AR107990A1 - Formulación granulada de 5-metil-1-fenil-2-(1h)-piridona y método para elaborarla - Google Patents

Formulación granulada de 5-metil-1-fenil-2-(1h)-piridona y método para elaborarla

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Publication number
AR107990A1
AR107990A1 ARP170100761A ARP170100761A AR107990A1 AR 107990 A1 AR107990 A1 AR 107990A1 AR P170100761 A ARP170100761 A AR P170100761A AR P170100761 A ARP170100761 A AR P170100761A AR 107990 A1 AR107990 A1 AR 107990A1
Authority
AR
Argentina
Prior art keywords
piridone
phenyl
prepare
methyl
granulated formulation
Prior art date
Application number
ARP170100761A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57575344&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR107990(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR107990A1 publication Critical patent/AR107990A1/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418—Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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Abstract

Formulaciones granuladas de pirfenidona y métodos para elaborar estas formulaciones. Reivindicación 89: Un método para tratar una afección fibrótica o inhibir las acciones de citocinas, que comprende administrar la formulación granulada de acuerdo con cualquiera de las reivindicaciones 1 a 35 a un paciente que tiene esa afección fibrótica o que tiene un trastorno mediado por citocinas.
ARP170100761A 2016-03-29 2017-03-28 Formulación granulada de 5-metil-1-fenil-2-(1h)-piridona y método para elaborarla AR107990A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662314933P 2016-03-29 2016-03-29

Publications (1)

Publication Number Publication Date
AR107990A1 true AR107990A1 (es) 2018-07-04

Family

ID=57575344

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170100761A AR107990A1 (es) 2016-03-29 2017-03-28 Formulación granulada de 5-metil-1-fenil-2-(1h)-piridona y método para elaborarla

Country Status (13)

Country Link
US (2) US10188637B2 (es)
EP (2) EP3895696B1 (es)
JP (2) JP7456721B2 (es)
KR (1) KR102552615B1 (es)
CN (2) CN108883072A (es)
AR (1) AR107990A1 (es)
AU (2) AU2017241530B2 (es)
CA (1) CA2937365C (es)
ES (1) ES2883595T3 (es)
IL (1) IL261745B2 (es)
MX (1) MX2018011819A (es)
PL (1) PL3435985T3 (es)
WO (1) WO2017172602A1 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20180100869A (ko) * 2017-03-02 2018-09-12 영진약품 주식회사 피르페니돈의 입자크기 조절에 따른 타정성이 개선된 약제학적 조성물 및 이의 제조방법
US11510877B2 (en) 2017-10-10 2022-11-29 Capsugel Belgium Nv Gelling multiparticulates
EP3494965B1 (en) * 2017-12-11 2021-06-02 Laurus Labs Limited An improved process for the preparation of pirfenidone
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MX2018011819A (es) 2019-07-04
EP3895696A1 (en) 2021-10-20
CA2937365C (en) 2018-09-18
EP3435985A1 (en) 2019-02-06
AU2017241530A1 (en) 2018-10-04
CN108883072A (zh) 2018-11-23
KR20180123067A (ko) 2018-11-14
EP3895696B1 (en) 2023-08-09
JP7456721B2 (ja) 2024-03-27
IL261745B2 (en) 2023-06-01
JP2019513145A (ja) 2019-05-23
CN114533688A (zh) 2022-05-27
AU2017241530B2 (en) 2022-12-15
EP3435985B1 (en) 2021-05-12
ES2883595T3 (es) 2021-12-09
US10188637B2 (en) 2019-01-29
CA2937365A1 (en) 2016-12-22
WO2017172602A1 (en) 2017-10-05
PL3435985T3 (pl) 2021-11-22

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