |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG106734A true BG106734A (en) | 2003-02-28 |
Family
ID=27255677
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG106734A BG106734A (en) | 1999-11-25 | 2002-05-22 | Pyrazolo[1,5-d][1,2,4]triazines for enhancing cognition |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US6355638B1 (ru) |
| EP (1) | EP1235829A2 (ru) |
| JP (1) | JP2003514909A (ru) |
| KR (1) | KR20020053091A (ru) |
| CN (1) | CN1391574A (ru) |
| AU (1) | AU1533001A (ru) |
| BG (1) | BG106734A (ru) |
| BR (1) | BR0015126A (ru) |
| CA (1) | CA2391103A1 (ru) |
| CZ (1) | CZ20021813A3 (ru) |
| EA (1) | EA200200599A1 (ru) |
| EE (1) | EE200200260A (ru) |
| HK (1) | HK1046406A1 (ru) |
| HU (1) | HUP0203579A3 (ru) |
| IL (1) | IL149051A0 (ru) |
| MX (1) | MXPA02005233A (ru) |
| NO (1) | NO20022456L (ru) |
| PL (1) | PL355637A1 (ru) |
| SK (1) | SK8952002A3 (ru) |
| WO (1) | WO2001038331A2 (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0128499D0 (en) * | 2001-11-28 | 2002-01-23 | Merck Sharp & Dohme | Therapeutic agents |
| EP2298296A1 (en) * | 2009-08-25 | 2011-03-23 | CNRS Centre National De La Recherche Scientifique | Composition and method for treating cognitive impairments in down syndrome subjects |
| JP5911476B2 (ja) * | 2010-05-26 | 2016-04-27 | スノビオン プハルマセウトイカルス インコーポレイテッド | ヘテロアリール化合物及びその使用方法 |
| US20150374705A1 (en) * | 2012-02-14 | 2015-12-31 | Shanghai Institues for Biological Sciences | Substances for treatment or relief of pain |
| CN107344938B (zh) * | 2016-05-06 | 2022-05-06 | 上海赛默罗生物科技有限公司 | 吡唑-三嗪类衍生物、其制备方法、药物组合物和用途 |
| CN107344936B (zh) * | 2016-05-06 | 2022-06-03 | 上海赛默罗生物科技有限公司 | 三唑哒嗪类衍生物、其制备方法、药物组合物和用途 |
| MX2021015874A (es) * | 2019-06-19 | 2022-02-03 | Biomarin Pharm Inc | Inhibidores de glicolato oxidasa para el tratamiento de enfermedades. |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA002436B1 (ru) * | 1996-07-25 | 2002-04-25 | Мерк Шарп Энд Домэ Лимитед | Замещенные производные триазоло-пиридазина в качестве лигандов рецепторов гамк |
| GB9715977D0 (en) * | 1997-07-29 | 1997-10-01 | Merck Sharp & Dohme | Therapeutic agents |
| WO1999036423A1 (en) * | 1998-01-14 | 1999-07-22 | Merck Sharp & Dohme Limited | Triazolo-pyridazine derivatives as ligands for gaba receptors |
| GB9806102D0 (en) * | 1998-03-20 | 1998-05-20 | Merck Sharp & Dohme | Therapeutic agents |
| AU755855B2 (en) * | 1998-06-16 | 2002-12-19 | Merck Sharp & Dohme Limited | Triazolo-pyridine derivatives as ligands for GABA receptors |
| ES2291043T3 (es) * | 1998-10-16 | 2008-02-16 | MERCK SHARP & DOHME LIMITED | Derivados de pirazolotriazina como ligandos para receptores de gaba. |
-
2000
- 2000-11-21 US US09/717,423 patent/US6355638B1/en not_active Expired - Lifetime
- 2000-11-22 KR KR1020027006672A patent/KR20020053091A/ko not_active Application Discontinuation
- 2000-11-22 IL IL14905100A patent/IL149051A0/xx unknown
- 2000-11-22 SK SK895-2002A patent/SK8952002A3/sk unknown
- 2000-11-22 MX MXPA02005233A patent/MXPA02005233A/es not_active Application Discontinuation
- 2000-11-22 EA EA200200599A patent/EA200200599A1/ru unknown
- 2000-11-22 BR BR0015126-2A patent/BR0015126A/pt not_active Application Discontinuation
- 2000-11-22 WO PCT/GB2000/004450 patent/WO2001038331A2/en not_active Application Discontinuation
- 2000-11-22 EP EP00977692A patent/EP1235829A2/en not_active Withdrawn
- 2000-11-22 AU AU15330/01A patent/AU1533001A/en not_active Abandoned
- 2000-11-22 HU HU0203579A patent/HUP0203579A3/hu unknown
- 2000-11-22 JP JP2001540094A patent/JP2003514909A/ja not_active Withdrawn
- 2000-11-22 CZ CZ20021813A patent/CZ20021813A3/cs unknown
- 2000-11-22 CN CN00816013A patent/CN1391574A/zh active Pending
- 2000-11-22 CA CA002391103A patent/CA2391103A1/en not_active Abandoned
- 2000-11-22 PL PL00355637A patent/PL355637A1/xx not_active Application Discontinuation
- 2000-11-22 EE EEP200200260A patent/EE200200260A/xx unknown
-
2002
- 2002-05-22 BG BG106734A patent/BG106734A/xx unknown
- 2002-05-24 NO NO20022456A patent/NO20022456L/no not_active Application Discontinuation
- 2002-10-29 HK HK02107821.8A patent/HK1046406A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2003514909A (ja) | 2003-04-22 |
| EE200200260A (et) | 2003-06-16 |
| KR20020053091A (ko) | 2002-07-04 |
| US6355638B1 (en) | 2002-03-12 |
| IL149051A0 (en) | 2002-11-10 |
| HUP0203579A3 (en) | 2003-07-28 |
| CA2391103A1 (en) | 2001-05-31 |
| NO20022456D0 (no) | 2002-05-24 |
| EA200200599A1 (ru) | 2002-12-26 |
| PL355637A1 (en) | 2004-05-04 |
| EP1235829A2 (en) | 2002-09-04 |
| CZ20021813A3 (cs) | 2002-08-14 |
| HK1046406A1 (zh) | 2003-01-10 |
| AU1533001A (en) | 2001-06-04 |
| BR0015126A (pt) | 2002-07-02 |
| MXPA02005233A (es) | 2002-11-07 |
| NO20022456L (no) | 2002-05-24 |
| SK8952002A3 (en) | 2002-10-08 |
| HUP0203579A2 (hu) | 2003-03-28 |
| WO2001038331A2 (en) | 2001-05-31 |
| WO2001038331A3 (en) | 2001-11-08 |
| CN1391574A (zh) | 2003-01-15 |
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