BG106173A - Халогенови производни на 9-дезоксо-9а-аза-9а-хомеритромицин а - Google Patents

Халогенови производни на 9-дезоксо-9а-аза-9а-хомеритромицин а Download PDF

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Publication number
BG106173A
BG106173A BG106173A BG10617301A BG106173A BG 106173 A BG106173 A BG 106173A BG 106173 A BG106173 A BG 106173A BG 10617301 A BG10617301 A BG 10617301A BG 106173 A BG106173 A BG 106173A
Authority
BG
Bulgaria
Prior art keywords
meaning
oxygen
compound according
same
sulfur
Prior art date
Application number
BG106173A
Other languages
Bulgarian (bg)
English (en)
Inventor
Zorica Marusic-Istuk
Nedjelko Kujundzic
Gabrijela Kobrehel
Stjepan Mutak
Natasa Marsic
Original Assignee
Pliva-Istrazivacki Institut D.O.O.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva-Istrazivacki Institut D.O.O. filed Critical Pliva-Istrazivacki Institut D.O.O.
Publication of BG106173A publication Critical patent/BG106173A/bg

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BG106173A 1999-05-03 2001-12-03 Халогенови производни на 9-дезоксо-9а-аза-9а-хомеритромицин а BG106173A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HR990130A HRP990130B1 (en) 1999-05-03 1999-05-03 HALOGEN DERIVATIVES 9a-N-(N'-ARYLCARBAMOYL)- AND 9a-N-(N'-ARYLTHIOCARBAMOYL)-9-DEOXO-9a-AZA-9a OF HOMOERYTHROMYCIN A
PCT/HR2000/000013 WO2000066603A1 (en) 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a

Publications (1)

Publication Number Publication Date
BG106173A true BG106173A (bg) 2002-07-31

Family

ID=10946916

Family Applications (1)

Application Number Title Priority Date Filing Date
BG106173A BG106173A (bg) 1999-05-03 2001-12-03 Халогенови производни на 9-дезоксо-9а-аза-9а-хомеритромицин а

Country Status (33)

Country Link
US (1) US6872707B1 (pt)
EP (1) EP1175429B1 (pt)
JP (1) JP2002543213A (pt)
KR (1) KR100714740B1 (pt)
CN (1) CN1140535C (pt)
AT (1) ATE244258T1 (pt)
AU (1) AU767681B2 (pt)
BG (1) BG106173A (pt)
BR (1) BR0010231A (pt)
CA (1) CA2372977A1 (pt)
CZ (1) CZ20013913A3 (pt)
DE (1) DE60003671T2 (pt)
DK (1) DK1175429T3 (pt)
EA (1) EA005214B1 (pt)
EE (1) EE05007B1 (pt)
ES (1) ES2202107T3 (pt)
GE (1) GEP20032928B (pt)
HK (1) HK1045522B (pt)
HR (1) HRP990130B1 (pt)
HU (1) HUP0201146A3 (pt)
IL (2) IL145986A0 (pt)
IS (1) IS6115A (pt)
MX (1) MXPA01011038A (pt)
NO (1) NO320138B1 (pt)
NZ (1) NZ515278A (pt)
PL (1) PL351402A1 (pt)
PT (1) PT1175429E (pt)
SI (1) SI1175429T1 (pt)
SK (1) SK284513B6 (pt)
TR (1) TR200103143T2 (pt)
UA (1) UA71962C2 (pt)
WO (1) WO2000066603A1 (pt)
ZA (1) ZA200108484B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010146B1 (en) * 2001-02-28 2005-10-31 Pliva D.D. 9a-N-(N'-(PHENYLSULFONYL)CARBAMOYL) DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMYCIN A AND OF 5-O-DESOSAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHRONOLIDE A
HRP20020886A2 (en) * 2002-11-11 2005-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. SUBSTITUTED 9a-N-[N'-(BENZENSULFONYL)CARBAMOYL-γ-AMINOPROPYL) AND 9a-N(N' -(?-CYANOETHIL)-N' -(b
HRP20020885B1 (en) 2002-11-11 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A
HRP20020991A2 (en) * 2002-12-12 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de
HRP20030381B1 (en) * 2003-05-14 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. 3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
ATE429921T1 (de) * 2005-01-14 2009-05-15 Glaxosmithkline Zagreb 9a-carbamoyl- und thiocarbamoylazalide mit antimalariawirkung
US20090118506A1 (en) * 2007-09-17 2009-05-07 In Jong Kim 6,11-bridged biaryl macrolides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU43116B (en) * 1979-04-02 1989-04-30 Pliva Pharm & Chem Works Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
WO1992006991A1 (fr) * 1990-10-15 1992-04-30 Taisho Pharmaceutical Co., Ltd. Erythromycine modifiee en 2' ou derive de cette substance
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A

Also Published As

Publication number Publication date
ZA200108484B (en) 2003-03-26
BR0010231A (pt) 2002-02-19
SK15702001A3 (sk) 2002-04-04
IL145986A0 (en) 2002-07-25
TR200103143T2 (tr) 2002-04-22
CN1140535C (zh) 2004-03-03
HK1045522A1 (en) 2002-11-29
HUP0201146A3 (en) 2003-03-28
DK1175429T3 (da) 2003-10-20
HK1045522B (zh) 2004-08-20
KR20020007397A (ko) 2002-01-26
WO2000066603A1 (en) 2000-11-09
NO20015346L (no) 2001-11-01
SI1175429T1 (en) 2003-12-31
JP2002543213A (ja) 2002-12-17
PT1175429E (pt) 2003-11-28
KR100714740B1 (ko) 2007-05-07
EP1175429B1 (en) 2003-07-02
ATE244258T1 (de) 2003-07-15
EA005214B1 (ru) 2004-12-30
US6872707B1 (en) 2005-03-29
NZ515278A (en) 2003-06-30
GEP20032928B (en) 2003-03-25
HRP990130A2 (en) 2001-10-31
DE60003671T2 (de) 2004-06-17
UA71962C2 (en) 2005-01-17
DE60003671D1 (de) 2003-08-07
EE05007B1 (et) 2008-04-15
EE200100582A (et) 2003-02-17
AU4135000A (en) 2000-11-17
IS6115A (is) 2001-10-19
HUP0201146A2 (hu) 2002-07-29
PL351402A1 (en) 2003-04-07
AU767681B2 (en) 2003-11-20
EP1175429A1 (en) 2002-01-30
NO320138B1 (no) 2005-10-31
NO20015346D0 (no) 2001-11-01
HRP990130B1 (en) 2004-06-30
MXPA01011038A (es) 2002-07-22
EA200101170A1 (ru) 2002-04-25
IL145986A (en) 2006-10-31
CZ20013913A3 (cs) 2002-04-17
CN1351606A (zh) 2002-05-29
SK284513B6 (sk) 2005-05-05
ES2202107T3 (es) 2004-04-01
CA2372977A1 (en) 2000-11-09

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