BE882703A - Nouveaux derives de omega-(4-diphenylmethyl-piperidino)-1-phenylalcanols et leur procede de preparation. - Google Patents
Nouveaux derives de omega-(4-diphenylmethyl-piperidino)-1-phenylalcanols et leur procede de preparation.Info
- Publication number
- BE882703A BE882703A BE0/200161A BE200161A BE882703A BE 882703 A BE882703 A BE 882703A BE 0/200161 A BE0/200161 A BE 0/200161A BE 200161 A BE200161 A BE 200161A BE 882703 A BE882703 A BE 882703A
- Authority
- BE
- Belgium
- Prior art keywords
- phenylalcanols
- diphenylmethyl
- piperidino
- derivatives
- preparation process
- Prior art date
Links
- -1 4-DIPHENYLMETHYL-PIPERIDINO Chemical class 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/028,813 US4254129A (en) | 1979-04-10 | 1979-04-10 | Piperidine derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE882703A true BE882703A (fr) | 1980-07-31 |
Family
ID=21845568
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/200161A BE882703A (fr) | 1979-04-10 | 1980-04-09 | Nouveaux derives de omega-(4-diphenylmethyl-piperidino)-1-phenylalcanols et leur procede de preparation. |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US4254129A (esLanguage) |
| JP (1) | JPS55141469A (esLanguage) |
| AT (1) | AT376208B (esLanguage) |
| AU (1) | AU531146B2 (esLanguage) |
| BE (1) | BE882703A (esLanguage) |
| CA (1) | CA1123438A (esLanguage) |
| CH (1) | CH643245A5 (esLanguage) |
| DE (1) | DE3007498A1 (esLanguage) |
| DK (1) | DK153709C (esLanguage) |
| ES (1) | ES8103735A1 (esLanguage) |
| FR (1) | FR2453854A1 (esLanguage) |
| IL (1) | IL59158A (esLanguage) |
| IT (1) | IT1143960B (esLanguage) |
| NL (2) | NL190580C (esLanguage) |
| NO (2) | NO154521C (esLanguage) |
| NZ (1) | NZ192653A (esLanguage) |
| PH (1) | PH17023A (esLanguage) |
| SE (1) | SE448726B (esLanguage) |
| ZA (1) | ZA80332B (esLanguage) |
Families Citing this family (117)
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| CN102659667B (zh) * | 2012-04-20 | 2013-08-14 | 浙江启明药业有限公司 | 一种非索非那定关键中间体的合成方法 |
| CN103333100B (zh) * | 2013-06-06 | 2016-04-06 | 池州东升药业有限公司 | 一种盐酸非索非那定的合成工艺 |
| ITMI20131652A1 (it) | 2013-10-07 | 2015-04-08 | Dipharma Francis Srl | Procedimento per la purificazione di derivati dell'acido 2-fenil-2-metil-propanoico |
| CN104557671B (zh) * | 2013-10-10 | 2018-04-13 | 池州东升药业有限公司 | 一种非索非那定及中间体的合成方法 |
| EP2949321A1 (en) | 2014-05-26 | 2015-12-02 | Sanovel Ilac Sanayi ve Ticaret A.S. | Multilayer formulations of fexofenadine and montelukast |
| CN107428678B (zh) | 2015-01-22 | 2021-01-01 | 赛诺菲-安万特德国有限公司 | 用于制备2-[4-(环丙烷羰基)苯基]-2-甲基-丙腈的方法 |
| HRP20200106T1 (hr) | 2015-10-22 | 2020-04-03 | Sanofi-Aventis Deutschland Gmbh | Postupak za pripravu feksofenadina i međuprodukata koji se u njemu koriste |
| GB2629127A (en) | 2022-08-31 | 2024-10-23 | Novumgen Ltd | An orodispersible tablet of fexofenadine and its process of preparation |
| KR20250133597A (ko) | 2023-01-20 | 2025-09-08 | 오펠라 헬스케어 그룹 에스에이에스 | 파라벤 프리 펙소페나딘 제제 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
| ZA728544B (en) * | 1972-01-28 | 1974-02-27 | Richardson Merrell Inc | Alpha-aryl-4-substituted piperidinoalkanol derivatives |
| US3878217A (en) * | 1972-01-28 | 1975-04-15 | Richardson Merrell Inc | Alpha-aryl-4-substituted piperidinoalkanol derivatives |
