AU2017241530B2 - Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same - Google Patents

Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same Download PDF

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Publication number
AU2017241530B2
AU2017241530B2 AU2017241530A AU2017241530A AU2017241530B2 AU 2017241530 B2 AU2017241530 B2 AU 2017241530B2 AU 2017241530 A AU2017241530 A AU 2017241530A AU 2017241530 A AU2017241530 A AU 2017241530A AU 2017241530 B2 AU2017241530 B2 AU 2017241530B2
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Prior art keywords
formulation
disease
pirfenidone
fibrosis
amount
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Revoked
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AU2017241530A
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AU2017241530A1 (en
Inventor
Siddharthya Krishnachandan Mujumdar
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F Hoffmann La Roche AG
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F Hoffmann La Roche AG
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Publication of AU2017241530A1 publication Critical patent/AU2017241530A1/en
Priority to AU2022275529A priority Critical patent/AU2022275529A1/en
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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AU2017241530A 2016-03-29 2017-03-27 Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same Revoked AU2017241530B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2022275529A AU2022275529A1 (en) 2016-03-29 2022-11-25 Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same

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US201662314933P 2016-03-29 2016-03-29
US62/314,933 2016-03-29
PCT/US2017/024280 WO2017172602A1 (en) 2016-03-29 2017-03-27 Granulate formulation of 5-methy|-1-pheny|-2(1h)-pyridone and method of making the same

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AU2022275529A Division AU2022275529A1 (en) 2016-03-29 2022-11-25 Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same

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AU2017241530A1 AU2017241530A1 (en) 2018-10-04
AU2017241530B2 true AU2017241530B2 (en) 2022-12-15

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AU2017241530A Revoked AU2017241530B2 (en) 2016-03-29 2017-03-27 Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same
AU2022275529A Abandoned AU2022275529A1 (en) 2016-03-29 2022-11-25 Granulate formulation of 5-methyl-1-phenyl-2(1H)-pyridone and method of making the same

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US (2) US10188637B2 (https=)
EP (2) EP3435985B1 (https=)
JP (2) JP7456721B2 (https=)
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