| US3806526A (en) * | 1972-01-28 | 1974-04-23 | Richardson Merrell Inc | 1-aroylalkyl-4-diphenylmethyl piperidines |
| BE794596A (fr) * | 1972-01-28 | 1973-05-16 | Richardson Merrell Inc | Piperidinoalcanone-oximes substituees et leur procede de preparation |
| BE794598A (fr) * | 1972-01-28 | 1973-05-16 | Richardson Merrell Inc | Nouveaux derives olefiniques de piperidines substituees en 4 et leur procede de preparation |
| US3965257A (en) * | 1972-01-28 | 1976-06-22 | Richardson-Merrell Inc. | Compositions and methods for the treatment of the symptoms of histamine induced allergic reactions |
| US3941795A (en) * | 1974-02-08 | 1976-03-02 | Richardson-Merrell Inc. | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
| US3931197A (en) * | 1974-02-08 | 1976-01-06 | Richardson-Merrell Inc. | Substituted piperidine derivatives |
| US3946022A (en) * | 1974-03-04 | 1976-03-23 | Richardson-Merrell Inc. | Piperidine derivatives |
| US3956296A (en) * | 1974-12-11 | 1976-05-11 | A. H. Robins Company, Incorporated | 1-Substituted-4-benzylpiperidines |
| US3922276A (en) * | 1974-12-11 | 1975-11-25 | Robins Co Inc A H | 1-Substituted-4-benzylidenepiperidines |
-
1979
- 1979-04-10 US US06/028,813 patent/US4254129A/en not_active Expired - Lifetime
-
1980
- 1980-01-18 CA CA344,020A patent/CA1123438A/en not_active Expired
- 1980-01-18 NZ NZ192653A patent/NZ192653A/xx unknown
- 1980-01-18 IL IL59158A patent/IL59158A/xx unknown
- 1980-01-21 ZA ZA00800332A patent/ZA80332B/xx unknown
- 1980-01-29 AU AU55016/80A patent/AU531146B2/en not_active Expired
- 1980-02-07 NL NL8000754A patent/NL190580C/xx not_active IP Right Cessation
- 1980-02-28 DE DE19803007498 patent/DE3007498A1/de active Granted
- 1980-03-05 CH CH174180A patent/CH643245A5/de not_active IP Right Cessation
- 1980-03-17 AT AT0144880A patent/AT376208B/de not_active IP Right Cessation
- 1980-03-24 IT IT48245/80A patent/IT1143960B/it active Protection Beyond IP Right Term
- 1980-03-26 ES ES489934A patent/ES8103735A1/es not_active Expired
- 1980-03-27 DK DK132980A patent/DK153709C/da not_active IP Right Cessation
- 1980-03-28 PH PH23831A patent/PH17023A/en unknown
- 1980-04-08 SE SE8002634A patent/SE448726B/sv not_active IP Right Cessation
- 1980-04-09 BE BE0/200161A patent/BE882703A/fr not_active IP Right Cessation
- 1980-04-09 JP JP4577180A patent/JPS55141469A/ja active Granted
- 1980-04-09 FR FR8007992A patent/FR2453854A1/fr active Granted
- 1980-04-09 NO NO801014A patent/NO154521C/no unknown
-
1998
- 1998-04-08 NL NL980013C patent/NL980013I2/nl unknown
- 1998-05-29 NO NO1998017C patent/NO1998017I1/no unknown
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Free format text: 097C0100, EXPIRES: 20050409 |
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| RE20 | Patent expired |
Owner name: MERRELL PHARMACEUTICALS INC. Effective date: 20000409 |
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| CCRE | Expiry of a supplementary protection certificate |
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| CCRE | Expiry of a supplementary protection certificate |
Free format text: PRODUCT NAME: FEXOFENADINUM HYDROCHLORIDUM; NAT. REG. NO/DATE: 354 IS 355 F 3 19970414; FIRST REG.:GB PL 04425/0155 19960311 Spc suppl protection certif: 97C0100 Filing date: 19970902 Expiry date: 20000409 Extension date: 20050409 |